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AMPAR

AMPAR

货号 产品名 CAS号 信息
CSN13605 β-ODAP 5302-45-4 β-ODAP is an analog of glutamic acid present in Lathyrus sativus (grass pea) that activates AMPA receptors.
CSN17953 ZK200775 161605-73-8 ZK200775 is a highly selective AMPA/kainate antagonist with little activity against NMDA with Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively.
CSN17630 ZK200775 Hydrate 1255517-78-2 ZK200775 is a highly selective AMPA/kainate antagonist with little activity against NMDA and has Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively.
CSN23205 YM 90K HCl 154164-30-4 YM90K hydrochloride is an AMPA receptor antagonist.
CSN23175 UBP 282 544697-47-4 UBP-282 is an α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) and kainate receptor antagonist.
CSN24615 UBP 310 902464-46-4 UBP 310 is an antagonist of GluK1 (formerly GLUK5) kainate receptor with IC50 of 130 nM.
CSN24617 (S)-2-((3-(2-Amino-2-carboxyethyl)-2,6-dioxo-2,3-dihydropyrimidin-1(6H)-yl)methyl)benzoic acid 745055-91-8 UBP 302 is a potent and selective GluK1 (formally GluR5)-subunit containing kainate receptor antagonist with KD of 402 nM.
CSN17301 SYM2206 173952-44-8 SYM2206 is a potent, non-competitive AMPA receptor antagonist (IC50= 2.8 μM).
CSN20167 Selurampanel 912574-69-7 Selurampanel is a competitive AMPA/kainate receptor antagonist drug for epilepsy.
CSN13810 Piracetam 7491-74-9 Piracetam is a cyclic derivative of GABA which works as a positive allosteric modulator of the AMPA receptor.
CSN24155 Philanthotoxin 74 2HCl 1227301-51-0 Philanthotoxin 74 dihydrochloride (PhTx 74) is an AMPAR antagonist; inhibits GluR3 and GluR1 with IC50s of 263 and 296 nM, respectively.
CSN17813 PEPA 141286-78-4 PEPA is an allosteric modulator of AMPA receptors and binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity.
CSN25561 PD-161989 186268-07-5 PD-161989 is an AMPA receptor antagonist.
CSN23006 NPEC-caged-(S)-AMPA 1257323-84-4 NPEC-caged-(S)-AMPA is an agonist at the AMPA receptor.
CSN13580 Noopept 157115-85-0 Noopept is a potent nootropic that improves cognitive ability.
CSN17585 Naspm 122306-11-0 Naspm is a potent and selective Ca2+ permeable AMPA receptor (Ca-perm AMPAR) blocker.
CSN17275 Naspm 3HCl 1049731-36-3 Naspm 3HCl is a potent and selective Ca2+ permeable AMPA receptor (Ca-perm AMPAR) blocker.
CSN16970 LY451395 375345-95-2 LY451395 is a potent and highly selective potentiator of the AMPA receptors.
CSN15793 LY450108 376594-67-1 LY450108 is an alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid (AMPA) receptor potentiator.
CSN20510 LY3130481 1610802-47-5 LY3130481 is the the first α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor antagonist that is dependent on the presence of TARP γ-8. LY3130481 is fully protective against pentylenetetrazole-induced convulsions in rats without the motor impairment associated with non-TARP-dependent AMPA receptor antagonists.
CSN22957 LY 404187 211311-95-4 LY 404187 is a selective positive allosteric modulator of AMPA receptors with IC50s of 0.15, 0.21, 1.66 and 5.65 μM for GluA2i, GluA4i, GluA3i and GluA1i respectively.
CSN11282 Lentinan 37339-90-5 Lentinan, a natural product isolated and purified from shiitake mushroom (Lentinus edodes), is an intravenous anti-tumor polysaccharide isolated from the fruit body of shiitake.
CSN25435 Lentinan 37339-90-5 Lentinan, a natural product isolated and purified from shiitake mushroom (Lentinus edodes), is an intravenous anti-tumor polysaccharide isolated from the fruit body of shiitake.
CSN16600 L-Theanine 3081-61-6 L-theanine is an amino acid found most commonly in tea leaves and binds to ionotropic glutamate receptors in the micromolar range, including the AMPA and kainate receptors and, to a lesser extent, the NMDA receptor.
