欢迎来到 CSNpharm! 产品仅用于科研!
首页 400-920-2911

Src

Src

货号 产品名 CAS号 信息
CSN16229 WH-4-023 837422-57-8 WH-4-023 is an inhibitor of Lck and Src with IC50 of 2 nM, 6 nM, respectively.
CSN17744 WEHI-345 Analog 1354825-62-9 WEHI-345 analog is a Src inhibitor.
CSN13096 TG 100801 867331-82-6 TG 100801 is the prodrug of TG 100572, which is a multi-targeted kinase inhibitor that inhibit select growth factor receptor tyrosine kinases and Src family kinases with IC50 values of 2/7/2/1/0.5 nM of VEGFR1/VEGFR2/FGFR1/Src/Fyn kianse respectively.
CSN18504 TG 100572 867334-05-2 TG 100572 is a multi-targeted kinase inhibitor that inhibit select growth factor receptor tyrosine kinases and Src familt kinases with IC50 values of 2/7/2/1/0.5 nM for VEGFR1/VEGFR2/FGFR1/Src/Fyn kianse respectively.
CSN18503 TG 100572 HCl 867331-64-4 TG 100572 hydrochloride is a multi-targeted kinase inhibitor that inhibits select growth factor receptor tyrosine kinases and Src familt kinases with IC50 values of 2/7/2/1/0.5 nM for VEGFR1/VEGFR2/FGFR1/Src/Fyn kianse respectively.
CSN17735 T338C Src-IN-2 1351927-00-8 T338C Src-IN-2 is a potent mutant c-Src T338C kinase inhibitor with IC50 of 317 nM and also inhibits T338C/V323A and T338C/V323S with IC50 of 57 nM/19 nM.
CSN17734 T338C Src-IN-1 1351926-90-3 T338C Src-IN-1 is a potent mutant-Src T338C inhibitor and exhibits the most potent inhibition of T338C (IC50=111 nM) relative to WT c-Src(10-fold increase).
CSN18218 SU6656 330161-87-0 SU 6656 is an inhibitor of Src kinases and can target Src, Yes, Lyn, and Fyn with IC50 of 280 nM, 20 nM, 130 nM, 170 nM, respectively.
CSN17355 Src Inhibitor 1 179248-59-0 Src inhibitor 1 is an inhibitor of Src and Lck with IC50 of 44 nM and 88nM.
CSN12259 Saracatinib 379231-04-6 Saracatinib is Src inhibitor with IC50 of 2.7 nM.
CSN23720 RK 24466 213743-31-8 RK-24466 is an inhibitor of Lck (64-509) and LckCD isoforms with IC50s of <2 nM.
CSN11759 PP2 172889-27-9 PP2 is a ATP-competitive inhibitor of the Src family of protein tyrosine kinases. The IC50s for p56lck, p59fynT, Hck, Src are 4 nM, 5 nM, 5 nM, 100 nM, respectively.
CSN11758 PP1 172889-26-8 PP1 is a selective inhibitor of Src and Lck/Fyn with IC50 of 5 nM, 6 nM, respectively.
CSN12857 PD173955 260415-63-2 PD173955 is an src family-selective tyrosine kinase inhibitor with IC50 of ~22 nM for Src, Yes and Abl kinase and is less potent for FGFRα and no activity on InsR and PKC.
CSN17507 MCB-613 1162656-22-5 MCB-613 is a stimulator of steroid receptor coactivator (SRC).
CSN16563 Lck Inhibitor 847950-09-8 Lck inhibitor is a class of compounds that are potent inhibitors of Lck with an IC50 value of 7 nM.
CSN18620 Lck Inhibitor 2 944795-06-6 Lck inhibitor 2 is a bis-anilinopyrimidine inhibitor of tyrosine kinases including LCK, BTK, LYN, SYK, and TXK. The IC50 values are 13nM, 9nM, 3nM, 26nM and 2nM for Lck, Btk, Lyn, Btk and Txk respectively.
CSN18935 KX2-391 Mesylate 1080645-95-9 KX2-391 mesylate is an inhibitor of Src that targets the peptide substrate site of Src, with GI50 of 9-60 nM in cancer cell lines.
CSN16540 KX2-391 897016-82-9 KX2-391 is an inhibitor of Src with IC50 of 9 nM-60 nM in cancer cells. It is the first clinical and peptidomimetic class Src inhibitor.
CSN16378 KX2-391 2HCl 1038395-65-1 KX2-391 dihydrochloride is the first clinical Src inhibitor (peptidomimetic class) that targets the peptide substrate site of Src, with GI50 of 9-60 nM in cancer cell lines.
CSN13760 KX1-004 518058-84-9 KX1-004 is a potent small molecule inhibitor of Src-PTK as a potential protective drug for NIHL.
CSN19857 KB SRC 4 1380088-03-8 KB SRC 4 is a potent and selective c-Src inhibitor (Ki = 44 nM) and does not inhibit c-Abl at concentrations up to 125 μM.
CSN11935 Bosutinib 380843-75-4 Bosutinib is an inhibitor of Src and Abl with IC50 of 1.2 nM and 1 nM.
CSN18293 AZM475271 476159-98-5 AZM475271 is a potent and selective Src kinase inhibitor with IC50 of 5 nM showing no inhibitory activity on Flt3, KDR, Tie-2.
CSN17121 AMG-47a 882663-88-9 AMG-47a is a Lck inhibitor that can decrease T cell proliferation with anti-inflammatory activity.
CSN17856 A 419259 3HCl 1435934-25-0 A 419259 trihydrochloride is a broad-spectrum pyrrolo-pyrimidine inhibitor, designed to enhance selectivity towards the Src family with IC50 of 9 nM, < 3 nM and < 3 nM for Src, Lck and Lyn, respectively.
CSN18243 A 419259 364042-47-7 A 419259 is an apoptosis inducing agent that inhibits Src family kinases (c-Src) and also induces apoptosis in CML cell ines and blocks Stat5 and Erk activation.
CSN21118 7-Hydroxy-4-chromone 59887-89-7 7-Hydroxychromone is a Src kinase inhibitor with an IC50 of <300 μM.
CSN13856 1-Naphthyl PP1 221243-82-9 1-Naphthyl PP1 is a selective inhibitor of src family kinases v-Src and c-Fyn as well as the tyrosine kinase c-Abl (IC50 values are 1.0, 0.6, 0.6, 18 and 22 μM for v-Src, c-Fyn, c-Abl, CDK2 and CAMK II respectively).
CSN15753 1-Naphthyl PP1 HCl 956025-47-1 1-Naphthyl PP1 hydrochloride is a selective inhibitor of src family kinases v-Src and c-Fyn as well as the tyrosine kinase c-Abl (IC50 values are 1.0, 0.6, 0.6, 18 and 22 μM for v-Src, c-Fyn, c-Abl, CDK2 and CAMK II respectively).
CSN23025 PD 166285 2HCl 212391-63-4
<< PREV 1 2 NEXT >>