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SRPK

SRPK

货号 产品名 CAS号 信息
CSN19078 WNK463 2012607-27-9 WNK463 is a potant With-No-Lysine (WNK) kinase inhibitor with IC50s of 5/1/6/9 nM for WNK1/2/3/4.
CSN23723 WNK-IN-11 2123489-30-3 WNK-IN-11 is a potent, selective and orally active inhibitor of WNK1 kinase with IC50 of 6 nM.
CSN13762 SRPIN340 218156-96-8 SRPIN340 is an inhibitor of serine/arginine-rich protein kinase SRPK1 with IC50 of 0.89 μM.
CSN23673 SPHINX31 1818389-84-2 SPHINX31 is a potent and selective inhibitor of serine/arginine-rich protein kinase 1 (SRPK1), with an IC50 of 5.9 nM. SPHINX31 inhibits phosphorylation of serine/arginine-rich splicing factor 1 (SRSF1). SPHINX31 is a potential topical therapeutic for neovascular eye disease[1].
CSN23063 rac-CCT 250863 1364269-06-6 rac-CCT-250863 is a potent Nek2 inhibitor. exhibiting selectivity for Nek2 over PLK1, MPS1, Cdk2 and Aurora A.
CSN20434 PROTAC TBK1 C3i 2052306-13-3 PROTAC TBK1 C3i is a potent hit (TBK1 DC50 = 12 nM, Dmax = 96%) with excellent selectivity against a related kinase IKKε, which was further used as a chemical tool to assess TBK1 as a target in mutant K-Ras cancer cells.
CSN17458 Pim1 AKK1-IN-1 1093222-27-5 Pim1 AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively and also inhibits MPSK1 and TNIK.
CSN17627 AR-13324 HCl 1253952-02-1 Netarsudil primarily targets cells in the conventional outflow tract, efficiently decreasing IOP in both human and non-human primate eyes.
CSN23000 NCL 00017509 1507367-00-1 NCL 00017509 is a potent and reversible NIMA related kinase 2 (Nek2) inhibitor with IC50 of 56 nM.
CSN17686 MK2-IN-1 1314118-92-7 MK2-IN-1 is a potent and selecitve MAPKAPK2 (MK2) inhibitor (IC50=0.11 μM) with a non-ATP competitive binding mode.
CSN17687 MK2-IN-1 HCl 1314118-94-9 MK2-IN-1 HCl is a non-ATP competitive inhibitor of MAPKAPK2 (MK2) with IC50 of 0.11 μM.
CSN18951 ILK-IN-2 2070015-22-2 ILK-IN-2 is a ILK inhibitor.
CSN17699 ILK-IN-1 1333146-24-9 ILK-IN-1 is an ILK inhibitor with IC50 of 0.6 μM.
CSN24084 GSK8612 2361659-62-1 GSK8612 is a potent and highly selective Tank-binding Kinase-1 (TBK1) inhibitor with pIC50 of 6.8 for recombinant TBK1.
CSN15402 Cycloheterophyllin 36545-53-6 Cycloheterophyllin, a natural product isolated and purified from the herbs of Artocarpus heterophyllus, exerts a concentration-dependent inhibition of neutrophil cytosolic protein kinase C (PKC) and rat brain PKC by the O2- generation in rat neutrophils, but has no effect on porcine heart protein kinase A (PKA).
CSN20021 Bryostatin 1 83314-01-6 Bryostatin 1 is a Protein kinase C (PKC) activator that binds with high affinity (Ki = 1.35 nM).
CSN12528 4μ8C 14003-96-4 4μ8C is a potent and selective IRE1 Rnase inhibitor with IC50 of 76 nM.
CSN24165 GSK8612 2361659-62-1
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