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Pim

Pim

货号 产品名 CAS号 信息
CSN22892 TP-3654 1361951-15-6 TP-3654 is a selective Pim kinase inhibitor with Ki values of 5nM, 239nM and 42nM for Pim-1, Pim-2 and Pim-3, respectively, as well as with an average EC50 of 67nM for cellular PIM-1 inhibition in the PIM-1/BAD overexpression system and with moderate potency to FLT3.
CSN15804 SMI-4a 438190-29-5 SMI-4a is a potent inhibitor of Pim1 with IC50 of 17 nM, modestly potent to Pim-2, does not significantly inhibit any other serine/threonine- or tyrosine-kinases.
CSN17458 Pim1 AKK1-IN-1 1093222-27-5 Pim1 AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively and also inhibits MPSK1 and TNIK.
CSN19123 PIM-447 1210608-43-7 PIM-447 is pan-PIM kinase inhibitor, including Moloney Murine Leukemia (PIM)1, 2, and 3 Kinase.
CSN19124 PIM-447 2HCl 1820565-69-2 PIM-447 2HCl is pan-PIM kinase inhibitor, including Moloney Murine Leukemia (PIM)1, 2, and 3 Kinase.
CSN20612 pan-PIM Inhibitor CS11 2139294-71-4 pan-PIM inhibitor CS11 is a pan-PIM kinase inhibitor, which inhibits PIM1 and PIM2 with IC50 of 1 nM and 6 nM, respectively.
CSN17786 M-110 1395048-49-3 M-110 is a highly selective inhibitor of PIM kinases and inhibits the proliferation of prostate cancer cell lines with IC50s of 0.6 to 0.9 μM, with no activity on normal human peripheral blood mononuclear cells up to 40 μM.
CSN20019 GNE-955 1527523-39-2 GNE-955 is a pan-Pim inhibitor with bioavailability bioavailability and a potential hematologic–oncology use.
CSN17835 GDC-0339 1428569-85-0 GDC-0339 is a Pim kinase inhibitor with IC50 of 43.6 nM for BaF3 PIM1.
CSN16136 CX-6258 1202916-90-2 CX-6258 is a selective and potent Pim inhibitor with IC50 values of 5nM, 25nM and 16nM for Pim-1, Pim-2 and Pim-3 (measured by SAR assay), respectively.
CSN19180 CX-6258 HCl 1353859-00-3 CX-6258 HCl is a potent, orally efficacious pan-Pim kinase inhibitor with IC50 of 5 nM, 25 nM and 16 nM for Pim1, Pim2, and Pim3, respectively.
CSN17740 CX-6258 HCl H2O 1353858-99-7 CX-6258 HCl hydrate is the HCl hydrate form of CX-6258. CX-6258 is a selective and potent Pim inhibitor with IC50 values of 5nM, 25nM and 16nM for Pim-1, Pim-2 and Pim-3 (measured by SAR assay), respectively.
CSN19008 (1S,3R,5R)-PIM447 2HCl N/A (1S,3R,5R)-PIM447 2HCl an PIM inhibitor with IC50 values of 0.095 μM for Pim1, 0.522 μM for Pim2 and 0.369 μM for Pim3.
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