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货号 产品名 CAS号 信息
CSN10426 β-Estradiol 17-acetate 1743-60-8 β-Estradiol 17-acetate is a metabolite of estradiol.
CSN17211 α-Estradiol 57-91-0 α-Estradiol is an endogenous estrogen receptor ligand (Ki values are 0.2 and 1.2 nM for ERα and ERβ receptors respectively).
CSN16334 XCT790 725247-18-7 XCT-790 is an agonist of estrogen related receptor alpha (ERRα) and can induce death of cancer cells resistant to chemotherapy.
CSN17140 Ulipristal 159811-51-5 Ulipristal is a selective progesterone receptor modulator (SPRM) for inhibiting or delaying ovulation.
CSN16793 Toremifene Citrate 89778-27-8 Toremifene citrate is a modulator of estrogen receptor that is used in the treatment of advanced breast cancer.
CSN11752 Tesmilifene 98774-23-3 Tesmilifene is an agent that augments cytotoxicity of various chemotherapeutic agents both in vitro and in vivo.
CSN16637 Tectoridin 611-40-5 Tectoridin, an isoflavone, is a natural product isolated and purified from the rhizomes of belamcanda chinensis (L.) DC. with anti-inflammatory activities.
CSN12029 Tamoxifen Citrate 54965-24-1 Tamoxifen citrate (ICI 46474) is a competitive antagonist of the estrogen receptor via its active metabolite 4-hydroxytamoxifen.
CSN13942 SNG-1153 1446712-19-1 SNG1153, a derivate of icaritin, is a modulator of ER-α36 and an inducer of phosphorylation of β-catenin.
CSN12984 Raloxifene HCl 82640-04-8 Raloxifene hydrochloride is an selective antagonist of estrogen receptor that exhibits estrogenic activity in bone cells without stimulating breast or uterine tissues.
CSN11817 Quinestrol 152-43-2 Quinestrol is a synthetic estrogen which is used in hormone replacement therapy.
CSN15897 Ospemifene 128607-22-7 Ospemifene is a non-hormonal estrogen receptor modulator (SERM) with IC50 values of 827 nM and 1633 nM for ERα and ERβ. Ospemifene is one of the active metabolites of toremifene.
CSN13823 Nafoxidine HCl 1847-63-8 Nafoxidine hydrochloride is a non-steroidal selective estrogen receptor modulator (SERM) or partial antiestrogen of the triphenylethylene group that was developed for the treatment of advanced breast cancer.
CSN11387 Mestranol 72-33-3 Mestranol is an agonist of estrogen receptor. It is used as contraceptives.
CSN23280 Lynestrenol 52-76-6 Lynestrenol is a progesterone receptor agonist. It is synthetic progestational hormone.
CSN16424 Licochalcone A 58749-22-7 Licochalcone A, an estrogenic flavanoid, can be an inhibitor of p-glycoprotein and has anti-inflammatory actions.
CSN16955 Lasofoxifene Tartrate 190791-29-8 Lasofoxifene tartrate, a non-steroidal compound, is a modulator of estrogen receptor.
CSN16382 Kaempferol 520-18-3 Kaempferol acts as an inverse agonist that directly binds ERRα and ERRγ. It is a natural flavonol with antitumor activity.
CSN11148 Hexestrol 84-16-2 Hexestrol can bind to ERα and ERβ selectively with EC50 of 0.07 nM and 0.175 nM respectively.
CSN15815 GDC-0810 1365888-06-7 GDC-0810 is an orally bioavailable selective estrogen receptor degrader (SERD) with IC50 of 0.7 nM.
CSN11061 Fulvestrant 129453-61-8 Fulvestrant is a representative pure antiestrogen and a Selective Estrogen Receptor Down-regulator (SERD) with IC50 of 0.94 nM.
CSN10968 Etonogestrel 54048-10-1 Etonogestrel, a steroidal progestin, is used in hormonal contraceptives.
CSN10946 Ethisterone 434-03-7 Ethisterone is a progestogen hormone that could be used to treat prostate cancer.
CSN16404 Ethynyl Estradiol 57-63-6 Ethinyl Estradiol is an estrogen used in formulations of combined contraceptive pills.
CSN10938 Piperazine Estronesulfate 7280-37-7 Estropipate, deriving from estrogen, is used to treat symptoms of menopause and to prevent osteoporosis.
CSN16386 Estrone 53-16-7 Estrone is an estrogenic hormone secreted by the ovary as well as adipose tissue.
