优势价格
快速发货
品质保证
技术支持
400-920-2911 sales@csnpharm.cn
ERR
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN17211 | α-Estradiol | 57-91-0 | α-Estradiol is an endogenous estrogen receptor ligand (Ki values are 0.2 and 1.2 nM for ERα and ERβ receptors respectively). |
| CSN16334 | XCT790 | 725247-18-7 | XCT-790 is an agonist of estrogen related receptor alpha (ERRα) and can induce death of cancer cells resistant to chemotherapy. |
| CSN20458 | WAY-200070 | 440122-66-7 | WAY200070 selectively activates ERβ (EC50 = 2 nM) receptor over ERα (EC50 = 155 nM). It shows anti-depressive and anti-anxiolytic activities. |
| CSN17140 | Ulipristal | 159811-51-5 | Ulipristal is a selective progesterone receptor modulator (SPRM) for inhibiting or delaying ovulation. |
| CSN19977 | tracheloside | 33464-71-0 | Tracheloside, a natural product isolated and purified from the herbs of Trachelospermum jasminoides (Lindl.) Lem., significantly decreases the activity of alkaline phosphatase (AP), an estrogen-inducible marker enzyme, with an IC50 value of 0.31 mg/mL, a level of inhibition comparable to that of tamoxifen (IC50 = 0.43 mg/mL). |
| CSN21231 | MK-6913 | 1398510-92-3 | Tetrahydrofluoroene 52 is a potent and selective estrogen receptor β agonist. |
| CSN11752 | DPPE Fumarate | 98774-23-3 | Tesmilifene is an agent that augments cytotoxicity of various chemotherapeutic agents both in vitro and in vivo. |
| CSN16637 | Tectoridin | 611-40-5 | Tectoridin, an isoflavone, is a natural product isolated and purified from the rhizomes of belamcanda chinensis (L.) DC. with anti-inflammatory activities. |
| CSN13942 | 3,5,7-Trihydroxy-8-(3-methylbut-2-en-1-yl)-2-(4-(trifluoromethyl)phenyl)-4H-chromen-4-one | 1446712-19-1 | SNG1153, a derivate of icaritin, is a modulator of ER-α36 and an inducer of phosphorylation of β-catenin. |
| CSN11817 | Quinestrol | 152-43-2 | Quinestrol is a synthetic estrogen which is used in hormone replacement therapy. |
| CSN18316 | Prinaberel | 524684-52-4 | Prinaberel is an agonist of ERβ. |
| CSN19690 | PHTPP | 805239-56-9 | PHTPP has selective antagonism of estrogen ERβ receptor . |
| CSN20291 | Ormeloxifene | 31477-60-8 | Ormeloxifene, an estrogen receptor regulator, suppresses prostate tumor growth and metastatic phenotypes via inhibition of oncogenic β-catenin signaling and EMT progression |
| CSN21337 | Nitromifene | 10448-84-7 | Nitromifene is an antagonist of estrogen receptor (ER). |
| CSN13823 | 1-(2-(4-(6-Methoxy-2-phenyl-3,4-dihydronaphthalen-1-yl)phenoxy)ethyl)pyrrolidine hydrochloride | 1847-63-8 | Nafoxidine HCl is a non-steroidal selective estrogen receptor modulator (SERM) or partial antiestrogen of the triphenylethylene group that was developed for the treatment of advanced breast cancer. |
| CSN11387 | Mestranol | 72-33-3 | Mestranol is an agonist of estrogen receptor. It is used as contraceptives. |
| CSN21092 | LSZ-102 | 2135600-76-7 | LSZ102 is a potent ERα antagonist and degrader. LSZ102 showed ERα degradation IC50 = 0.2 nM. LSZ102 demonstrated IC50 for MCF-7 cells = 1.7 nM. Upon administration of LSZ102, this agent binds to the ER and induces the degradation of the receptor. This prevents ER activation and ER-mediated signaling, and inhibits the growth and survival of ER-expressing cancer cells. |
| CSN16424 | Licochalcone A | 58749-22-7 | Licochalcone A, an estrogenic flavanoid, can be an inhibitor of p-glycoprotein and has anti-inflammatory actions. |
| CSN16955 | Lasofoxifene tartrate | 190791-29-8 | Lasofoxifene tartrate, a non-steroidal compound, is a modulator of estrogen receptor. |
| CSN16382 | 3,5,7-Trihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one | 520-18-3 | Kaempferol acts as an inverse agonist that directly binds ERRα and ERRγ. It is a natural flavonol with antitumor activity. |
| CSN11148 | rel-4,4'-((3R,4S)-Hexane-3,4-diyl)diphenol | 84-16-2 | Hexestrol can bind to ERα and ERβ selectively with EC50 of 0.07 nM and 0.175 nM respectively. |
