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HSP

HSP

货号 产品名 CAS号 信息
CSN16304 XL888 1149705-71-4 XL888 is a specific and ATP-competitive Hsp90 inhibitor with IC50 of 24 nM.
CSN13596 VER-50589 747413-08-7 VER-50589 is an isoxazole compound that inhibits Hsp90 with an IC50 value of 21 nM.
CSN18335 VER-49009 558640-51-0 VER-49009 is a pyrazole compound that inhibits Hsp90 with an IC50 value of 47 nM.
CSN13116 VER-155008 1134156-31-2 VER-155008 is a potent Hsp70 family inhibitor with IC50 of 0.5 μM, 2.6 μM, and 2.6 μM in cell-free assays for HSP70, HSC70, and GRP78, respectively, > 100-fold selectivity over HSP90.
CSN20344 TRC051384 HCl 1333327-56-2 TRC051384 is an inducer of heat shock protein Hsp70. it reduces stroke-associated neuronal injury and increases survival in a rat model of transient ischemic stroke and activates heat shock factor-1 and results in elevated chaperone and anti-inflammatory activity.
CSN20345 TRC051384 867164-40-7 TRC051384 is a inducer of Hsp70.
CSN12051 Teprenone 6809-52-5 Teprenone is used as an anti-ulcer drug, a cardioprotective agent, a hepatoprotective agent, a nephroprotective agent, a neuroprotective agent and a Hsp70 inducer.
CSN22232 TAS-116 1260533-36-5 TAS-116 is a potent and selective HSP90α/β inhibitor with Kis of 34.7 nM, 21.3 nM, respectively.
CSN16517 SNX-2112 908112-43-6 SNX-2112 is a potent synthetic heat shock protein 90 (HSP90) inhibitor with an IC50 of 0.92 μM for K562 cells.
CSN18481 Retaspimycin 857402-23-4 Retaspimycin is a small-molecule inhibitor of heat shock protein 90 (HSP90) with antiproliferative and antineoplastic activities.
CSN18482 Retaspimycin HCl 857402-63-2 Retaspimycin HCl is the HCl salt of a small-molecule inhibitor of heat shock protein 90 (HSP90) with antiproliferative and antineoplastic activities.
CSN15760 PU-WS13 1454619-14-7 PU-WS13 is a potent, Grp94-specific Hsp90 inhibitor of the purine scaffold class.
CSN16046 PU-H 71 873436-91-0 PU-H71 is a potent Hsp90 inhibitor with IC50 of 50 nM.
CSN18943 PU-H 71 HCl 2095432-24-7 PU-H71 HCl is a potent Hsp90 inhibitor with IC50 of 50 nM.
CSN17514 PF-04929113 Mesylate 1173111-67-5 PF-04929113 mesylate is a potent and selective Hsp90 inhibitor with an IC50 of median 50 nM.
CSN16541 PF-04929113 908115-27-5 PF-04929113 is a potent and selective HSP90 inhibitor with Kd of 41 nM and induces Her-2 degradation with IC50 of 37 nM.
CSN15852 HSP990 934343-74-5 NVP-HSP990 is a potent and selective HSP90 inhibitor for HSP90α/β with IC50 of 0.6 nM/0.8 nM.
CSN17190 NVP-BEP800 847559-80-2 NVP-BEP800 is a fully synthetic HSP90β inhibitor with IC50 of 58 nM, exhibits> 70-fold selectivity against Hsp90 family members Grp94 and Trap-1.
CSN16765 NMS-E973 1253584-84-7 NMS-E973 is a potent and selective Hsp90 inhibitor with DC50 of < 10 nM for Hsp90 binding, no activiy against a panel of 52 diverse protein kinases.
CSN17387 ML346 100872-83-1 ML346 is an activator of Hsp70 with EC50 of 4600 nM in HeLa cell toxicity assay.
CSN21425 MKT-077 147366-41-4 MKT-077 (FJ-776) is a water-soluble rhodacyanine dye with antitumor activity. It can bind to Hsp70 family member mortalin-2 and inhibit its interactions with p53.
CSN22959 Macbecin I 73341-72-7 Macbecin I is a Hsp90 inhibitor with IC50 of 2 μM.
