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Adrenergic Receptor

Adrenergic Receptor

货号 产品名 CAS号 信息
CSN10049 UK-14304 59803-98-4 UK-14304 is an adrenergic receptor α2 agonist which can activate ERK in epicardial coronary artery culture, inhibit R-type calcium currents, as well as inhibit hormone-sensitive lipase activity and suppresses lipogenesis in adipose tissue.
CSN10410 Tizanidine 51322-75-9 Tizanidine is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
CSN25553 SR59230A 174689-39-5 SR59230A is a potent and selective Adrenergic Receptor β3 antagonist with IC50 values of 40, 408, and 648nM for Adrenergic Receptor β3, β1 and β2, respectively. It shows blood-brain barrier penetrability.
CSN24703 1-(4-(4-Amino-6,7-dimethoxyquinazolin-2-yl)piperazin-1-yl)-2-(2-isopropyl-6-methoxyphenoxy)ethanone hydrochloride 173059-17-1 REC-2615 (HCl) is a α1B-adrenoceptor antagonist potentially for the treatment of female sexual dysfunction.
CSN10098 Nebivolol HCl 152520-56-4 Nebivolol HCl selectively inhibits β1- adrenergic receptor with IC50 of 0.8 nM. Nebivolol HCl is a cardioselective β1- adrenergic receptor antagonist with IC50 value of 0.8 nM.
CSN11521 Naphazoline HCl 550-99-2 Naphazoline HCl is a direct-acting sympathomimetic amine with vasoconstrictive activity.
CSN11368 Medetomidine 86347-14-0 Medetomidine is an agonist of α2-adrenoceptor with Ki value of 1.08 nM, used as both a surgical anesthetic and analgesic.
CSN11360 Maprotiline HCl 10347-81-6 Maprotiline HCl is a bridged-ring tetracyclic antidepressant with adrenergic activity and sedative properties, exerting its effect by blocking the re-uptake of norepinephrine, thereby increasing the synaptic concentration of norepinephrine in the central nervous system and subsequently prolonging the action of norepinephrine on central receptors.
CSN23830 Lofexidine 31036-80-3 Lofexidine is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal[1][2].
CSN23826 Landiolol HCl 144481-98-1 Landiolol hydrochloride (ONO1101 hydrochloride) is a highly beta1 selective ultra-short acting beta-blocker (β1/β2 selectivity = 255:1, a half-life of 4 min), acts as an adrenoceptor antagonist[1].
CSN10675 L-(-)-α-Methyldopa Hydrate 41372-08-1 L-(-)-α-Methyldopa is an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive drug used as a sympatholytic or antihypertensive.
CSN11205 Indoramin HCl 38821-52-2 Indoramin HCl belongs to a group of medicines called alpha-adrenoreceptor blockers.
CSN11167 Hydrocortisone 17-Butyrate 13609-67-1 Hydrocortisone 17-butyrate is an adrenocortico hormone
CSN11127 Guanfacine 29110-47-2 Guanfacine is a selective α2A receptor agonist.
CSN23785 GUANABENZ 5051-62-7 Guanabenz is an agonist of α2-adrenergic receptor with antihypertensive effect and is enerally used in combination with diuretics.
CSN11125 Guanabenz Acetate 23256-50-0 Guanabenz acetate is a centrally-acting α-2 adrenergic receptor agonist that is used as an antihypertensive drug to treat hypertension.
CSN10861 Doxazosin 74191-85-8 Doxazosin is a quinazoline-derivative that selectively antagonizes postsynaptic α1-adrenergic receptors.
CSN10855 Dopexamine 86197-47-9 Dopexamine is a synthetic analogue of dopamine that is administered intravenously in hospitals to reduce exacerbations of heart failure and to treat heart failure following cardiac surgery.
CSN10784 Dexmedetomidine 113775-47-6 Dexmedetomidine is a new generation highly selective α2-adrenergic receptor (α2-AR) agonist with Ki value of 1.08 nM, which is associated with sedative and analgesic sparing effects, reduced delirium and agitation, perioperative sympatholysis, cardiovascular stabilizing effects, and preservation of respiratory function.
CSN10781 Detomidine HCl 90038-01-0 Detomidine HCl is an imidazole-derived α2-adrenergic agonist, used in veterinary medicine for sedation of large animals.
CSN10770 Deoxycorticosterone Acetate 56-47-3 Deoxycorticosterone acetate is a corticosteroid hormone which can induce hypertension dependent on altered regulation of central pressor mechanisms including the brain renin-angiotensin system.
CSN10681 Clorprenaline HCl 6933-90-0 Clorprenaline HCl is a phenethylamine-derived β2-receptor agonist, acting as a bronchodilator.
CSN10677 Clonidine HCl 4205-91-8 Clonidine HCl is a centrally-acting and brain-permeable α2-adrenergic agonist, which can induce a decrease in blood pressure.
CSN11164 Cadralazine 64241-34-5 Cadralazine is an antihypertensive of the hydrazinophthalazine chemical class.
CSN10507 Bunazosin HCl 52712-76-2 Bunazosin HCl, is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.
CSN10444 Bevantolol 59170-23-9 Bevantolol is a drug candidate for angina and hypertension that acted as both a beta blocker and a calcium channel blocker.
CSN10351 Atipamezole 104054-27-5 Atipamezole is a synthetic competitive α2 adrenergic receptor antagonist with Ki value of 1.6 nM.
CSN10338 Arotinolol 68377-92-4 Arotinolol is a blocker of both α- and β-receptor, and also acts as a β3 receptor agonist. It is used in the treatment of high blood pressure and essential tremor.
CSN10322 Apraclonidine 66711-21-5 Apraclonidine is a clonidine derivative with selective alpha-2-adrenergic agonistic activity. Upon ocular administration, apraclonidine enhances aqueous humor uveoscleral outflow and decreases aqueous production by vasoconstriction. This may decrease intraocular pressure (IOP).
CSN10277 Amezinium Methylsulfate 30578-37-1 Amezinium methylsulfate can stimulate α and β-1 receptors and inhibit noradrenaline and tyramine uptake, used as a sympathomimetic drug for the treatment of low blood pressure.
CSN10237 Alfuzosin 81403-80-7 Alfuzosin is an α1 adrenergic receptor antagonist used to treat benign prostatic hyperplasia (BPH).
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