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Histamine Receptor

Histamine Receptor

货号 产品名 CAS号 信息
CSN12374 Tripelennamine HCl 154-69-8 Tripelennamine HCl is an antagonist of H1-receptor that used as a psychoactive drug with antipruritic activity.
CSN12316 Rupatadin Fumarate 182349-12-8 Rupatadine fumarate is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively.
CSN11869 Roxatidine Acetate 78628-28-1 Roxatidine acetate is a specific and competitive histamine H2 receptor antagonist drug that is used to treat gastric ulcers, Zollinger–Ellison syndrome, erosive esophagitis, gastro-oesophageal reflux disease, and gastritis.
CSN13086 Roxatidine Acetate HCl 93793-83-0 Roxatidine acetate HCl is a slective antagonist of histamin H2 receptor.
CSN13516 Ranitidine HCl 66357-59-3 Ranitidine HCl is an antagonist of histamine H2-receptor that can inhibit stomach acid production.
CSN11722 Pimethixene 314-03-4 Pimethixene is an antihistamine and anticholinergic agent, that is often used to treat hyperactivity, anxiety, sleep disorders, and allergy.
CSN11691 Pheniramine Maleate 132-20-7 Pheniramine maleate can acts as an antihistamine and vasoconstrictor.
CSN11668 Pemirolast Potassium 100299-08-9 Pemirolast potassium is an antagonist of histamine H1 and mast cell stabilizer with antiallergic effect.
CSN11604 Olopatadine HCl 140462-76-6 Olopatadine HCl can block the release of histamine (IC50 = 559 µM) and stabilize mast cell.
CSN11565 Nizatidine 76963-41-2 Nizatidine is an antagonist of histamine H2 receptor that can inhibit the secretion of gastric acid.
CSN12482 Mizolastine 108612-45-9 Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
CSN11437 Mianserin 24219-97-4 Mianserin is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant.
CSN10479 Mianserin HCl 21535-47-7 Mianserin HCl is inverse agonist of H1 receptor and can be act as a psychoactive agent of the tetracyclic antidepressant.
CSN11809 Mepyramine Maleate 59-33-6 Mepyramine maleate is an antagonist of histamine H1 receptor.
CSN14575 Marmin 14957-38-1 Marmin, a natural product isolated and purified from the herbs of Citrus maxima with potent anti-ulcer, antibacterial, fungicidal, and algicidal properties, can inhibit contraction of the guinea-pig tracheal smooth muscle, especially by interfering histamine receptor, inhibiting the histamine release from mast, inhibiting intracellular Ca2+ release from the intracellular store and the Ca2+ influx through voltage-dependent Ca2+ channels, is potential to develop as antihistamine agents, especially as histamine H1 receptor antagonists by interacting with amino acid residues, Asp107, Lys179, Lys191, Asn198, and Trp428 of histamine H1 receptor, shows a cell-growth inhibitory effect against L1210 and K562 in vitro.
CSN11321 Lodoxamide Tromethamine 63610-09-3 Lodoxamide tromethamine is used as an ophthalmic solution that specially applying to the eye.
CSN25565 LML-134 1542135-76-1 LML134 is an orally active and high selective Histamine 3 receptor (H3R) inverse agonist with Kis of 0.3 nM and 12 nM for hH3R cAMP and hH3R bdg. LML134 penetrates the brain rapidly, leading to high H3R occupancy, and disengages its target with a fast kinetic profile. LML134 has the potential for excessive sleep disorders.
CSN13135 Levodropropizine 99291-25-5 Levodropropizine is a histamine receptor inhibitor, and is an effective and very well tolerated peripheral antitussive drug.
CSN11264 Lafutidine 118288-08-7 Lafutidine is an antagonist of histamine H(2)-receptor that inhibits gastric acid secretion.
CSN25273 JNJ-5207852 398473-34-2 JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
CSN11177 Hydroxyzine Pamoate 10246-75-0 Hydroxyzine pamoate is a histamine H1-receptor antagonist.
CSN11153 Histamine phosphate 51-74-1 Histamine phosphate can dilate arteries and capillaries mediated by H1- and H2-receptors.
CSN11010 Fexofenadine 83799-24-0 Fexofenadine is an antihistamine pharmaceutical drug used in the treatment of allergy symptoms, such as hay fever, nasal congestion, and urticaria.
