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Vasopressin Receptor

Vasopressin Receptor

货号 产品名 CAS号 信息
CSN16162 Xipamide 14293-44-8 Xipamide, a sulfonamide diuretic drug, can block sodium reabsorption in distal tubules of the kidney and the cystic fibrosis transmembrane conductance regulator (CFTR) chloride channel. It is used for the treatment of oedema and hypertension.
CSN12057 Terlipressin 14636-12-5 Terlipressin, an analog of vasopressin, acts as vasoconstrictor via V1 receptors on arteriolar smooth muscle cells and can reduce visceral blood flow. It is used to treat hypotension.
CSN20586 SR49059 150375-75-0 SR49059 is a potent and selective non-peptide vasopressin V1A receptor antagonist which is devoid of agonist activity. SR49059 displays high affinity and efficacy at both rat (Ki = 1.6 nM) and human (Ki = 1.1 - 6.3 nM) V1A receptors and potently antagonizes arginine vasopressin-induced effects in vitro (IC50 = 3.7 nM for inhibition of human platelet aggregation) and is orally active in vivo.
CSN20548 Selepressin 876296-47-8 Selepressin is a potent, selective vasopressin V1a receptor agonist potentially for the treatment of septic shock.
CSN21427 RO5028442 920022-47-5 RO5028442 is a potent and selective brain-penetrant vasopressin 1a (V1a) receptor antagonist with Kis of 1 nM (hV1a) and 39 nM (mV1a).
CSN12760 Mozavaptan 137975-06-5 Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
CSN10777 Desmopressin 16679-58-6 Desmopressin is the synthetic analogue of the antidiuretic hormone arginine vasopressin.
CSN10778 Desmopressin Acetate 62288-83-9 Desmopressin acetate is the synthetic analogue of the antidiuretic hormone arginine vasopressin.
CSN13437 Conivaptan HCl 168626-94-6 Conivaptan hydrochloride is an inhibitor of antidiuretic hormone or antagonist of vasopressin receptor. It can inhibit rat liver V1A receptor and kidney V2 receptor with Ki of 0.48 nM and 3.04 nM, respectively.
CSN10352 Atosiban 90779-69-4 Atosiban is competitive antagonist of vasopressin and oxytocin receptors. It is a nonapeptide and the analogue of desamino-oxytocin.
CSN22355 Balovaptan 1228088-30-9
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