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Opioid Receptor

Opioid Receptor

货号 产品名 CAS号 信息
CSN18678 [D-Ala2]Leucine-Enkephalin 64963-01-5 [D-Ala2]Leucine-Enkephalin is a potent, long-acting Leu-enkephalin analog agonist of delta opioid receptor.
CSN20210 TRV0109101 1401027-29-9 TRV0109101, a G protein-biased agonist of the µ-opioid receptor, which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia.
CSN20211 TRV0109101 HCl 2101210-22-2 TRV0109101 HCl, a G protein-biased agonist of the µ-opioid receptor, which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia.
CSN17789 TRV 130 Racemate 1401028-25-8 TRV 130 racemate is the racemate form of TRV130, which a μ-opioid receptor (MOR) G protein-biased ligand.
CSN17788 TRV 130 1401028-24-7 TRV 130 is a μ-opioid receptor (MOR) G protein-biased ligand and elicits robust G protein signaling (pEC50=8.1), with potency and efficacy similar to morphine, but with far less β-arrestin recruitment and receptor internalization.
CSN15841 TRV 130 HCl 1401031-39-7 TRV 130 HCl is a μ-opioid receptor (MOR) G protein-biased ligand and elicits robust G protein signaling (pEC50=8.1), with potency and efficacy similar to morphine, but with far less β-arrestin recruitment and receptor internalization.
CSN12642 Trimebutine Maleate 34140-59-5 Trimebutine Maleate is an agonist effect on peripheral μ, k and δ opiate receptors, and also shows antimuscarinic effect.
CSN12147 Trimebutine 39133-31-8 Trimebutine is an agonist effect on peripheral μ, k and δ opiate receptors, and also shows antimuscarinic effect.
CSN21214 PZM-21 1997387-43-5 PZM21 is a potent and selective μ opioid receptor agonist with an EC50 of 1.8 nM.
CSN22475 ORL1 Antagonist 1 1174985-59-1 ORL1 antagonist 1 is an opioid receptor-like 1 (ORL1) antagonist with an IC50 of 61 nM.
CSN17742 Naloxegol Oxalate 1354744-91-4 Naloxegol oxalate is a CYP3A4 enzyme inhibitor, is a peripherally-selective opioid antagonist, for the treatment of opioid-induced constipation.
CSN18476 Naloxegol 854601-70-0 Naloxegol is both a peripherally selective opioid receptor antagonist and a CYP3A4 enzyme inhibitor.
CSN11529 N-Desmethylclozapine 6104-71-8 N-Desmethylclozapine is a dengue virus inhibitor, and an agonist of δ-opioid receptor.
CSN11162 Met-Enkephalin 58569-55-4 Met-enkephalin is an Opioid related peptide work as a potent agonist of the δ-opioid receptor, and to a lesser extent the μ-opioid receptor, with little to no effect on the κ-opioid receptor.
CSN11381 Meptazinol HCl 59263-76-2 Meptazinol HCl is both a partial agonist of μ1 opioid receptor and an AChE inhibitor.
CSN17469 MCOPPB triHCl 1108147-88-1 MCOPPB 3HCl is a nociceptin receptor agonist with pKi of 10.07, displaying weaker activity at other opioid receptors.
CSN17719 LY2795050 1346133-08-1 LY2795050 is a selective κ-opioid Receptor (KOR) antagonist (IC50=0.72 nM) and has the potential as a PET tracer to image KOR in vivo.
CSN20227 LY2444296 1346133-11-6 LY2444296 is a short-acting kappa opioid receptor antagonist.
CSN23719 LY-2940094 Tartrate 1307245-87-9 LY-2940094 tartrate is the tartrate form of LY-2940094 which is an antagonist of nociceptin receptor that is used for the treatment of major depressive disorder and alcoholism.
CSN20601 LY2456302 1174130-61-0 LY-2456302 is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM.
CSN11327 Loperamide 53179-11-6 Loperamide is a medication used to decrease the frequency of diarrhea.