CSN10840 Kynurenic Acid 492-27-3 Kynurenic Acid is a broad spectrum glutamatergic antagonist which can antagonize NMDA, kainate and AMPA receptors.
CSN24076 JNJ-61432059   2035814-50-5 JNJ-61432059 is an oral active and selective negative modulator of AMPAR associated with trans-membrane AMPAR regulatory protein (TARP) γ-8, with a pIC50 of 9.7 for GluA1/γ-8. Exhibits time- and dose-dependent AMPAR/γ-8 receptor occupancy in mouse hippocampus, resulting in robust seizure protection in corneal kindling and pentylenetetrazole (PTZ) anticonvulsant models[1].
CSN22868 JNJ 55511118 2036081-86-2 JNJ 55511118 is a high affinity and selective negative modulator of AMPA receptors containing TARP-γ8 with Ki of 26 nM.
CSN22846 GYKI 52466 2HCl 102771-26-6 GYKI 52466 2HCl is a selective non-competitive AMPA receptor antagonist with IC50 of 10-20 μM.
CSN21401 L-Quisqualic Acid 52809-07-1 Glutamate receptor agonist acting at AMPA receptors and metabotropic glutamate receptors positively linked to phosphoinositide hydrolysis. Sensitizes neurons in hippocampus to depolarization by L-AP6 (the so called 'quis' effect).
CSN10853 DNQX 2379-57-9 DNQX is a selective non-NMDA iGluR antagonist.
CSN12690 CX-546 215923-54-9 CX-546 is a AMPAR potentiator which can destabilize the desensitized receptor conformation.
CSN22784 CX 614 191744-13-5 CX 614 is a positive allosteric modulator of AMPA receptors.
CSN19847 CP 465022 199655-36-2 CP 465022 HCl is a selective, non-competitive AMPA receptor antagonist (IC50 = 25 nM in rat cortical neurons) that displays potent anticonvulsant activity.
CSN12675 Coluracetam 135463-81-9 Coluracetam a nootropic which can increase the potency of AMPA receptors.
CSN22766 CNQX 115066-14-3 CNQX is a potent and selective non-NMDA iGluR antagonist.
CSN22767 CNQX Disodium Salt 479347-85-8 CNQX Disodium Salt is a AMPA/kainate antagonist and also available as part of the Kainate Receptor.
CSN18250 CMPDA 380607-77-2 CMPDA is a positive allosteric modulator of AMPA receptors with EC50s of 45.4 ± 4.2 nM/63.4 ± 5.6 nM for GluA2i/GluA2o receptor.
CSN17062 CFM-2 178616-26-7 CFM-2 is a selective non-competitive AMPAR antagonist.
CSN24616 ATPA 140158-50-5 ATPA is a selective and potent GluK1 kainate receptor agonist with Ki of 4.3 nM.
CSN10315 Aniracetam 72432-10-1 Aniracetam is an allosteric modulator of AMPAR which can reduce glutamate receptor desensitization and potentiate metabotropic glutamate receptor activity.
CSN10196 Ampalex 154235-83-3 Ampalex is a positive allosteric modulator of AMPAR and is researched as a treatment for Alzheimer's disease.
CSN25263 1-BCP 34023-62-6 1-BCP is can modulate AMPA receptor gated currents and enhence memory.
CSN11876 (S)-Willardiine 21416-43-3 (S)-Willardiine is a potent agonist of AMPA/kainate receptors with EC50 of 44.8 μM.
CSN23429 L-Glutamic Acid 56-86-0 (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system.
CSN22635 (S)-AMPA 83643-88-3 (S)-AMPA is a selective AMPA agonist.
CSN17029 (S)-(-)-5-Fluorowillardiine 140187-23-1 (S)-(-)-5-Fluorowillardiine is a potent and specific AMPAR agonist.
CSN17690 (S)-(-)-5-Fluorowillardiine HCl 1321546-70-6 (S)-(-)-5-Fluorowillardiine HCl is a potent and specific AMPAR agonist.
CSN19840 (RS)-AMPA Hydrobromide 171259-81-7 (RS)-AMPA hydrobromide is a class of glutamate agonist structurally related to ibotenic acid.
CSN22625 (R)-3,4-DCPG 201730-10-1 (R)-3,4-DCPG is a AMPA receptor antagonist.
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