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Adrenergic Receptor

Adrenergic Receptor

货号 产品名 CAS号 信息
CSN10438 Betaxolol 63659-18-7 βxolol is a competitive and cardioselective β1 adrenergic receptor antagonist, used to treat hypertension, arrhythmias, coronary heart disease, glaucoma, and reduce non-fatal cardiac events in patients with heart failure with elimination half-life of 14–22 hours.
CSN10439 Betaxolol HCl 63659-19-8 βxolol HCl is a competitive and cardioselective β1 adrenergic receptor antagonist, used to treat hypertension, arrhythmias, coronary heart disease, glaucoma, and reduce non-fatal cardiac events in patients with heart failure with elimination half-life of 14–22 hours.
CSN10410 Tizanidine 51322-75-9 Tizanidine is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
CSN10098 Nebivolol HCl 152520-56-4 Nebivolol HCl selectively inhibits β1- adrenergic receptor with IC50 of 0.8 nM. Nebivolol HCl is a cardioselective β1- adrenergic receptor antagonist with IC50 value of 0.8 nM.
CSN11521 Naphazoline HCl 550-99-2 Naphazoline HCl is a direct-acting sympathomimetic amine with vasoconstrictive activity.
CSN11512 Naftopidil 57149-07-2 Naftopidil is a selective α1-adrenergic receptor antagonist or α blocker used for treatment for lower urinary tract symptoms (LUTS) due to benign prostatic hyperplasia (BPH).
CSN11513 Naftopidil 2HCl 57149-08-3 Naftopidil HCl is a selective α1-adrenergic receptor antagonist or α blocker used for treatment for lower urinary tract symptoms (LUTS) due to benign prostatic hyperplasia (BPH).
CSN11429 Metoprolol Succinate 98418-47-4 Metoprolol succinate is a cardioselective β1-adrenergic blocking agent used to treat high blood pressure, chest pain, and heart stress after a heart attack.
CSN10092 Methoxyphenamine HCl 5588-10-3 Methoxyphenamine HCl is a β-adrenergic receptor agonist of the amphetamine class used as a bronchodilator.
CSN11389 Metaraminol Tartrate 33402-03-8 Metaraminol tartrate is an α1-adrenergic receptor agonist, is a potent sympathomimetic amine used in the prevention and treatment of hypotension, particularly as a complication of anesthesia.
CSN11368 Medetomidine 86347-14-0 Medetomidine is an agonist of α2-adrenoceptor with Ki value of 1.08 nM, used as both a surgical anesthetic and analgesic.
CSN11360 Maprotiline HCl 10347-81-6 Maprotiline HCl is a bridged-ring tetracyclic antidepressant with adrenergic activity and sedative properties, exerting its effect by blocking the re-uptake of norepinephrine, thereby increasing the synaptic concentration of norepinephrine in the central nervous system and subsequently prolonging the action of norepinephrine on central receptors.
CSN11290 Levobetaxolol HCl 116209-55-3 Levoβxolol HCl a selective β-1 adrenergic receptor antagonist used to lower the pressure in the eye in treating conditions such as glaucoma with Ki values of 0.76 nM and 32.6 nM for cloned human β1 and β2 receptors, respectively, which is the S-isomer of βxolol.
CSN11259 Labetalol HCl 32780-64-6 Laβlol HCl is a third generation selective α-1-adrenergic antagonist and non-selective β-adrenergic antagonist, used to treat high blood pressure.
CSN10675 L-(-)-α-Methyldopa Hydrate 41372-08-1 L-(-)-α-Methyldopa is an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive drug used as a sympatholytic or antihypertensive.
CSN11239 Ivabradine HCl 148849-67-6 Ivabradine HCl is the first selective sinus node I(f) channel, used for the symptomatic management of stable heart-related chest pain and heart failure not fully managed by β blockers.
CSN11205 Indoramin HCl 38821-52-2 Indoramin hydrochloride belongs to a group of medicines called alpha-adrenoreceptor blockers.
CSN11167 Hydrocortisone 17-Butyrate 13609-67-1 Hydrocortisone 17-butyrate is an adrenocortico hormone
CSN11127 Guanfacine 29110-47-2 Guanfacine is a selective α2A receptor agonist.
CSN11125 Guanabenz Acetate 23256-50-0 Guanabenz acetate is a centrally-acting α-2 adrenergic receptor agonist that is used as an antihypertensive drug to treat hypertension.