CSN10937 Estriol 50-27-1 Estriol is G-protein coupled estrogen receptor antagonist in estrogen receptor-negative breast cancer cells. It is a major urinary estrogen which is largely produced by the placenta during pregnancy.
CSN10936 Estradiol Valeate 979-32-8 Estradiol valerate is a synthetic estrogen. Formulations containing estradiol valerate with other steroid hormones have been used to treat endometriosis.
CSN17215 Estradiol 50-28-2 Estradiol is an estrogenic hormone that is produced in the ovaries, placenta, testis.
CSN10771 Estradiol Cypionate 313-06-4 Estradiol cypionate is a synthetic ester. Compared to other commonly used estradiol esters, via the intramuscular route, estradiol cypionate is found to have the longest duration of action with a duration of ~11 days,
CSN10935 Estradiol Benzoate 50-50-0 Estradiol benzoate is an estradiol analog which binds to the human, murine and chicken ERα with IC50 of 22-28 nM.
CSN12284 Equol 531-95-3 Equol, a non-steroidal estrogen, is a selective agonist of ERβ. It is produced from the metabolism of the isoflavonoid phytoestrogen daidzen by human intestinal microflora.
CSN17408 Endoxifen Z-Isomer HCl 1032008-74-4 Endoxifen Z-isomer hydrochloride is the most important Tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα). Endoxifen Z-isomer hydrochloride inhibits hERG tail currents at 50 mV in a concentration-dependent manner with IC50 values of 1.6 μM.
CSN17474 Endoxifen Z-Isomer 112093-28-4 Endoxifen is the most important tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα).
CSN17545 Endoxifen E-isomer HCl 1197194-61-8 Endoxifen E-isomer hydrochloride is a tamoxifen metabolite and potent Selective Estrogen Response Modifier (SERM).
CSN10880 DY131 95167-41-2 DY131 is an agonist of ERRβ/ERRγ receptor (EC50 = 130 nM) with minimal activity for ERRα, ERα and ERβ.
CSN15920 DPN 1428-67-7 DPN is a non-steroidal estrogen receptor β (ER β) selective ligand.
CSN10805 Diethylstilbestrol 56-53-1 Diethylstilbestrol is a synthetic nonsteroidal estrogen that produces all the pharmacological and therapeutic effects of natural estradiol. It is mainly used for functional hemorrhage caused by estrogen hypoxia and hormonal imbalance, amenorrhea.
CSN10799 Dienestrol 84-17-3 Dienestrol is an agonist of estrogen receptor which is used for the treatment of menopausal symptoms.
CSN17329 Daidzein 486-66-8 Daidzein can act as an inhibitor of tyrosine kinase and an activator of estrogen receptor. It is inactive analogue of genistein.
CSN10717 Cyclofenil 2624-43-3 Cyclofenil is a modulator of non-steroidal estrogen receptor. The selectivity to ERβ is better than ERα.
CSN17299 Clomiphene Citrate 50-41-9 Clomifene citrate is a modulator of estrogen receptor Erα (Ki = 0.9 nM) and Erβ (Ki = 1.2 nM). It has been used to treat ovulation induction.
CSN10623 Chlorotrianisene 569-57-3 Chlorotrianisene, a synthetic and non-steroidal estrogen, is a modulator of estrogen receptor.
CSN12297 Bazedoxifene 198481-32-2 Bazedoxifene is a selective estrogen receptor modulator (SERM) currently in development for osteoporosis prevention and treatment.
CSN10382 Bazedoxifene Acetate 198481-33-3 Bazedoxifene acetate can selectively modulate estrogen receptor (SERM), the IC50 values are 26 nM and 99 nM for ERα and ERβ respectively.
CSN15663 Bavachin 19879-32-4 Bavachin, a flavonoid phytoestrogen, can activate the estrogen receptors ERα (EC50 = 320 nM) and ERβ (EC50 = 680 nM).
CSN17980 AZD9496 1639042-08-2 AZD9496 is a selective antagonist of estrogen receptor Erα (IC50 = 0.28 nM).
CSN13183 17A-Hydroxyprogesterone 68-96-2 17α-hydroxyprogesterone is an endogenous progestogen. It is also a chemical intermediate for many other endogenous steroids.
CSN17213 17-Caproxyprogesterone 630-56-8 17-Caproxyprogesterone is a steroidal progestin. It is a synthetic ester derivative of 17α-hydroxyprogesterone.
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