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Src

Src

货号 产品名 CAS号 信息
CSN17744 WEHI-345 Analog 1354825-62-9 WEHI-345 analog is a Src inhibitor.
CSN13096 TG 100801 867331-82-6 TG 100801 is the prodrug of TG 100572, which is a multi-targeted kinase inhibitor that inhibit select growth factor receptor tyrosine kinases and Src family kinases with IC50 values of 2/7/2/1/0.5 nM of VEGFR1/VEGFR2/FGFR1/Src/Fyn kianse respectively.
CSN18504 TG 100572 867334-05-2 TG 100572 is a multi-targeted kinase inhibitor that inhibit select growth factor receptor tyrosine kinases and Src familt kinases with IC50 values of 2/7/2/1/0.5 nM for VEGFR1/VEGFR2/FGFR1/Src/Fyn kianse respectively.
CSN18503 TG 100572 HCl 867331-64-4 TG 100572 HCl is a multi-targeted kinase inhibitor that inhibits select growth factor receptor tyrosine kinases and Src familt kinases with IC50 values of 2/7/2/1/0.5 nM for VEGFR1/VEGFR2/FGFR1/Src/Fyn kianse respectively.
CSN17735 T338C Src-IN-2 1351927-00-8 T338C Src-IN-2 is a potent mutant c-Src T338C kinase inhibitor with IC50 of 317 nM and also inhibits T338C/V323A and T338C/V323S with IC50 of 57 nM/19 nM.
CSN17734 T338C Src-IN-1 1351926-90-3 T338C Src-IN-1 is a potent mutant-Src T338C inhibitor and exhibits the most potent inhibition of T338C (IC50=111 nM) relative to WT c-Src(10-fold increase).
CSN17355 Src Inhibitor 1 179248-59-0 Src inhibitor 1 is an inhibitor of Src and Lck with IC50 of 44 nM and 88nM.
CSN23720 RK 24466 213743-31-8 RK-24466 is an inhibitor of Lck (64-509) and LckCD isoforms with IC50s of <2 nM.
CSN11759 PP2 172889-27-9 PP2 is a ATP-competitive inhibitor of the Src family of protein tyrosine kinases. The IC50s for p56lck, p59fynT, Hck, Src are 4 nM, 5 nM, 5 nM, 100 nM, respectively.
CSN12857 PD173955 260415-63-2 PD173955 is an src family-selective tyrosine kinase inhibitor with IC50 of ~22 nM for Src, Yes and Abl kinase and is less potent for FGFRα and no activity on InsR and PKC.
CSN23025 PD 166285 2HCl 212391-63-4 PD 166285 inhibited Src nonreceptor tyrosine kinase, fibroblast growth factor receptor-1, epidermal growth factor receptor and platelet-derived growth factor receptor beta subunit (PDGFR-beta), tyrosine kinases with half-maximal inhibitory potencies (IC50 values) of 8.4 +/- 2.3 nM (n = 6), 39.3 +/- 2.8 nM (n = 16), 87.5 +/- 13.7 nM (n = 6) and 98.3 +/- 7.9 nM (n = 16), respectively.
CSN16563 Lck Inhibitor 847950-09-8 Lck inhibitor is a class of compounds that are potent inhibitors of Lck with an IC50 value of 7 nM.
CSN18620 Lck Inhibitor 2 944795-06-6 Lck inhibitor 2 is a bis-anilinopyrimidine inhibitor of tyrosine kinases including LCK, BTK, LYN, SYK, and TXK. The IC50 values are 13nM, 9nM, 3nM, 26nM and 2nM for Lck, Btk, Lyn, Btk and Txk respectively.
CSN18935 KX2-391 Mesylate 1080645-95-9 KX2-391 mesylate is an inhibitor of Src that targets the peptide substrate site of Src, with GI50 of 9-60 nM in cancer cell lines.
CSN16378 KX2-391 2HCl 1038395-65-1 KX2-391 2HCl is the first clinical Src inhibitor (peptidomimetic class) that targets the peptide substrate site of Src, with GI50 of 9-60 nM in cancer cell lines.
CSN13760 KX1-004 518058-84-9 KX1-004 is a potent small molecule inhibitor of Src-PTK as a potential protective drug for NIHL.
CSN19857 KB SRC 4 1380088-03-8 KB SRC 4 is a potent and selective c-Src inhibitor (Ki = 44 nM) and does not inhibit c-Abl at concentrations up to 125 μM.
CSN25623 Hck-IN-1 1473404-51-1 Hck Blocker compound B9 is a Nef-dependent Hck blocker with IC50 value of 2.8μM for Nef-Hck complex but >20μM for Hck alone. It binds directly to Nef via a pocket formed by the Nef dimerization interface and disrupts Nef dimerization in cells.
CSN27592 CH6953755 2055918-71-1 CH6953755 is a selective inhibitor of YES1 kinase with IC50 of 1.8 nM.
CSN18293 AZM475271 476159-98-5 AZM475271 is a potent and selective Src kinase inhibitor with IC50 of 5 nM showing no inhibitory activity on Flt3, KDR, Tie-2.
CSN18508 A-770041 869748-10-7 A-770041 is selective and orally active Src-family Lck inhibitor and is a 147 nM inhibitor of Lck(1 mM ATP) and is 300-fold selective against Fyn, the other Src family kinase involved in T-cell signaling.
CSN18243 A 419259 364042-47-7 A 419259 is an apoptosis inducing agent that inhibits Src family kinases (c-Src) and also induces apoptosis in CML cell ines and blocks Stat5 and Erk activation.
CSN17856 A 419259 3HCl 1435934-25-0 A 419259 3HCl is a broad-spectrum pyrrolo-pyrimidine inhibitor, designed to enhance selectivity towards the Src family with IC50 of 9 nM, < 3 nM and < 3 nM for Src, Lck and Lyn, respectively.
CSN21118 7-Hydroxy-4-chromone 59887-89-7 7-Hydroxychromone is a Src kinase inhibitor with an IC50 of <300 μM.
CSN13856 1-Naphthyl PP1 221243-82-9 1-Naphthyl PP1 is a selective inhibitor of src family kinases v-Src and c-Fyn as well as the tyrosine kinase c-Abl (IC50 values are 1.0, 0.6, 0.6, 18 and 22 μM for v-Src, c-Fyn, c-Abl, CDK2 and CAMK II respectively).
CSN15753 1-Naphthyl PP1 HCl 956025-47-1 1-Naphthyl PP1 HCl is a selective inhibitor of src family kinases v-Src and c-Fyn as well as the tyrosine kinase c-Abl (IC50 values are 1.0, 0.6, 0.6, 18 and 22 μM for v-Src, c-Fyn, c-Abl, CDK2 and CAMK II respectively).
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