| CSN15815 | Brilanestrant | 1365888-06-7 | GDC-0810 is an orally bioavailable selective estrogen receptor degrader (SERD) with IC50 of 0.7 nM. |
| CSN16404 | Ethynylestradiol | 57-63-6 | Ethynyl Estradiol is an estrogen used in formulations of combined contraceptive pills. |
| CSN17215 | (8R,9S,13S,14S,17S)-13-Methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthrene-3,17-diol | 50-28-2 | Estradiol is an estrogenic hormone that is produced in the ovaries, placenta, testis. |
| CSN12284 | (-)-(S)-Equol | 531-95-3 | Equol, a non-steroidal estrogen, is a selective agonist of ERβ. It is produced from the metabolism of the isoflavonoid phytoestrogen daidzen by human intestinal microflora. |
| CSN21329 | Eprotirome | 355129-15-6 | Eprotirome is a liver-selective thyroid hormone receptor agonist. |
| CSN17408 | Endoxifen Z-isomer HCl | 1032008-74-4 | Endoxifen Z-isomer HCl is the most important Tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα). Endoxifen Z-isomer HCl inhibits hERG tail currents at 50 mV in a concentration-dependent manner with IC50 values of 1.6 μM. |
| CSN17474 | Endoxifen (Z-isomer) | 112093-28-4 | Endoxifen is the most important tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα). |
| CSN19261 | Endoxifen HCl | 1197194-41-4 | Endoxifen HCl, the active metabolite of Tamoxifen, is a potent antiestrogen that targets estrogen receptor. |
| CSN19119 | Endoxifen (E-isomer) | 114828-90-9 | Endoxifen E-isomer is the E-isomer of (Z)-Endoxifen, which is an active metabolite generated via actions of CYP3A4/5 and CYP2D6, is a more potent selective estrogen receptor modulator (SERM) than Tamoxifen. |
| CSN17545 | Endoxifen E-isomer HCl | 1197194-61-8 | Endoxifen E-isomer HCl is a tamoxifen metabolite and potent Selective Estrogen Response Modifier (SERM). |
| CSN19762 | Elacestrant | 722533-56-4 | Elacestrant is an orally available, selective estrogen receptor degrader (SERD) and selective estrogen receptor modulator (SERM), with potential antineoplastic and estrogen-like activities. |
| CSN19763 | Elacestrant 2HCl | 1349723-93-8 | Elacestrant 2HCl is an orally available, selective estrogen receptor degrader (SERD) and selective estrogen receptor modulator (SERM), with potential antineoplastic and estrogen-like activities. |
| CSN15920 | DPN | 1428-67-7 | DPN is a non-steroidal estrogen receptor β (ER β) selective ligand. |
| CSN17329 | 7-Hydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one | 486-66-8 | Daidzein can act as an inhibitor of tyrosine kinase and an activator of estrogen receptor. It is inactive analogue of genistein. |
| CSN18336 | BHPI | 56632-39-4 | BHPI is a potent inhibitor of nuclear estrogen–ERα-regulated gene expression and elicits sustained ERα-dependent activation of the endoplasmic reticulum (EnR) stress sensor, the unfolded protein response (UPR), and persistent inhibition of protein synthesis. |
| CSN15663 | Bavachin | 19879-32-4 | Bavachin, a flavonoid phytoestrogen, can activate the estrogen receptors ERα (EC50 = 320 nM) and ERβ (EC50 = 680 nM). |
| CSN17981 | AZD9496 maleate | 1639042-28-6 | AZD9496 maleate is a potent and orally bioavailable selective estrogen receptor downregulator (Ki=0.7 nM) and antagonist. |
| CSN17980 | AZD9496 | 1639042-08-2 | AZD9496 is a selective antagonist of estrogen receptor Erα (IC50 = 0.28 nM). |
| CSN13183 | (8R,9S,10R,13S,14S,17R)-17-Acetyl-17-hydroxy-10,13-dimethyl-6,7,8,9,10,11,12,13,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-3(2H)-one | 68-96-2 | 17α-hydroxyprogesterone is an endogenous progestogen. It is also a chemical intermediate for many other endogenous steroids. |
| CSN17213 | Hydroxy progesterone caproate | 630-56-8 | 17-Caproxyprogesterone is a steroidal progestin. It is a synthetic ester derivative of 17α-hydroxyprogesterone. |
| CSN27120 | (8R,9S,10R,13S,14S,17R)-17-Acetyl-17-hydroxy-10,13-dimethyl-6,7,8,9,10,11,12,13,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-3(2H)-one | 68-96-2 |