CSN11328 Loperamide HCl 34552-83-5 Loperamide HCl is a potent and selective μ-opioid receptor agonist.
CSN16622 JTC-801 244218-51-7 JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, and weakly inhibits receptors δ, κ, and μ.
CSN16488 JDTic 361444-66-8 JDTic is a highly selective antagonist for the κ-opioid receptor and without affecting the μ- or δ-opioid receptors.
CSN18435 JDTic 2HCl 785835-79-2 JDTic 2HCl is a highly selective antagonist for the κ-opioid receptor without affecting the μ- or δ-opioid receptors.
CSN19796 GSK-1521498 1007573-18-3 GSK-1521498 is a μ-opioid receptor antagonist. It has been shown to attenuate reward-driven compulsive behaviours, such as stimulant drug seeking or binge eating, in animals and humans.
CSN10947 Ethoheptazine 77-15-6 Ethoheptazine is an opioid analgesic from the phenazepane family.
CSN10924 Eptazocine 72522-13-5 Eptazocine interacts with opioid receptor, and is classified as one of the opiate agonist-antagonist analgesics.
CSN21147 DADLE 63631-40-3 DADLE ([D-Ala2, D-Leu5]-Enkephalin) is a water soluble Opioid Receptor peptide agonist.
CSN19110 Cebranopadol (1α,4α)stereoisomer 863513-93-3 Cebranopadol(1α,4α)stereoisomer is a stereoisomer of cebranopadol.
CSN13503 Cebranopadol 863513-91-1 Cebranopadol is an analgesic NOP and opioid receptor agonist with Kis/EC50s of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, 18 nM/110 nM for human NOP, MOP, KOP and delta-opioid peptide (DOP) receptor, respectively.
CSN25444 BRL 52537 hydrochloride 112282-24-3 BRL-52537 hydrochloride is a potent and highly selective κ-opioid agonist. It has neuroprotective effects in animal studies, and is used for research into potential treatments for stroke and heart attack as well as more general brain research.
CSN27537 Bevenopran 676500-67-7 Bevenopran is a peripheral μ-opioid receptor antagonist.
CSN17791 BAN ORL 24 1401463-54-4 BAN ORL 24 is a potent and selective NOP receptor antagonist. (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively).
CSN23662 AR-M 1000390 HCl 209808-47-9 AR-M 1000390 HCl is a non-peptidic and low-internalizing δ-selective opioid receptor agonist.
CSN13513 Alvimopan 156053-89-3 Alvimopan is a peripherally selective opioid mu receptor antagonist.
CSN13650 Alvimopan Dihydrate 170098-38-1 Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery.
CSN17774 Alvimopan Monohydrate 1383577-62-5 Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery.
CSN14746 Akuammigine 642-17-1 Akuammidine, a natural product isolated and purified from the herbs of Picralima nitida with in vitro antimalarial activity, shows a preference for mu-opioid binding sites with Ki values of 0.6, 2.4 and 8.6 mM at mu-, delta- and kappa-opioid binding sites, respectively and the agonist actions of akuammidine in the mouse-isolated vas deferens were antagonised by naloxone and the mu-opioid receptor selective antagonist D-Phe-Cys-Tyr-D-Trp-Orn-Thr-Pen-Thr-NH2 (CTOP) confirming an action at mu-opioid receptors, and competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding pA2 values of 4.68.
CSN12425 ADL-5859 HCl 850173-95-4 ADL-5859 HCl is both a δ-opioid receptor agonist (Ki=0.84 nM, EC50=20 nM) and selectivity against opioid receptor κ, μ, and weak inhibitory activity at the hERG channel with IC50 value of 78 µM.
CSN11317 (-)-Menthol 2216-51-5 (-)-Menthol is a natural product obtained from the oils of corn mint, peppermint, or other mints, as a weak kappa opioid receptor agonist. It has local anesthetic and counterirritant qualities, and used to relieve minor throat irritation.
CSN19330 (+)-Matrine 519-02-8 (+)-Matrine is a naturally occuring κ-opioid and μ-opioid receptor agonist.
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