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Opioid Receptor

Opioid Receptor

货号 产品名 CAS号 信息
CSN18678 [D-Ala2]Leucine-Enkephalin 64963-01-5 [D-Ala2]Leucine-Enkephalin is a potent, long-acting Leu-enkephalin analog agonist of delta opioid receptor.
CSN20210 TRV0109101 1401027-29-9 TRV0109101, a G protein-biased agonist of the µ-opioid receptor, which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia.
CSN20211 TRV0109101 HCl 2101210-22-2 TRV0109101 hydrochloride, a G protein-biased agonist of the µ-opioid receptor, which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia.
CSN17789 TRV 130 Racemate 1401028-25-8 TRV 130 racemate is the racemate form of TRV130, which a μ-opioid receptor (MOR) G protein-biased ligand.
CSN17788 TRV 130 1401028-24-7 TRV 130 is a μ-opioid receptor (MOR) G protein-biased ligand and elicits robust G protein signaling (pEC50=8.1), with potency and efficacy similar to morphine, but with far less β-arrestin recruitment and receptor internalization.
CSN15841 TRV 130 HCl 1401031-39-7 TRV 130 hydrochloride is a μ-opioid receptor (MOR) G protein-biased ligand and elicits robust G protein signaling (pEC50=8.1), with potency and efficacy similar to morphine, but with far less β-arrestin recruitment and receptor internalization.
CSN12642 Trimebutine Maleate 34140-59-5 Trimebutine Maleate is an agonist effect on peripheral μ, k and δ opiate receptors, and also shows antimuscarinic effect.
CSN12147 Trimebutine 39133-31-8 Trimebutine is an agonist effect on peripheral μ, k and δ opiate receptors, and also shows antimuscarinic effect.
CSN21214 PZM-21 1997387-43-5 PZM21 is a potent and selective μ opioid receptor agonist with an EC50 of 1.8 nM.
CSN22475 ORL1 Antagonist 1 1174985-59-1 ORL1 antagonist 1 is an opioid receptor-like 1 (ORL1) antagonist with an IC50 of 61 nM.
CSN11518 Naltrexone HCl 16676-29-2 Naltrexone HCl is an antagonist of μ-opioid receptor.
CSN17742 Naloxegol Oxalate 1354744-91-4 Naloxegol oxalate is a CYP3A4 enzyme inhibitor, is a peripherally-selective opioid antagonist, for the treatment of opioid-induced constipation.
CSN18476 Naloxegol 854601-70-0 Naloxegol is both a peripherally selective opioid receptor antagonist and a CYP3A4 enzyme inhibitor.
CSN11529 N-Desmethylclozapine 6104-71-8 N-Desmethylclozapine is a dengue virus inhibitor, and an agonist of δ-opioid receptor.
CSN11162 Met-Enkephalin 58569-55-4 Met-enkephalin is an Opioid related peptide work as a potent agonist of the δ-opioid receptor, and to a lesser extent the μ-opioid receptor, with little to no effect on the κ-opioid receptor.
CSN11381 Meptazinol HCl 59263-76-2 Meptazinol HCl is both a partial agonist of μ1 opioid receptor and an AChE inhibitor.
CSN17469 MCOPPB triHCl 1108147-88-1 MCOPPB trihydrochloride is a nociceptin receptor agonist with pKi of 10.07, displaying weaker activity at other opioid receptors.
CSN17719 LY2795050 1346133-08-1 LY2795050 is a selective κ-opioid Receptor (KOR) antagonist (IC50=0.72 nM) and has the potential as a PET tracer to image KOR in vivo.
CSN20227 LY2444296 1346133-11-6 LY2444296 is a short-acting kappa opioid receptor antagonist.
CSN23719 LY-2940094 Tartrate 1307245-87-9 LY-2940094 tartrate is the tartrate form of LY-2940094 which is an antagonist of nociceptin receptor that is used for the treatment of major depressive disorder and alcoholism.
CSN20601 LY2456302 1174130-61-0 LY-2456302 is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM.
CSN11327 Loperamide 53179-11-6 Loperamide is a medication used to decrease the frequency of diarrhea.
CSN11328 Loperamide HCl 34552-83-5 Loperamide HCl is a potent and selective μ-opioid receptor agonist.
CSN16622 JTC-801 244218-51-7 JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, and weakly inhibits receptors δ, κ, and μ.
CSN16488 JDTic 361444-66-8 JDTic is a highly selective antagonist for the κ-opioid receptor and without affecting the μ- or δ-opioid receptors.
CSN18435 JDTic 2HCl 785835-79-2 JDTic dihydrochloride is a highly selective antagonist for the κ-opioid receptor without affecting the μ- or δ-opioid receptors.
CSN22567 DAMGO 78123-71-4 Highly selective peptide agonist for the μ opioid receptor.
CSN19796 GSK-1521498 1007573-18-3 GSK-1521498 is a μ-opioid receptor antagonist. It has been shown to attenuate reward-driven compulsive behaviours, such as stimulant drug seeking or binge eating, in animals and humans.
CSN10947 Ethoheptazine 77-15-6 Ethoheptazine is an opioid analgesic from the phenazepane family.
CSN10924 Eptazocine 72522-13-5 Eptazocine interacts with opioid receptor, and is classified as one of the opiate agonist-antagonist analgesics.
CSN21147 DADLE 63631-40-3 DADLE ([D-Ala2, D-Leu5]-Enkephalin) is a water soluble Opioid Receptor peptide agonist.
CSN19110 Cebranopadol (1α,4α)stereoisomer 863513-93-3 Cebranopadol(1α,4α)stereoisomer is a stereoisomer of cebranopadol.
CSN13503 Cebranopadol 863513-91-1 Cebranopadol is an analgesic NOP and opioid receptor agonist with Kis/EC50s of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, 18 nM/110 nM for human NOP, MOP, KOP and delta-opioid peptide (DOP) receptor, respectively.
CSN17791 BAN ORL 24 1401463-54-4 BAN ORL 24 is a potent and selective NOP receptor antagonist. (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively).
CSN23662 AR-M 1000390 HCl 209808-47-9 AR-M 1000390 HCl is a non-peptidic and low-internalizing δ-selective opioid receptor agonist.
CSN13513 Alvimopan 156053-89-3 Alvimopan is a peripherally selective opioid mu receptor antagonist.
CSN13650 Alvimopan Dihydrate 170098-38-1 Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery.
CSN17774 Alvimopan Monohydrate 1383577-62-5 Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery.
CSN12425 ADL-5859 HCl 850173-95-4 ADL-5859 HCl is both a δ-opioid receptor agonist (Ki=0.84 nM, EC50=20 nM) and selectivity against opioid receptor κ, μ, and weak inhibitory activity at the hERG channel with IC50 value of 78 µM.
CSN18860 (R)-ZINC-3573 2089389-15-9 (R)-ZINC-3573 can activate endogenous MRGPRX2 in a human mast cell line and induce degranulation and calcium release.
CSN17203 (-)-Naltrexone 16590-41-3 (-)-Naltrexone is an opioid receptor antagonist used primarily in the management of alcohol dependence and opioid dependence.
CSN11317 (-)-Menthol 2216-51-5 (-)-Menthol is a natural product obtained from the oils of corn mint, peppermint, or other mints, as a weak kappa opioid receptor agonist. It has local anesthetic and counterirritant qualities, and used to relieve minor throat irritation.
CSN19330 (+)-Matrine 519-02-8 (+)-Matrine is a naturally occuring κ-opioid and μ-opioid receptor agonist.
CSN14746 Akuammigine 642-17-1
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