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NK Receptor

NK Receptor

货号 产品名 CAS号 信息
CSN19815 Tradipitant 622370-35-8 Tradipitant is the 2nd generation neurokinin-1 receptor antagonist, which showed activity in preclinical anxiety models.
CSN13678 Talnetant 174636-32-9 Talnetant is a potent and selective NK3 receptor antagonist (ki=1.4 nM, hNK-3-CHO), and is 100-fold selective for the hNK-3 versus hNK-2 receptor, with no affinity for the hNK-1 at concentrations up to 100 μM.
CSN18094 Talnetant HCl 204519-66-4 Talnetant hydrochloride is a potent and selective NK3 receptor antagonist (ki=1.4 nM, hNK-3-CHO), 100-fold selective for the hNK-3 versus hNK-2 receptor, with no affinity for the hNK-1 at concentrations up to 100 μM.
CSN22504 Serlopitant 860642-69-9 Serlopitant is a selective Neurokinin-1 (NK-1) receptor antagonist.
CSN17283 SB-222200 174635-69-9 SB-222200 is a selective, reversible and competitive antagonist of human NK-3 receptor (Ki=4.4 nM) that effectively crosses the blood-brain barrier.
CSN22503 Saredutant 142001-63-6 Saredutant is a selective NK2 receptor antagonist.
CSN19715 Rolapitant 552292-08-7 Rolapitant inhibits CYP2D6, breast cancer resistance protein (BCRP), and Neurokinin (NK)1 Receptor.
CSN16098 Rolapitant HCl H2O 914462-92-3 Rolapitant HCl H2O is a long-acting, selective and competitive NK-1 receptor antagonist.
CSN18026 NKP608 177707-12-9 NKP608 is a non-peptidic derivative of 4-aminopiperidine which acts as a selective, specific and potent antagonist at the neurokinin-1 (NK-1) receptor both in vitro (IC50=2.6 nM) and in vivo.
CSN16120 Netupitant 290297-26-6 Netupitant a potent and highly selective NK1 receptor antagonist with Ki of 0.95 nM.
CSN19286 MLE4901 941690-55-7 MLE4901 is an antagonist of Neurokinin 3 Receptor and a potential drug for Polycystic ovary syndrome and menopausal hot flushes.
CSN22464 MEN 15596 522664-63-7 MEN 15596 is a potent and selective tachykinin NK2 receptor antagonist with a pKi of 10.1.
CSN17887 Maropitant 147116-67-4 Maropitant is a neurokinin (NK1) receptor antagonist.
CSN18008 Fosaprepitant 172673-20-0 Fosaprepitant is a neurokinin-1 receptor antagonist for the prevention of chemotherapy-induced nausea and vomiting.
CSN12336 Fosaprepitant Dimeglumine 265121-04-8 Fosaprepitant Dimeglumine is a prodrug for aprepitant which is a selective and high-affinity antagonist of NK1 receptor.
CSN10324 Aprepitant 170729-80-3 Aprepitant is a selective and high-affinity neurokinin-1 receptor antagonist with IC50 of 0.1 nM.
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