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Neurological Disease

货号 产品名 CAS号 信息
CSN16643 LY2979165 1311385-32-6 LY2979165 is a mGlu2 agonist, a drug candidate drug used to treat bipolar disorder.
CSN16651 2-((1-Benzylpiperidin-4-yl)methyl)-5,6-dimethoxy-2,3-dihydro-1H-inden-1-one 120014-06-4 Donepezil is a centrally acting reversible AchE inhibitor with IC50 of 8.12 nM and 11.6 nM for bAChE and hAChE, respectively, a medication used to treat Alzheimer's disease.
CSN16705 Dapoxetine HCl 129938-20-1 Dapoxetine HCl is an inhibitor of serotonin reuptake. It can treat premature ejaculation.
CSN16772 Phenytoin sodium 630-93-3 Phenytoin sodium is a stabilizer of inactive voltage-gated sodium channel.
CSN16779 7-((3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo[c,f][1,2]thiazepin-11-yl)amino)heptanoic acid 72797-41-2 Tianeptine is a unique tricyclic antidepressant, in contrast to SSRIs, which can increase serotonin uptake in the brain and reduce stress-induced atrophy of neuronal dendrites.
CSN16789 Dibucaine 85-79-0 Cinchocaine is amide type local anesthetic that is generally used for surface anesthesia.
CSN16795 Tetracaine 94-24-6 Tetracaine can interfer the entry of sodium ions into nerve cells and used as a topical local anesthetic.
CSN16796 3-(Aminocarbonyl)pyridine 98-92-0 Nicotinamide can act as an inhibitor of sirtuins and it is the active component of NAD and NADP.
CSN16886 Ramosetron HCl 132907-72-3 Ramosetron HCl is a potent and selective 5-HT3 receptor antagonist for the treatment of nausea and vomiting.
CSN16934 P7C3 301353-96-8 P7C3 is a brain-penetrant NAMPT activator with proneurogenic and neuroprotective effect.
CSN16786 Ethyl 8-fluoro-5-methyl-6-oxo-5,6-dihydro-4H-benzo[f]imidazo[1,5-a][1,4]diazepine-3-carboxylate 78755-81-4 Flumazenil is a non-selective antagonist of benzodiazepine towards α1, α2, α3 or α5-containing GABAA receptors.
CSN16682 Lomerizine 2HCl 101477-54-7 Lomerizine 2HCl is an L- and T-type calcium channel blocker used in the treatment of migraine.
CSN16737 Oxcarbazepine 28721-07-5 Oxcarbazepine is a voltage-gated sodium channel blocker with IC50 of 160 μM and it is used for the treatment of partial seizure.
CSN16724 Clomipramine HCl 17321-77-6 Clomipramine HCl is a dibenzazepine-derived 5-HT reuptake inhibitor and a tricyclic antidepressant.
CSN16709 Tetracaine HCl 136-47-0 Tetracaine HCl is a potent local anaesthetic and a channel function allosteric inhibitor.
CSN16627 VU0152100 409351-28-6 VU 0152100 is a potent and selective allosteric potentiator of M4 mAChR with an EC50 of 380 ± 93 nM.
CSN16622 JTC-801 244218-51-7 JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, and weakly inhibits receptors δ, κ, and μ.
CSN16855 (±)-Huperzine A 120786-18-7 (±)-Huperzine A is an active Lycopodium alkaloid extracted from traditional Chinese herbs of Lycopodium serratum, is a potent, selective and reversible acetylcholinesterase (AChE) inhibitor and has been widely used in China for the treatment of Alzheimer's disease (AD).
CSN16735 Nicergoline 27848-84-6 Nicergoline is a non-selective alpha-adrenergic receptor antagonist which can decrease vascular resistance and increase arterial blood flow in the brain, improving the utilization of oxygen and glucose by brain cells.
CSN16841 (7S,7aR,14S,14aS)-Tetradecahydro-7,14-methanodipyrido[1,2-a:1',2'-e][1,5]diazocine 90-39-1 (-)-Sparteine is a class 1a antiarrhythmic agent and a sodium channel blocker.
CSN16680 topride HCl 122892-31-3 Itopride HCl is a D2 antagonist and an AChE inhibitor with an IC50 value of 2.04±0.27 μM. It is a prokinetic benzamide derivative unlike domperidone.
CSN16775 Atracurium besylate 64228-81-5 Atracurium besylate is a non-depolarizing neuromuscular blocking agent with short duration of action.
CSN16653 Olanzapine 132539-06-1 Olanzapine is a multiple-target antagonist for 5-HT2A receptors and D2 dopamine receptors, as well as muscarinic M3 receptor.
