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Cannabinoid Receptor

Cannabinoid Receptor

货号 产品名 CAS号 信息
CSN21516 β-Caryophyllene 87-44-5 β-Caryophyllene is an agonist of the cannabinoid (CB) receptor CB2 with Ki of 155 nM.
CSN12586 (R)-(5-Methyl-3-(morpholinomethyl)-2,3-dihydro-[1,4]oxazino[2,3,4-hi]indol-6-yl)(naphthalen-1-yl)methanone methanesulfonate 131543-23-2 WIN 55212-2 mesylate is a potent aminoalkylindole cannabinoid (CB) receptor agonist with a Ki of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively.
CSN25682 VDM 11 313998-81-1 VDM 11 is a selective inhibitor of the anandamide membrane transporter (AMT) with IC50 values of 4 - 11 μM.
CSN25626 1-(2,4-Dichlorophenyl)-4-ethyl-N-(piperidin-1-yl)-5-(5-((4-(trifluoromethyl)phenyl)ethynyl)thiophen-2-yl)-1H-pyrazole-3-carboxamide 1253641-65-4 TM38837 is a novel, largely peripherally restricted CB1 antagonist with limited penetrance to the brain. Oral dose of TM38837 (100 mg/kg) induced a significant increase in freezing behavior.
CSN18972 Taranabant ((1R,2R)stereoisomer) 701977-08-4 Taranabant(1R,2R)stereoisomer is the R-Enantiomer of taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist.
CSN12382 Taranabant 701977-09-5 Taranabant is a cannabinoid 1 receptor inverse agonist with IC50 of 0.3 nM.
CSN19427 Rimonabant 168273-06-1 Rimonabant is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM.
CSN10030 Rimonabant HCl 158681-13-1 Rimonabant HCl is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM.
CSN24663 PF-514273 851728-60-4 PF 514273 is a selective CB1 receptor antagonist with Ki values of 1 and > 10000 nM at CB1 and CB2 receptors respectively.
CSN18394 Otenabant 686344-29-6 Otenabant is a selective, potent and competitive CB1 receptor antagonist with Ki of 0.7 nM.
CSN16613 Otenabant HCl 686347-12-6 Otenabant HCl is a recently discovered selective, high affinity, competitive CB1 receptor antagonist with Ki of 0.7 nM.
CSN13721 Org 27569 868273-06-7 Org 27569 is an allosteric modulator of cannabinoid CB1 receptor, induces a CB1 receptor state that is characterized by enhanced agonist affinity and decreased inverse agonist affinity.
CSN24683 OMDM-2 616884-63-0 OMDM-2 is a stable and selective inhibitor of anandamide cellular uptake with Ki of 3 μM.
CSN25339 MAFP 188404-10-6 MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM.
CSN19472 LY320135 176977-56-3 LY-320135 is a potent and selective Canniboid CB1 receptor antagonist/inverse agonist. LY-320135 is selective (~70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki = 6.4 μM) and muscarinic receptors (Ki = 2.1 μM).
CSN24685 Leelamine HCl 16496-99-4 Leelamine hydrochloride is an agonist of cannabinoid Receptor 1 (CB1).
CSN24684 JTE-907 282089-49-0 JTE 907 is a highly selective cannabinoid CB2 receptor inverse agonist that binds with high affinity to rat, mouse and human CB2 receptors with Ki of 0.38, 1.55 and 35.9 nM respectively.
CSN20218 JD-5037 1392116-14-1 JD-5037 is a peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.
CSN19173 GW842166X 666260-75-9 GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor.
CSN21228 CB2R-IN-1 1257555-79-5 CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.
CSN20330 CB2 Agonist C8 2052602-31-8 CB2 agonist C8 is an agonists of cannabinoid receptor type 2.
CSN20331 CB2 Agonist C36 2097512-96-2 CB2 agonist C36 is an agonists of cannabinoid receptor type 2.
CSN17330 CB1-IN-1 1429239-98-4 CB1-IN-1 is a peripherally restricted CB1R antagonist, with Ki of 0.3 nM and 21 nM for CB1R (EC50 = 3 nM) and CB2R, respectively.
CSN10473 BML-190 2854-32-2 BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor.
CSN10421 β-Amyrin 559-70-6 beta-Amyrin, a natural cannabinoid receptors agonist isolated and purified from the stem bark of Alstonia boonei, has anti-inflammatory activity. Beta-Amyrin significantly inhibits PGE2, IL-6 secretion, and NF-κB activation in a concentration-dependent manner on LPS-induced hPBMCs.
CSN15642 β-Amyrin acetate 1616-93-9 beta-Amyrin acetrate, a natural cannabinoid receptor isolated and purified from the herbs of Alstonia boone, shows significant HMG-CoA-reductase and sEH inhibitory activities.
CSN18739 Bay 59-3074 406205-74-1 Bay 59-3074 is a selective CB1/CB2 receptor partial agonist with Kis of 48.3 and 45.5 nM at human CB1 and CB2 receptors respectively .
CSN25672 Arvanil 128007-31-8 Arvanil is an antagonist of cannabinoid CB1 and vanilloid TRPV1 (VR1) with Ki values are 0.5 and 0.3 μM respectively.
CSN12849 (6-Iodo-2-methyl-1-(2-morpholinoethyl)-1H-indol-3-yl)(4-methoxyphenyl)methanone 164178-33-0 AM630 is a selectivity CB2 antagonist with Ki of 31.2 nM with a > 150 fold selectivity over CB1 receptor.
CSN24665 CB1 antagonist 2 614726-85-1 AM 4113 is selective CB1 antagonist with Kd of 0.89 nM.
CSN24666 Arachidonylcyclopropylamide 229021-64-1 ACPA is a selective agonist of CB1 with Ki of 2.2 nM.
CSN18640 A-836339 959746-77-1 A-836339 is a cannabinoid CB2 receptor-selective agonist and exhibits high potencies at CB(2) and selectivity over CB(1) receptors.
CSN21999 (±)-Ibipinabant 362519-49-1 (±)-SLV319 is a selective antagonist of cannabinoid-1 (CB1) receptor with Ki value of 7.8 nM and it has a weaker activation effect on CB2.
CSN24668 (R)-Methanandamide 157182-49-5 (R)-(+)-Methanandamide, the stable anandamide analog, is a selective agonist for the CB1 receptor with Ki values of 20 and 815 nM for CB1 and CB2 receptors respectively.
CSN12783 (-)-gallocatechin 3371-27-5 (-)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor.
CSN15641 (+)-Gallocatechin 970-73-0 (+)-Gallocatechin, a natural product isolated and purified from the wood of Acacia catechu (L.F.) Willd., has moderate affinity to the human cannabinoid receptor.
CSC24669 ACEA 220556-69-4
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