CSN12462 Fexofenadine HCl 153439-40-8 Fexofenadine inhibits histamine H1 receptor with IC50 of 246 nM.
CSN10917 Epinastine HCl 108929-04-0 Epinastine HCl is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
CSN10884 Ebrotidine 100981-43-9 Ebrotidine is a competitive H2-receptor antagonist (Ki= 127.5 nM) with a potent antisecretory activity and evidenced gastroprotection.
CSN10883 Ebastine 90729-43-4 Ebastine is a selective H1-histamine receptor antagonist.
CSN10864 Doxylamine succinate salt 562-10-7 Doxylamine Succinate Salt is an antihistamine which inhibits histamine H1 receptors. It can be used as a short-term sedative and anticholinergic agent.
CSN10783 Dexchlorpheniramine Maleate 2438-32-6 Dexchlorpheniramine maleate is an antihistamine, with anticholinergic properties, used to treat allergic conditions.
CSN10775 Desloratadine 100643-71-8 Desloratadine is an antagonist of histamine H1 receptor that is used to treat allergies.
CSN10757 Decloxizine 3733-63-9 Decloxizine is a histamine 1 receptor antagonist.
CSN22573 Cyclizine 2HCl 5897-18-7 Cyclizine is a histamine H1 receptor antagonist of the piperazine class.
CSN10664 Clemizole 442-52-4 Clemizole is an antagonist of H1 histamine receptor that can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.
CSN10663 Clemastine Fumarate 14976-57-9 Clemastine fumarate is a selective antagonist of histamine H1 receptor with IC50 of 3 nM.
CSN12549 Cinnarizine 298-57-7 Cinnarizine, an antihistamine, can block calcium channel and promote cerebral blood flow. It is used to treat post-trauma cerebral symptoms and cerebral arteriosclerosis.
CSN10624 Chlorphenoxamine 77-38-3 Chlorphenoxamine is an antihistamine and anticholinergic and can be used as antipruritic and antiparkinsonian agent.
CSN10076 Chlorpheniramine Maleate 113-92-8 Chlorpheniramine maleate is an antagonist of histamine H1 receptor with IC50 of 12 nM.
CSN23808 Chlorcyclizine HCl 14362-31-3 Chlorcyclizine hydrochloride is a histamine H1 antagonist.
CSN10600 Cetirizine 83881-51-0 Cetirizine, a second-generation antihistamine, is a major metabolite of hydroxyzine, and a racemic selective H1 receptor inverse agonist used in the treatment of allergies, hay fever, angioedema, and urticaria.
CSN12995 Cetirizine 2HCl 83881-52-1 Cetirizine 2HCl, a metabolite of hydroxyzine, is racemic selective and inverse agonist of H1 receptor used in the treatment of allergies and hay fever.
CSN10548 Carbinoxamine Maleate 3505-38-2 Carbinoxamine maleate is a blocker of histamine-H1 receptor with antihistamine and anticholinergic effects.
CSN10500 Buclizine 2HCl 129-74-8 Buclizine 2HCl, the derivative of piperazine, is an antihistamine and anticholinergic agent.
CSN10492 Brompheniramine Maleate 980-71-2 Brompheniramine maleate is an antagonist of histamine H1 receptors.
CSN25269 Bromazine HCl 1808-12-4 Bromazine hydrochloride is an antagonist of histamine H1 receptor.
CSN10402 Bilastine 202189-78-4 Bilastine selectively antagonizes histamine H1 receptor and it is used to treat allergic rhinoconjunctivitis and urticaria.
CSN25225 Betahistine 5638-76-6 Betahistine is a histamine analog and H1 receptor agonist.
CSN24137 Bepotastine 125602-71-3 Bepotastine is a non-sedating and selective antagonist of the histamine 1 (H1) receptor.
CSN10365 Azatadine 3964-81-6 Azatadine is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.
CSN10364 Azatadine Dimaleate 3978-86-7 Azatadine dimaleate is an inhibitor of histamine and cholinergic with IC50 of 6.5 nM and 10 nM, respectively.
CSN10231 Alcaftadine 147084-10-4 Alcaftadine is a high affinity ligand for the H1 receptor, with a pKi (8.5) that is comparable with that of other H1 antihistamines.
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