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AChR

AChR

货号 产品名 CAS号 信息
CSN10132 Varenicline HCl 230615-23-3 Varenicline HCl is a nicotinic receptor partial agonist and it stimulates nicotine receptors more weakly than nicotine itself does.
CSN12157 Trospium Chloride 10405-02-4 Trospium chloride is a competitive antagonist at muscarinic cholinergic receptors, used to treat symptoms of an overactive bladder.
CSN12156 Tropicamide 1508-75-4 Tropicamide is a mAchR M4 antagonist, used to dilate the pupil and help with examination of the eye.
CSN10848 Trihexyphenidyl HCl 52-49-3 Trihexyphenidyl HCl works as an antiparkinsonian agent which binds to the M1 muscarinic receptor.
CSN11994 Succinylcholine Chloride Dihydrate 6101-15-1 Succinylcholine chloride is a nAchR which acts as a depolarizing neuromuscular blocke, used as a quaternary skeletal muscle relaxant.
CSN23115 SIB 1553A HCl 191611-89-9 SIB-1553A is a nicotinic acetylcholine receptor agonist potentially for the treatment of Alzheimer’s disease (AD).
CSN24694 (R)-N-(Quinuclidin-3-yl)-2,3-dihydrobenzo[b][1,4]dioxine-6-carboxamide fumarate 527680-57-5 Selective α7 nAChR agonist
CSN23842 Scopolamine N-Oxide HydrobroMide Monohydrate N/A Scopolamine N-oxide hydrobromide is an antagonist of the muscarinic acetylcholine.
CSN11852 Rivastigmine Tartrate 129101-54-8 Rivastigmine tartrate is an AchR inhibitor use for treatment of mild to moderate Alzheimer's disease and Parkinson's disease with elimination half-life of ‎1.5 hours.
CSN11810 Pyrithioxin 2HCl 10049-83-9 Pyrithioxin 2HCl is a neurodynamic compound, combined with a short period of hyperventilation (HV) was applied in cerebral infarct patients with Hemiplegia.
CSN11802 Pyrantel 15686-83-6 Pyrantel is a medication used to treat a number of parasitic worm infections.
CSN11794 Protriptyline HCl 1225-55-4 Protriptyline HCl is a tricyclic antidepressant (TCA), specifically a secondary amine, for the treatment of depression and ADHD.
CSN10107 Procaine HCl 51-05-8 Procaine HCl is a local anesthetic drug of the amino ester group.
CSN11494 PNU-120596 501925-31-1 PNU-120596 is a a type II positive allosteric modulator of α7 nAChRs with an EC50 of 0.2 μM.
CSN25236 Pirmenol 68252-19-7 Pirmenol inhibited the muscarinic acetylcholine receptor-operated K+ current (I[K.ACh]) in atrial cells and on experimental atrial fibrillation in isolated guinea-pig hearts.
CSN11734 Pirenzepine 2HCl 29868-97-1 Pirenzepine 2HCl is a is an anticholinergic agent and induces the dimerization of muscarinic M1 receptors, used to treat myopia, gastric and duodenal ulcers.
CSN24691 (R)-N-(Furo[2,3-c]pyridin-5-ylmethyl)quinuclidin-3-amine 478149-53-0 PHA-543613 acts as a potent and selective agonist for the α7 subtype of neural nicotinic acetylcholine receptors, with a high level of brain penetration and good oral bioavailability. It is under development as a possible treatment for cognitive deficits in schizophrenia.
CSN11636 Oxybutynin HCl 1508-65-2 Oxybutynin HCl a synthetic anticholinergic agent used for treatment of urinary incontinence and overactive bladder syndrome, with elimination half-life of ‎12.4–13.2 hours. Oxybutynin HCl is the HCl form of Oxybutynin.
CSN11635 Oxybutynin 5633-20-5 Oxybutynin a synthetic anticholinergic agent used for treatment of urinary incontinence and overactive bladder syndrome, with elimination half-life of ‎12.4–13.2 hours.
CSN24546 N,N,N-Trimethyl-4-(2-oxopyrrolidin-1-yl)but-2-yn-1-aminium iodide 3854-04-4 Oxotremorine M iodide is a potent and selective muscarinic acetylcholine receptor (mAChR) agonist. Oxotremorine M iodide potentiates NMDA receptors by muscarinic receptor dependent and independent mechanisms[1].
CSN24692 3-(3-Bromothiophen-2-yl)-8-methyl-8-azabicyclo[3.2.1]oct-2-ene fumarate 216853-60-0 NS3861 is an α3β2 full agonist and an α3β4 partial agonist.
CSN11378 Mepenzolate Bromide 76-90-4 Mepenzolate bromide mAchR antagonist, working as a post-ganglionic parasympathetic inhibitor to decrease gastric acid and pepsin secretion and suppresse spontaneous contractions of the colon.
