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PAR

PAR

货号 产品名 CAS号 信息
CSN13782 Vorapaxar 618385-01-6 Vorapaxar is a thrombin receptor (protease-activated receptor, PAR-1) antagonist.
CSN17809 TRAP-6 141136-83-6 TRAP-6 is protease-activated receptor 1 (PAR1) agonist.
CSN23082 RWJ 56110 252889-88-6 RWJ-56110 is a selective protease-activated receptor-1 (PAR1) antagonist. It blocks thrombin-induced platelet aggregation and activation of MAPK in HUVECs.
CSN23119 SLIGKV-NH2 190383-13-2 Protease-Activated Receptor-2, amide (SLIGKV-NH2) is a highly potent protease-activated receptor-2 (PAR2) activating peptide.
CSN23110 SCH 79797 2HCl 1216720-69-2 Potent, selective non-peptide PAR1 antagonist
CSN13679 ML161 423735-93-7 ML-161 is an allosteric and reversible inhibitor of proteinase-activated receptor 1 (PAR1) with IC50 of 0.26 μM.
CSN25350 GB-88 1416435-96-5 GB-88 is an oral, selective non-peptide antagonist of PAR2. It inhibits PAR2 activated Ca2+ release with an IC50 of 2 µM.
CSN22824 FSLLRY-NH2 245329-02-6 FSLLRY-NH2 is a selective PAR2 peptide antagonist.
CSN22822 FR 171113 173904-50-2 FR 171113 is a protease-activated receptor 1 (PAR1) antagonist.
CSN24830 ENMD-1068 789488-77-3 ENMD-1068 is a PAR2 antagonist with IC50 value of 1.2 mM.
CSN22353 AZ3451 2100284-59-9 AZ3451 is a protease-activated receptor-2 (PAR2) antagonist.
CSN24081 E5555 751475-53-3 Atopaxar, also known as E5555, is a potent and orally-active PAR-1 inhibitor. E5555 inhibited the binding of a high-affinity thrombin receptor-activating peptide ([(3)H]haTRAP) to PAR-1 with a half maximal inhibitory concentration (IC(50)) value of 0.019μM. E5555 showed potent inhibitory effects on human platelet aggregation induced by thrombin and TRAP with IC(50) values of 0.064 and 0.031μM, respectively. E5555 showed potent and selective inhibitory effects on guinea pig platelet aggregation induced by thrombin and TRAP with IC(50) values of 0.13 and 0.097μM, respectively. E5555 could be a therapeutic option for atherothrombotic disease.
CSN18572 AC-55541 916170-19-9 AC-55541 is a small-molecule protease-activated receptor 2 (PAR2) agonist and activates PAR2 signaling in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays, with potencies ranging from 200 to 1000 nM.
CSN22664 AC 264613 1051487-82-1 AC 264613 is a potent and selective protease-activated receptor 2 (PAR2) agonist with pEC50 = 7.5.
CSN22646 2-Furoyl-LIGRLO-amide 729589-58-6 2-Furoyl-LIGRLO-amide is a potent and selective PAR2 receptor agonist with pD2 of 7.0.
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