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GSK-3

GSK-3

货号 产品名 CAS号 信息
CSN15707 TWS119 601514-19-6 TWS119 is inhibitor of glycogen synthase kinase-3β with IC50 of 30 nM.
CSN16043 Tideglusib   865854-05-3 Tideglusib is an irreversible GSK-3 inhibitor with IC50 of 5 nM and 60 nM for GSK-3βWT (1 h preincubation) and GSK-3βC199A (1 h preincubation), respectively.
CSN19500 TDZD-8 327036-89-5 TDZD-8, the derivative of thiadiazolidinone, is a selective inhibitor of GSK-3. It inhibits GSK-3β with IC50 of 2 μM.
CSN16568 SB-415286 264218-23-7 SB-415286 is an ATP-competitive inhibitor of GSK3α/GSK3β with IC50 of 78 nM and Ki of 31 nM.
CSN12268 SB-216763 280744-09-4 SB-216763 is potent and selective glycogen synthase kinase-3 (GSK-3) inhibitor (Ki = 9 nM) and competes with ATP.
CSN18355 LY2090314     603288-22-8 LY2090314 is a potent inhibitor of glycogen synthase kinase-3 (GSK-3) with IC50s of 1.5 nM and 0.9 nM for GSK-3α and GSK-3β respectively.
CSN22886 Lithium Carbonate 554-13-2 Lithium Carbonate inhibits GSK-3 in vivo.
CSN11250 Kenpaullone 142273-20-9 Kenpaullone is an ATP-competitive inhibitor of CDK1/cyclin B (IC50 = 0.4 µM), CDK2/cyclin A (IC50 = 0.68 µM), CDK5/p25 (IC50 = 0.85 µM), lymphocyte kinase (IC50 = 0.47 µM) , and GSK-3β (C50 = 0.23 μM).
CSN11201 Indirubin-3'-Monoxime 160807-49-8 Indirubin-3'-monoxime is a powerful inhibitor of GSK-3β with IC50 of 22nM, also inhibits CDK1/5 (IC50 = 180/100 nM).
CSN17487 IM-12 1129669-05-1 IM-12 is a GSK-3β inhibitor with IC50 of 53 nM.
CSN18354 GSK-3 Inhibitor 1 603272-51-1 GSK-3 inhibitor 1 is a potent GSK-3 inhibitor.
CSN17624 CP21R7 125314-13-8 CP21R7 is a slective inhibitor of GSK-3β.
CSN19149 CHIR-99021 3HCl 1782235-14-6 CHIR-99021 trihydrochloride is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM, showing > 500-fold selectivity for GSK-3 versus its closest homologs CDC2 and ERK2, as well as other protein kinases.
CSN13470 CHIR-99021     252917-06-9 CHIR-99021 is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM, exhibiting > 500-fold selectivity for GSK-3 versus its closest homologs CDC2 and ERK2, as well as other protein kinases.
CSN19176 CHIR-99021 HCl 1797989-42-4 CHIR-99021 hydrochloride is hydrochloride of CHIR-99021, which is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM and shows greater than 500-fold selectivity for GSK-3 versus its closest homologs Cdc2 and ERK2.
CSN20636 CHIR-98024 556813-39-9 CHIR-98014 is a reversible inhibitor of GSK3α and GSK3β with IC50 of 0.65 nM and 0.58 nM, respectively.
CSN23355 CHIR-98014 252935-94-7 CHIR-98014 (CT98014) is highly selective aminopyrimidine-derivatived inhibitor of GSK-3 with IC50 of 650nM and 580nM for GSK-3 and GSK-3(measured by kinase assays), respectively, and exhibits >1000-fold selectivity for GSK-3 over closely related kinases, such as cdc2.
CSN16227 BIO-Acetoxime 667463-85-6 BIO-acetoxime is an inhibitor of GSK3α and GSK3β with IC50 of 10 nM.
CSN16080 BIO 667463-62-9 BIO is an inhibitor of GSK-3 and CDK1–cyclinB complex. The IC50s of GSK-3αβ, CDK1, CDK5 are 5 nM, 320 nM and 83 nM, respectively.
CSN13082 Bikinin 188011-69-0 Bikinin acts as an ATP-competitive inhibitor of arabidopsis GSK-3 and effective activator of brassinosteroid (BR) signaling.
CSN13894 AZD2858 486424-20-8 AZD2858 is an inhibitor of GSK-3 with IC50 of 68 nM that can inhibit the tau phosphorylation of S396 site and activate Wnt signaling pathway.
CSN16226 AZD1080   612487-72-6 AZD1080 is a selective, orally active, brain permeable GSK3 inhibitor of GSK3α and GSK3β with Ki of 6.9 nM and 31 nM, respectively, shows > 14-fold selectivity against CDK2, CDK5, CDK1 and Erk2.
CSN15984 AR-A014418 487021-52-3 AR-A014418 is a selective inhibitor of GSK3β with IC50 of 104 ± 27 nM.
CSN23598 5-Bromoindole 10075-50-0 5-bromoindole is an inhibitor of glycogen synthase kinase 3 (GSK-3), it can be used as important pharmaceutical chemical intermediate.
CSN18742 1-Azakenpaullone 676596-65-9 1-Azakenpaullone is a potent and selective GSK-3β inhibitor with IC50 of 18 nM, > 100-fold selectivity over CDK1/cyclin B and CDK5/p25.
CSN22657 A 1070722 1384424-80-9
CSN22644 2B-(SP) 186901-17-7
CSN23154 TC-G 24 1257256-44-2
CSN23157 TCS 2002 1005201-24-0
CSN23173 TWS 119 1507095-58-0
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