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Cannabinoid Receptor

Cannabinoid Receptor

货号 产品名 CAS号 信息
CSN18972 Taranabant (1R,2R)stereoisomer 701977-08-4 Taranabant(1R,2R)stereoisomer is the R-Enantiomer of taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist.
CSN12382 Taranabant 701977-09-5 Taranabant is a cannabinoid 1 receptor inverse agonist with IC50 of 0.3 nM.
CSN19427 Rimonabant 168273-06-1 Rimonabant is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM.
CSN10030 Rimonabant HCl 158681-13-1 Rimonabant hydrochloride is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM.
CSN18394 Otenabant 686344-29-6 Otenabant is a selective, potent and competitive CB1 receptor antagonist with Ki of 0.7 nM.
CSN13721 Org 27569 868273-06-7 Org 27569 is an allosteric modulator of cannabinoid CB1 receptor, induces a CB1 receptor state that is characterized by enhanced agonist affinity and decreased inverse agonist affinity.
CSN22151 MK-9470 947371-30-4 MK-9470 is a selective, high-affinity, inverse agonist (human IC50=0.7 nM) for the cannabinoid CB1 receptor (CB1R) developed for use in human brain imaging.
CSN13453 MDA 19 1048973-47-2 MDA 19 is a selective human CB2 receptor agonist with Ki of 43.3 nM.
CSN19472 LY320135 176977-56-3 LY-320135 is a potent and selective Canniboid CB1 receptor antagonist/inverse agonist. LY-320135 is selective (~70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki = 6.4 μM) and muscarinic receptors (Ki = 2.1 μM).
CSN20218 JD5037 1392116-14-1 JD-5037 is a peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.
CSN19173 GW842166X 666260-75-9 GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor.
CSN21228 CB2R-IN-1 1257555-79-5 CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.
CSN20330 CB2 Agonist C8 2052602-31-8 CB2 agonist C8 is an agonists of cannabinoid receptor type 2.
CSN20331 CB2 Agonist C36 2097512-96-2 CB2 agonist C36 is an agonists of cannabinoid receptor type 2.
CSN10473 BML-190 2854-32-2 BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor.
CSN10421 beta-Amyrin 559-70-6 beta-Amyrin, a natural cannabinoid receptors agonist isolated and purified from the stem bark of Alstonia boonei, has anti-inflammatory activity. Beta-Amyrin significantly inhibits PGE2, IL-6 secretion, and NF-κB activation in a concentration-dependent manner on LPS-induced hPBMCs.
CSN18739 BAY 59-3074 406205-74-1 Bay 59-3074 is a selective CB1/CB2 receptor partial agonist with Kis of 48.3 and 45.5 nM at human CB1 and CB2 receptors respectively .
CSN12849 AM630 164178-33-0 AM630 is a selectivity CB2 antagonist with Ki of 31.2 nM with a > 150 fold selectivity over CB1 receptor.
CSN18640 A-836339 959746-77-1 A-836339 is a cannabinoid CB2 receptor-selective agonist and exhibits high potencies at CB(2) and selectivity over CB(1) receptors.
CSN21999 (±)-SLV319 362519-49-1 (±)-SLV319 is a selective antagonist of cannabinoid-1 (CB1) receptor with Ki value of 7.8 nM and it has a weaker activation effect on CB2.
CSN12783 (-)-Gallocatechin 3371-27-5 (-)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor.
CSN15641 (+)-Gallocatechin 970-73-0 (+)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor.
CSN15642 beta-Amyrin Acetate 1616-93-9
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