CSN16711 Agomelatine 138112-76-2 Agomelatine is a melatonin structurely similar 5-HT2C receptor antagonist as well as a potent melatonin receptor agonist, used to treat major depressive disorder.
CSN16669 Gabapentin HCl 60142-95-2 Gabapentin is a GABA analogue, used to treat seizures and neuropathic pain.
CSN16659 CTEP 871362-31-1 CTEP is a selective allosteric mGluR5 antagonist with IC50 value of 2.2 nM.
CSN16751 Intepirdine 607742-69-8 SB-742457 is a selective 5-HT6 receptor antagonist with Ki value of 1.4 nM, showing potential cognition, memory, and learning-enhancing effects.
CSN16715 Pancuronium dibromide 15500-66-0 Pancuronium dibromide is a competitive nAchR antagonist, causing skeletal muscle relaxation and paralysis through competitively binding to the nicotinic receptor at the neuromuscular junction.
CSN16726 Tegaserod maleate 189188-57-6 Tegaserod Maleate is a potent full agonist at 5-HT4 receptors with an EC50 value of 7 nM, used to treat irritable bowel syndrome associated with constipation and chronic constipation.
CSN16954 Xanomeline oxalate 141064-23-5 Xanomeline Oxalate is a selective M1 muscarinic receptor agonist.
CSN16914 Nav1.7 inhibitor 1355631-24-1 Nav1.7 inhibitor is a sulfonamide derivative with potent Nav1.7 inhibition activity.
CSN16747 2-(1H-Imidazol-4-yl)ethan-1-amine 51-45-6 Histamine is an organic nitrogenous compound involved in local immune responses as well as regulating physiological function in the gut and acting as a neurotransmitter.
CSN16753 LX-1031 945976-76-1 LX1031 is an oral, small molecule tryptophan 5-hydroxylase (TPH) inhibitor that reduces serotonin(5-HT) synthesis peripherally.
CSN16686 Ondansetron HCl 99614-01-4 Ondansetron is a serotonin 5-HT3 receptor antagonist used mainly as anantiemetic (to treat nausea and vomiting), often following chemotherapy.
CSN16969 Telotristat ethyl 1033805-22-9 LX1606 is an orally-delivered inhibitor of tryptophan hydroxylase that reduces serotonin production.
CSN16745 Adiphenine HCl 50-42-0 Adiphenine HCl is a nicotinic receptor inhibitor with IC50 of 15 μM, used as an antispasmodic drug.
CSN16693 Granisetron 109889-09-0 Granisetron is a serotonin 5-HT3 receptor antagonist used as an antiemetic to treat nausea and vomiting following chemotherapy.
CSN16865 NBI-98782 85081-18-1 NBI-98782 is a vesicular monoamine transporter (VMAT2) inhibtior with an Ki value of 0.97 nM.
CSN16591 CP-809101 HCl 1215721-40-6 CP-809101 HCl is a potent and selective 5-HT2C receptor agonist with pEC50 of 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors respectively.
CSN16899 Phenelzine 51-71-8 Phenelzine is a non-selective and irreversible monoamine oxidase inhibitor (MAOI), used as an antidepressant and anxiolytic.
CSN16799 WAY-100635 162760-96-5 WAY-100635 is a potent and selective 5-hydroxytryptamine1A antagonist with an IC50 of 0.95 ± 0.12 nM for 5-HT.
CSN16857 QNZ46 1237744-13-6 QNZ46 is a noncompetitive and voltage-independent GluN2C/GluN2D-selective NMDA antagonist with IC50 values of 3, 6, 229 μM for GluN2D, GluN2C, GluN2A, respectively.
CSN16936 S1RA 878141-96-9 S1RA is a potent and selective sigma-1 receptor (σ1R, Ki=17 nM) antagonist, showed good selectivity against σ2R (Ki > 1000 nM).
CSN16798 GW791343 2HCl 1019779-04-4 GW791343 2HCl is a P2X7 allosteric modulator exhibiting species-specific activity and acts as a negative allosteric modulator of human P2X7 (pIC50 = 6.9 - 7.2).
CSN16688 Tamsulosin 106133-20-4 Tamsulosin is an α1 adrenergic receptor blocker used to treat symptomatic benign prostatic hyperplasia (BPH), chronic prostatitis, and to help with the passage of kidney stones.
CSN16826 SB-674042 483313-22-0 SB-674042 is a potent and selective non-peptide orexin OX1 receptor antagonist (Kd = 3.76 nM) exhibiting 100-fold selectivity for OX1 over OX2 receptors.
CSN16823 HC-030031 349085-38-7 HC-030031 is a blocker of TRPA1 channel that exhibits antagonistic effect on AITC- and formalin-evoked calcium influx with IC50 of 6.2 μM and 5.3 μM respectively.
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