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Histamine Receptor

Histamine Receptor

货号 产品名 CAS号 信息
CSN12228 Zaltidine 85604-00-8 Zaltidine is a H2-receptor antagonist, which has the antisecretory action.
CSN12374 Tripelennamine HCl 154-69-8 Tripelennamine HCl is an antagonist of H1-receptor that used as a psychoactive drug with antipruritic activity.
CSN12316 Rupatadin Fumarate 182349-12-8 Rupatadine fumarate is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively.
CSN11869 Roxatidine Acetate 78628-28-1 Roxatidine acetate is a specific and competitive histamine H2 receptor antagonist drug that is used to treat gastric ulcers, Zollinger–Ellison syndrome, erosive esophagitis, gastro-oesophageal reflux disease, and gastritis.
CSN13086 Roxatidine Acetate HCl 93793-83-0 Roxatidine acetate HCl is a slective antagonist of histamin H2 receptor.
CSN13516 Ranitidine HCl 66357-59-3 Ranitidine HCl is an antagonist of histamine H2-receptor that can inhibit stomach acid production.
CSN11722 Pimethixene 314-03-4 Pimethixene is an antihistamine and anticholinergic agent, that is often used to treat hyperactivity, anxiety, sleep disorders, and allergy.
CSN11691 Pheniramine Maleate 132-20-7 Pheniramine maleate can acts as an antihistamine and vasoconstrictor.
CSN11668 Pemirolast Potassium 100299-08-9 Pemirolast potassium is an antagonist of histamine H1 and mast cell stabilizer with antiallergic effect.
CSN11604 Olopatadine HCl 140462-76-6 Olopatadine HCl can block the release of histamine (IC50 = 559 µM) and stabilize mast cell.
CSN11565 Nizatidine 76963-41-2 Nizatidine is an antagonist of histamine H2 receptor that can inhibit the secretion of gastric acid.
CSN12482 Mizolastine 108612-45-9 Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
CSN11437 Mianserin 24219-97-4 Mianserin is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant.
CSN10479 Mianserin HCl 21535-47-7 Mianserin HCl is inverse agonist of H1 receptor and can be act as a psychoactive agent of the tetracyclic antidepressant.
CSN11423 Metiamide 34839-70-8 Metiamide is a histamine H2-receptor antagonist developed from another H2 antagonist, burimamide.
CSN11809 Mepyramine Maleate 59-33-6 Mepyramine maleate is an antagonist of histamine H1 receptor.
CSN14575 Marmin 14957-38-1 Marmin, a natural product isolated and purified from the herbs of Citrus maxima with potent anti-ulcer, antibacterial, fungicidal, and algicidal properties, can inhibit contraction of the guinea-pig tracheal smooth muscle, especially by interfering histamine receptor, inhibiting the histamine release from mast, inhibiting intracellular Ca2+ release from the intracellular store and the Ca2+ influx through voltage-dependent Ca2+ channels, is potential to develop as antihistamine agents, especially as histamine H1 receptor antagonists by interacting with amino acid residues, Asp107, Lys179, Lys191, Asn198, and Trp428 of histamine H1 receptor, shows a cell-growth inhibitory effect against L1210 and K562 in vitro.
CSN13135 Levodropropizine 99291-25-5 Levodropropizine is a histamine receptor inhibitor, and is an effective and very well tolerated peripheral antitussive drug.
CSN11264 Lafutidine 118288-08-7 Lafutidine is an antagonist of histamine H(2)-receptor that inhibits gastric acid secretion.
CSN25273 JNJ-5207852 398473-34-2 JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
CSN11177 Hydroxyzine Pamoate 10246-75-0 Hydroxyzine pamoate is a histamine H1-receptor antagonist.
CSN11153 Histamine phosphate 51-74-1 Histamine phosphate can dilate arteries and capillaries mediated by H1- and H2-receptors.
CSN11010 Fexofenadine 83799-24-0 Fexofenadine is an antihistamine pharmaceutical drug used in the treatment of allergy symptoms, such as hay fever, nasal congestion, and urticaria.
CSN12462 Fexofenadine HCl 153439-40-8 Fexofenadine inhibits histamine H1 receptor with IC50 of 246 nM.