CSN24142 Mecamylamine HCl 826-39-1 Mecamylamine HCl is a non-competitive nicotinic acetylcholine receptor antagonist with antidepressant-like effects in mice.
CSN11213 Ipratropium Bromide' 22254-24-6 Ipratropium bromide is a synthetic derivative of the alkaloid atropine anticholinergic properties with anticholinergic properties.
CSN24690 1,4-Diazabicyclo[3.2.2]nonan-4-yl(5-(3-(trifluoromethyl)phenyl)furan-2-yl)methanone hydrochloride 753499-14-8 High affinity α7 nAChR partial agonist; anti-inflammatory
CSN11146 Hexamethonium Bromide 55-97-0 Hexamethonium bromide is a nicotinic cholinergic antagonist as the prototypical ganglionic blocker.
CSN11109 Glycopyrrolate 596-51-0 Glycopyrrolate is a muscarinic competitive antagonist used as an antispasmodic.
CSN11016 Flavoxate HCl 3717-88-2 Flavoxate HCl is a competitive AChR antagonist with IC50 of 12.2 μM, used as a muscle relaxant.
CSN10869 Dronedarone 141626-36-0 Dronedarone is a therapeutic agent with a structural resemblance to amiodarone and a better side effect profile and it is a multichannel blocker with antiadrenergic properties and has been evaluated in both rate and rhythm control strategies in the management of AF.
CSN10806 Diphenidol 972-02-1 Diphenidol is indicated in the prevention and symptomatic treatment of peripheral (labyrinthine) vertigo and associated nausea and vomiting that occur in such conditions as Meniere's disease and surgery of the middle and inner ear.
CSN10833 Diphenmanil Methylsulfate 62-97-5 Diphemanil methylsulfate can bind the muscarinic M3 receptor and decrease secretory excretion of stomach acids and saliva and sweat, as well as works as a direct smooth muscle spasmolytic activity.
CSN10756 Decamethonium Bromide 541-22-0 Decamethonium bromide is a nAChR partial agonist,working as short acting depolarizing muscle relaxant or neuromuscular blocking agent.
CSN11123 Cytisine 485-35-8 Cytisine is a naturally occuring alkaloid nAchR agonist with a short half-life of 4.8 hours.
CSN10656 Cisatracurium Besylate 96946-42-8 Cisatracurium besylate is an antagonize of AchR and inhibits neuromuscular transmission, a nondepolarizing skeletal muscle relaxant.
CSN10604 Cevimeline 107233-08-9 Cevimeline is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors and used in the treatment of dry mouth associated with sjogren's syndrome.
CSN10453 Biperiden 514-65-8 Biperiden is an antiparkinsonian agent, which is the selective central M1 cholinoreceptors blocker.
CSN11940 Benztropine Mesylate 132-17-2 Benztropine mesylate is a central muscarinic antagonist and a DAT inhibitor with IC50 of 118 nM, indicated for symptomatic relief of parkinsonism and drug-induced extrapyramidal reactions.
CSN10331 Arecoline Hydrobromide 300-08-3 Arecoline hydrobromide is a mAchR receptor agonist with EC50 values of 7, 95, 11, 410, and 69 nM for M1, M2, M3, M4, and M5, respectively, a nicotinic acid-based alkaloid found in the areca nut.
CSN10330 Arecaidine But-2-Ynyl Ester Tosylate 499-04-7 Arecaidine but-2-ynyl ester tosylate is a potent muscarinic agonist that shows 4.6-fold that is selectivity for mAChR M2 in the atrium versus those in the ileum.
CSN10316 Anisodamine 55869-99-3 Anisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant.
CSN10215 Aclidinium Bromide 320345-99-1 Aclidinium bromide is a long-acting, inhaled muscarinic antagonist as a maintenance treatment for chronic obstructive pulmonary disease (COPD).
CSN10209 Acetylcholine Iodide 2260-50-6 Acetylcholine iodide is an ester of choline and acetic acid, which acts as a transmitter substance of nerve impulses within the central and peripheral nervous systems.
CSN10208 Acetylcholine Chloride 60-31-1 Acetylcholine chloride is a neurotransmitter that can induce the opening of calcium channels.
CSN25275 (S)-PNU-282987 HCl 128311-08-0 (S)-PNU-282987 is the an absolute stereochemistry form of PNU-282987.
CSN25570 (-)-(S)-B-973B 2244989-34-0 (-)-(S)-B-973B is positive allosteric modulator of α7 nAChRs with EC50 of ~0.3 μM.
CSN24754 CCMI   917837-54-8
CSN25357 Ethyl (triphenylphosphoranylidene) acetate 1099-45-2
CSN25425 LY 2033298 New 886047-13-8
CSN25424 Cyclopentolate HCl 5870-29-1
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