CSN10875 Droxidopa 23651-95-8 Droxidopa is a synthetic amino acid precursor which acts as a prodrug to the neurotransmitters norepinephrine (noradrenaline) and epinephrine (adrenaline) and capable of crossing the protective blood–brain barrier.
CSN10861 Doxazosin 74191-85-8 Doxazosin is a quinazoline-derivative that selectively antagonizes postsynaptic α1-adrenergic receptors.
CSN10855 Dopexamine 86197-47-9 Dopexamine is a synthetic analogue of dopamine that is administered intravenously in hospitals to reduce exacerbations of heart failure and to treat heart failure following cardiac surgery.
CSN10784 Dexmedetomidine 113775-47-6 Dexmedetomidine is a new generation highly selective α2-adrenergic receptor (α2-AR) agonist with Ki value of 1.08 nM, which is associated with sedative and analgesic sparing effects, reduced delirium and agitation, perioperative sympatholysis, cardiovascular stabilizing effects, and preservation of respiratory function.
CSN10781 Detomidine HCl 90038-01-0 Detomidine HCl is an imidazole-derived α2-adrenergic agonist, used in veterinary medicine for sedation of large animals.
CSN10770 Deoxycorticosterone Acetate 56-47-3 Deoxycorticosterone acetate is a corticosteroid hormone which can induce hypertension dependent on altered regulation of central pressor mechanisms including the brain renin-angiotensin system.
CSN10747 Dapiprazole 72822-12-9 Dapiprazole is an alpha blocker. It is used to reverse mydriasis after eye examination.
CSN10681 Clorprenaline HCl 6933-90-0 Clorprenaline HCl is a phenethylamine-derived β2-receptor agonist, acting as a bronchodilator.
CSN10677 Clonidine HCl 4205-91-8 Clonidine HCl is a centrally-acting and brain-permeable α2-adrenergic agonist, which can induce a decrease in blood pressure.
CSN10555 Carvedilol 72956-09-3 Carvedilol can block β-1 and β-2 adrenergic receptors as well as the α-1 adrenergic receptors, indicated in the treatment of mild to moderate congestive heart failure.
CSN11164 Cadralazine 64241-34-5 Cadralazine is an antihypertensive of the hydrazinophthalazine chemical class.
CSN10507 Bunazosin HCl 52712-76-2 Bunazosin hydrochloride, is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.
CSN10049 Brimonidine 59803-98-4 Brimonidine is an adrenergic receptor α2 (α2-AR) agonist which can activate ERK in epicardial coronary artery culture, inhibit R-type calcium currents, as well as inhibit hormone-sensitive lipase activity and suppresses lipogenesis in adipose tissue.
CSN10444 Bevantolol 59170-23-9 Bevantolol is a drug candidate for angina and hypertension that acted as both a beta blocker and a calcium channel blocker.
CSN10351 Atipamezole 104054-27-5 Atipamezole is a synthetic competitive α2 adrenergic receptor antagonist with Ki value of 1.6 nM.
CSN10338 Arotinolol 68377-92-4 Arotinolol is a blocker of both α- and β-receptor, and also acts as a β3 receptor agonist. It is used in the treatment of high blood pressure and essential tremor.
CSN10322 Apraclonidine 66711-21-5 Apraclonidine is a clonidine derivative with selective alpha-2-adrenergic agonistic activity. Upon ocular administration, apraclonidine enhances aqueous humor uveoscleral outflow and decreases aqueous production by vasoconstriction. This may decrease intraocular pressure (IOP).
CSN10277 Amezinium Methylsulfate 30578-37-1 Amezinium methylsulfate can stimulate α and β-1 receptors and inhibit noradrenaline and tyramine uptake, used as a sympathomimetic drug for the treatment of low blood pressure.
CSN10237 Alfuzosin 81403-80-7 Alfuzosin is an α1 adrenergic receptor antagonist used to treat benign prostatic hyperplasia (BPH).
CSN10200 Acebutolol HCl 34381-68-5 Acebutolol HCl is a cardioselective β1 adrenergic antagonist with little effect on the bronchial receptors.
CSN10467 (±)-Bisoprolol Hemifumarate 104344-23-2 (±)-Bisoprolol hemifumarate is cardioselective β1-adrenoceptor antagonist, effective in the management of hypertension and angina pectoris.
CSN23830 Lofexidine 31036-80-3
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