CSN16562 KW-2478 819812-04-9 KW-2478 is a nonansamycin HSP90 inhibitor with IC50 of 3.8 nM.
CSN18942 KRIBB11 342639-96-7 KRIBB11 is an inhibitor of heat shock factor (HSF) inhibitor, with IC50 of 1.2 μM.
CSN17321 KNK437 218924-25-5 KNK437 is a pan-HSP inhibitor, which inhibits the synthesis of inducible HSPs, including HSP105, HSP72, and HSP40.
CSN24783 Grp94 Inhibitor-1   2234897-35-7 Grp94 Inhibitor-1 is a potent, selective Grp94 inhibitor with an IC50 value of 2 nM, and over 1000-fold selectivity to Grp94 against Hsp90α[1].
CSN11085 Geldanamycin 30562-34-6 Geldanamycin is a natural existing HSP90 inhibitor with Kd of 1.2 μM.
CSN22828 Gedunin 2753-30-2 Gedunin is a Hsp90 inhibitor and exhibits anticancer and antimalarial activity.
CSN15732 Ganetespib 888216-25-9 Ganetespib is a unique triazolone-containing Hsp90 inhibitor with an IC50 of 4 nM in OSA 8 cells.
CSN13554 Eupalinolide B 877822-41-8 Eupalinolide A is a natural product isolated and purified from the herbs of Eupatorium lindleyanum DC.
CSN12347 Elesclomol 488832-69-5 Elesclomol, an inhibitor of HSP90, is a potent oxidative stress inducer that elicits pro-apoptosis events among tumor cells.
CSN22799 EC 144 911397-80-3 EC 144 is a high affinity, potent and selective Hsp90 inhibitor with Ki of 0.2 nM and IC50 of 1.1 nM.
CSN18944 Debio 0932 1061318-81-7 Debio 0932 is a heat shock protein 90 (HSP90) inhibitor with strong affinity for HSP90 alpha/beta, high oral bioavailability and potent anti-proliferative activity against a broad range of cancer cell lines (with a mean IC50 of 220 nmol/L).
CSN27185 Col003   328565-16-8 Col003 is a cell penetrant, selective and potent inhibitor of the interaction of Hsp47 with collagen. Col003 is the cleavage product of AK778.It competitively inhibited the interaction and caused the inhibition of collagen secretion by destabilizing the collagen triple helix.
CSN19190 CH5138303 959763-06-5 CH5138303 is an orally available Hsp90 inhibitor with Kd of 0.48 nM.
CSN22743 CCT 018159 171009-07-7 CCT 018159 is a novel inhibitor of heat shock protein 90 (Hsp90) ATPase activity with IC50 of 5.7 μM.
CSN13441 BIIB021 848695-25-0 BIIB021 is an orally available, fully synthetic small-molecule inhibitor of HSP90 with Ki and EC50 of 1.7 nM and 38 nM, respectively.
CSN12421 Luminespib 747412-49-3 AUY922 is a highly potent HSP90 inhibitor for HSP90α/β with IC50 of 13 nM /21 nM, weaker potency against the HSP90 family members GRP94 and TRAP-1.
CSN16920 Onalespib 912999-49-6 AT13387 is a selective potent Hsp90 inhibitor with IC50 of 18 nM in A375 cells, displays a long duration of anti-tumor activity.
CSN18941 Apoptozole 1054543-47-3 Apoptozole is an inhibitor of heat shock protein 70 (HSP70) and Hsc70. It induces caspase-dependent apoptosis.
CSN16172 Alvespimycin 467214-20-6 Alvespimycin is a potent, water-soluble HSP90 inhibitor with IC50 of 62 nM.
CSN18284 Alvespimycin HCl 467214-21-7 Alvespimycin HCl is a potent, water-soluble HSP90 inhibitor with IC50 of 62 nM.
CSN17209 17-AAG 75747-14-7 17-AAG is a potent HSP90 inhibitor with IC50 of 5 nM, having a 100-fold higher binding affinity for HSP90 derived from tumour cells than HSP90 from normal cells.
CSN18562 17-AAG HCl 911710-03-7 17-AAG HCl is a potent HSP90 inhibitor with IC50 of 5 nM, having a 100-fold higher binding affinity for HSP90 derived from tumour cells than HSP90 from normal cells.
CSN25416 Ethoxyquin 91-53-2
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