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Adrenergic Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN12225 | Xylometazoline HCl | 1218-35-5 | Xylometazoline HCl a direct acting sympathomimetic adrenergic α-agonist, used to improve symptoms of nasal congestion, allergic rhinitis, and sinusitis with elimination half-life of >10 seconds. |
| CSN12104 | Tolazoline | 59-98-3 | Tolazoline is a non-selective competitive α-adrenergic receptor antagonist. |
| CSN12099 | Tizanidine HCl | 64461-82-1 | Tiamenidine HCl is a centrally-acting α1 and α2 adrenergic receptor antagonist with IC50 4.85 μM and 0.0091 μM, respectively, for the management of essential hypertension. |
| CSN12067 | Tetrahydroalstonine | 6474-90-4 | Tetrahydroalstonine, a natural product isolated and purified from the herbs of Uncaria rhynchophylla (Miq.) Miq. ex Havil., preferentially blocks the pressor responses of post-synaptic alpha-adrenergic receptor activation due to exogenous and endogenouse noradrenaline, respectively. |
| CSN12052 | (4-(4-Amino-6,7-dimethoxyquinazolin-2-yl)piperazin-1-yl)(tetrahydrofuran-2-yl)methanone hydrochloride dihydrate | 70024-40-7 | Terazosin HCl is an α-adrenergic (AL-fa ad-ren-ER-jik) blocker used in the therapy of hypertension and benign prostatic hypertrophy with climination half-life of 12 hours. |
| CSN12855 | Terazosin HCl | 63074-08-8 | Terazosin HCl is a selective antagonist for alpha-adrenergic receptor, used for treatment for hypertension and prostate enlargement (BPH) through lowering the blood pressure with elimination half-life of 12 hours. |
| CSN12031 | Tamsulosin HCl | 106463-17-6 | Tamsulosin HCl a selective antagonist at α-1A and α-1B-adrenoceptors, used to treat the symptoms of benign prostatic hyperplasia (BPH). |
| CSN12030 | Tampramine | 83166-17-0 | Tampramine is a tricyclic antidepressant (TCA). |
| CSN12335 | Silodosin | 160970-54-7 | Silodosinis a selective prostate α1-adrenoceptor antagonist for symptomatic treatment of benign prostatic hyperplasia. |
| CSN12682 | Scopine | 498-45-3 | Scopine is a naturally occuring α1-adrenergic receptor agonist which is the metabolite of anisodine, used in the treatment of acute circulatory shock. |
| CSN13046 | Scopine HCl | 85700-55-6 | Scopine HCl salt is a naturally occuring α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock and also s a potential brain-targeting moiety for enhancing the brain uptake efficiency of chlorambucil. |
| CSN11850 | Ritodrine HCl | 23239-51-2 | Ritodrine HCl activates β-2 adrenergic receptor through binding to β-2 adrenergic receptors on outer membrane of myometrial cell, used to stop premature labor. |
| CSN11847 | Rilmenidine phosphate | 85409-38-7 | Rilmenidine Phosphate is an oxazole-derived agonist of adrenergic receptor α2 and Imidazoline receptor, used in trials studying the treatment of hypertension and chronic kidney disease. |
| CSN13629 | Prazosin HCl | 19237-84-4 | Prazosin HCl is a selective α-1-adrenergic receptor antagonist used to treat hypertension, anxiety, and posttraumatic stress disorder (PTSD). |
| CSN12736 | Phenoxybenzamine HCl | 63-92-3 | Phenoxybenzamine HCl is a non-selective irreversible dibenzamine α adrenergic antagonist with antihypertensive and vasodilatory properties. |
| CSN13642 | (R)-2-(2-Aminothiazol-4-yl)-N-(4-(2-((2-hydroxy-2-phenylethyl)amino)ethyl)phenyl)acetamide | 223673-61-8 | Mirabegron is an agonist of β3 adrenergic receptor with EC50 value of 22.4nM, used for the treatment of overactive bladder. |
| CSN13464 | Guanfacine HCl | 29110-48-3 | Guanfacine HCl is a centrally acting antihypertensive with α2-adrenoceptor agonist with Kd value of 31 nM for α2A-adrenoceptor while displaying 60-fold selectivity over α2B-adrenoceptors, causing a decrease in heart rate and peripheral vascular resistance. |
| CSN12942 | Doxazosin mesylate | 77883-43-3 | Doxazosin mesylate is a selective α1-adrenergic receptor blocker, used to treat high blood pressure and urinary retention associated with benign prostatic hyperplasia (BPH). |
| CSN12451 | Dobutamine HCl | 49745-95-1 | Dobutamine HCl is a sympathomimetic drug used in the treatment of heart failure and cardiogenic shock. |
| CSN16164 | (S)-5-(1-(2,3-Dimethylphenyl)ethyl)-1H-imidazole hydrochloride | 145108-58-3 | Dexmedetomidine is a selectively activator of presynaptic alpha-2 adrenoceptors located in the brain. This leads to inhibition of postsynaptic activation of adrenoceptors through inhibiting the release of norepinephrine from synaptic vesicles, thereby leading to analgesia, sedation and anxiolysis. |
| CSN13917 | Brimonidine tartrate | 70359-46-5 | Brimonidine tartrate is an α-adrenergic receptor agonist with EC50 of 0.45 nM for the α2A adrenoreceptor, used to treat glaucoma through a dual mechanism of action by reducing aqueous humor production and increasing uveoscleral outflow. |
| CSN13005 | BMY 7378 | 21102-95-4 | BMY 7378 2HCl is a 5-HT1A partial agonist and a high-affinity α1D adrenoceptor antagonist with Ki values of 2, 800 and 600 nM for cloned rat α1D, rat α1A and hamster α1B receptors respectively. |
| CSN12452 | Bambuterol HCl | 81732-46-9 | Bambuterol HCl, a prodrug of terbutaline, is a long-acting β adrenoceptor agonist used in the treatment of asthma with elimination half-life of 13 hours. |
| CSN12750 | (R)-N-Methyl-3-phenyl-3-(o-tolyloxy)propan-1-amine hydrochloride | 82248-59-7 | Atomoxetine HCl is a phenoxy-3-propylamine-derived and selective non-stimulant, norepinephrine reuptake inhibitor with cognitive-enhancing activity. |
| CSN52437 | 3-(2-(4-(o-Tolyl)piperazin-1-yl)ethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine hydrochloride | 72822-13-0 |
