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货号 产品名 CAS号 信息
CSN10426 β-Estradiol 17-acetate 1743-60-8 β-Estradiol 17-acetate is a metabolite of estradiol.
CSN17211 α-Estradiol 57-91-0 α-Estradiol is an endogenous estrogen receptor ligand (Ki values are 0.2 and 1.2 nM for ERα and ERβ receptors respectively).
CSN16334 XCT790 725247-18-7 XCT-790 is an agonist of estrogen related receptor alpha (ERRα) and can induce death of cancer cells resistant to chemotherapy.
CSN17140 Ulipristal 159811-51-5 Ulipristal is a selective progesterone receptor modulator (SPRM) for inhibiting or delaying ovulation.
CSN11752 Tesmilifene 98774-23-3 Tesmilifene is an agent that augments cytotoxicity of various chemotherapeutic agents both in vitro and in vivo.
CSN16637 Tectoridin 611-40-5 Tectoridin, an isoflavone, is a natural product isolated and purified from the rhizomes of belamcanda chinensis (L.) DC. with anti-inflammatory activities.
CSN25280 SR19881 2213490-89-0 SR19881 is a ERRγ agonist.
CSN13942 SNG-1153 1446712-19-1 SNG1153, a derivate of icaritin, is a modulator of ER-α36 and an inducer of phosphorylation of β-catenin.
CSN23201 Y 134 849662-80-2 Selective estrogen receptor modulator (SERM), selective for ERα
CSN11817 Quinestrol 152-43-2 Quinestrol is a synthetic estrogen which is used in hormone replacement therapy.
CSN15897 Ospemifene 128607-22-7 Ospemifene is a non-hormonal estrogen receptor modulator (SERM) with IC50 values of 827 nM and 1633 nM for ERα and ERβ. Ospemifene is one of the active metabolites of toremifene.
CSN13823 Nafoxidine HCl 1847-63-8 Nafoxidine HCl is a non-steroidal selective estrogen receptor modulator (SERM) or partial antiestrogen of the triphenylethylene group that was developed for the treatment of advanced breast cancer.
CSN16424 Licochalcone A 58749-22-7 Licochalcone A, an estrogenic flavanoid, can be an inhibitor of p-glycoprotein and has anti-inflammatory actions.
CSN16382 Kaempferol 520-18-3 Kaempferol acts as an inverse agonist that directly binds ERRα and ERRγ. It is a natural flavonol with antitumor activity.
CSN11148 Hexestrol 84-16-2 Hexestrol can bind to ERα and ERβ selectively with EC50 of 0.07 nM and 0.175 nM respectively.
CSN21091 GDC-0927 1642297-01-5 GDC-0927, also known as SRN-927, is a next-generation oral SERD, appears to have greater potential than GDC-0810 to be a best-in-class SERD molecule.
CSN15815 GDC-0810 1365888-06-7 GDC-0810 is an orally bioavailable selective estrogen receptor degrader (SERD) with IC50 of 0.7 nM.
CSN10968 Etonogestrel 54048-10-1 Etonogestrel, a steroidal progestin, is used in hormonal contraceptives.
CSN16404 Ethynyl Estradiol 57-63-6 Ethynyl Estradiol is an estrogen used in formulations of combined contraceptive pills.
CSN10946 Ethisterone 434-03-7 Ethisterone is a progestogen hormone that could be used to treat prostate cancer.
CSN10938 Estropipate 7280-37-7 Estropipate, deriving from estrogen, is used to treat symptoms of menopause and to prevent osteoporosis.
CSN16386 Estrone 53-16-7 Estrone is an estrogenic hormone secreted by the ovary as well as adipose tissue.
CSN25302 Estrogen receptor modulator 1 63676-22-2 Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM), with a pIC50 of 0.46. It has been found to be both estrogenic and antiproliferative in ER-positive endocrine-resistant breast cancer cell lines that overexpress protein kinase C alpha (PKCα).
CSN10937 Estriol 50-27-1 Estriol is G-protein coupled estrogen receptor antagonist in estrogen receptor-negative breast cancer cells. It is a major urinary estrogen which is largely produced by the placenta during pregnancy.