CSN10917 Epinastine HCl 108929-04-0 Epinastine HCl is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
CSN10884 Ebrotidine 100981-43-9 Ebrotidine is a competitive H2-receptor antagonist (Ki= 127.5 nM) with a potent antisecretory activity and evidenced gastroprotection.
CSN10883 Ebastine 90729-43-4 Ebastine is a selective H1-histamine receptor antagonist.
CSN10864 Doxylamine succinate salt 562-10-7 Doxylamine Succinate Salt is an antihistamine which inhibits histamine H1 receptors. It can be used as a short-term sedative and anticholinergic agent.
CSN10783 Dexchlorpheniramine Maleate 2438-32-6 Dexchlorpheniramine maleate is an antihistamine, with anticholinergic properties, used to treat allergic conditions.
CSN10775 Desloratadine 100643-71-8 Desloratadine is an antagonist of histamine H1 receptor that is used to treat allergies.
CSN10757 Decloxizine 3733-63-9 Decloxizine is a histamine 1 receptor antagonist.
CSN22573 Cyclizine 2HCl 5897-18-7 Cyclizine is a histamine H1 receptor antagonist of the piperazine class.
CSN10664 Clemizole 442-52-4 Clemizole is an antagonist of H1 histamine receptor that can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.
CSN10663 Clemastine Fumarate 14976-57-9 Clemastine fumarate is a selective antagonist of histamine H1 receptor with IC50 of 3 nM.
CSN12549 Cinnarizine 298-57-7 Cinnarizine, an antihistamine, can block calcium channel and promote cerebral blood flow. It is used to treat post-trauma cerebral symptoms and cerebral arteriosclerosis.
CSN10624 Chlorphenoxamine 77-38-3 Chlorphenoxamine is an antihistamine and anticholinergic and can be used as antipruritic and antiparkinsonian agent.
CSN10076 Chlorpheniramine Maleate 113-92-8 Chlorpheniramine maleate is an antagonist of histamine H1 receptor with IC50 of 12 nM.
CSN23808 Chlorcyclizine HCl 14362-31-3 Chlorcyclizine hydrochloride is a histamine H1 antagonist.
CSN10600 Cetirizine 83881-51-0 Cetirizine, a second-generation antihistamine, is a major metabolite of hydroxyzine, and a racemic selective H1 receptor inverse agonist used in the treatment of allergies, hay fever, angioedema, and urticaria.
CSN12995 Cetirizine 2HCl 83881-52-1 Cetirizine 2HCl, a metabolite of hydroxyzine, is racemic selective and inverse agonist of H1 receptor used in the treatment of allergies and hay fever.
CSN10548 Carbinoxamine Maleate 3505-38-2 Carbinoxamine maleate is a blocker of histamine-H1 receptor with antihistamine and anticholinergic effects.
CSN10500 Buclizine 2HCl 129-74-8 Buclizine 2HCl, the derivative of piperazine, is an antihistamine and anticholinergic agent.
CSN10492 Brompheniramine Maleate 980-71-2 Brompheniramine maleate is an antagonist of histamine H1 receptors.
CSN25269 Bromazine HCl 1808-12-4 Bromazine hydrochloride is an antagonist of histamine H1 receptor.
CSN10402 Bilastine 202189-78-4 Bilastine selectively antagonizes histamine H1 receptor and it is used to treat allergic rhinoconjunctivitis and urticaria.
CSN25225 Betahistine 5638-76-6 Betahistine is a histamine analog and H1 receptor agonist.
CSN24137 Bepotastine 125602-71-3 Bepotastine is a non-sedating and selective antagonist of the histamine 1 (H1) receptor.
CSN10365 Azatadine 3964-81-6 Azatadine is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.
CSN10364 Azatadine Dimaleate 3978-86-7 Azatadine dimaleate is an inhibitor of histamine and cholinergic with IC50 of 6.5 nM and 10 nM, respectively.
CSN10231 Alcaftadine 147084-10-4 Alcaftadine is a high affinity ligand for the H1 receptor, with a pKi (8.5) that is comparable with that of other H1 antihistamines.
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