CSN10936 Estradiol Valeate 979-32-8 Estradiol Valeate is a synthetic estrogen. Formulations containing estradiol valerate with other steroid hormones have been used to treat endometriosis.
CSN17215 Estradiol 50-28-2 Estradiol is an estrogenic hormone that is produced in the ovaries, placenta, testis.
CSN10771 Estradiol Cypionate 313-06-4 Estradiol cypionate is a synthetic ester. Compared to other commonly used estradiol esters, via the intramuscular route, estradiol cypionate is found to have the longest duration of action with a duration of ~11 days,
CSN12284 Equol 531-95-3 Equol, a non-steroidal estrogen, is a selective agonist of ERβ. It is produced from the metabolism of the isoflavonoid phytoestrogen daidzen by human intestinal microflora.
CSN17408 Endoxifen Z-Isomer HCl 1032008-74-4 Endoxifen Z-isomer HCl is the most important Tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα). Endoxifen Z-isomer HCl inhibits hERG tail currents at 50 mV in a concentration-dependent manner with IC50 values of 1.6 μM.
CSN17474 Endoxifen Z-Isomer 112093-28-4 Endoxifen is the most important tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα).
CSN17545 Endoxifen E-isomer HCl 1197194-61-8 Endoxifen E-isomer HCl is a tamoxifen metabolite and potent Selective Estrogen Response Modifier (SERM).
CSN10880 DY131 95167-41-2 DY131 is an agonist of ERRβ/ERRγ receptor (EC50 = 130 nM) with minimal activity for ERRα, ERα and ERβ.
CSN15920 DPN 1428-67-7 DPN is a non-steroidal estrogen receptor β (ER β) selective ligand.
CSN10805 Diethylstilbestrol 56-53-1 Diethylstilbestrol is a synthetic nonsteroidal estrogen that produces all the pharmacological and therapeutic effects of natural estradiol. It is mainly used for functional hemorrhage caused by estrogen hypoxia and hormonal imbalance, amenorrhea.
CSN10799 Dienestrol 84-17-3 Dienestrol is an agonist of estrogen receptor which is used for the treatment of menopausal symptoms.
CSN17329 Daidzein 486-66-8 Daidzein can act as an inhibitor of tyrosine kinase and an activator of estrogen receptor. It is inactive analogue of genistein.
CSN14669 Cristacarpin 74515-47-2 Cristacarpin, a natural product isolated and purified from the herbs of Erythrina burana, exhibits moderate but selective activity towards DNA repair-deficient yeast mutants, and promotes endoplasmic reticulum (ER) stress, leading to sub-lethal reactive oxygen species (ROS) generation and which eventually terminates by triggering senescence in pancreatic and breast cancer cells through blocking the cell cycle in the G1 phase.
CSN10623 Chlorotrianisene 569-57-3 Chlorotrianisene, a synthetic and non-steroidal estrogen, is a modulator of estrogen receptor.
CSN18837 Bazedoxifene HCl 198480-56-7 Bazedoxifene is a third generation selective estrogen receptor modulator (SERM).
CSN12297 Bazedoxifene 198481-32-2 Bazedoxifene is a selective estrogen receptor modulator (SERM) currently in development for osteoporosis prevention and treatment.
CSN10382 Bazedoxifene Acetate 198481-33-3 Bazedoxifene acetate can selectively modulate estrogen receptor (SERM), the IC50 values are 26 nM and 99 nM for ERα and ERβ respectively.
CSN15663 Bavachin 19879-32-4 Bavachin, a flavonoid phytoestrogen, can activate the estrogen receptors ERα (EC50 = 320 nM) and ERβ (EC50 = 680 nM).
CSN13183 17A-Hydroxyprogesterone 68-96-2 17α-hydroxyprogesterone is an endogenous progestogen. It is also a chemical intermediate for many other endogenous steroids.
CSN17213 17-Caproxyprogesterone 630-56-8 17-Caproxyprogesterone is a steroidal progestin. It is a synthetic ester derivative of 17α-hydroxyprogesterone.
CSN25405 (±)-Equol 94105-90-5
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