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NMDAR

NMDAR

货号 产品名 CAS号 信息
CSN21328 UK-240455 178908-09-3 UK-240455 is a potent and selective N-methyl D-aspartate (NMDA) glycine site antagonist.
CSN12978 Traxoprodil 134234-12-1 Traxoprodil a selective antagonist of the NR2B subunit of the NMDA receptor.
CSN24287 Traxoprodil Mesylate 189894-57-3 Traxoprodil a selective antagonist of the NR2B subunit of the NMDA receptor.
CSN21414 Transcrocetin Meglumine Salt N/A Transcrocetin meglumine salt, extracted from saffron (Crocus sativus L.), acts as an NMDA receptor antagonist with high affinity.
CSN17823 Tiletamine HCl 14176-50-2 Tiletamine HCl is an NMDA receptor antagonist used as a dissociative anesthetic.
CSN11907 SDZ 220-581 174575-17-8 SDZ 220-581 is a potent, competitive antagonist at the NMDA glutamate receptor subtype (pKi= 7.7).
CSN18033 SDZ 220-581 HCl 179411-93-9 SDZ 220-581 hydrochloride is a potent, competitive antagonist at the NMDA glutamate receptor subtype (pKi= 7.7).
CSN18034 SDZ 220-581 Ammonium 179411-94-0 SDZ 220-581 ammonium is a potent, competitive antagonist at the NMDA glutamate receptor subtype (pKi= 7.7).
CSN15699 Sarcosine 107-97-1 Sarcosine is an NMDAR co-agonist at the glycine binding site. It is an intermediate and byproduct in glycine synthesis and degradation.
CSN17681 Ro 25-6981 Maleate 1312991-76-6 Ro 25-6981 maleate is a potent and selective activity-dependent blocker of NMDA receptors containing the NR2B subunit.
CSN17353 Ro 25-6981 169274-78-6 Ro 25-6981 is a potent and selective activity-dependent blocker of NMDA receptors containing the NR2B subunit.
CSN17520 Rapastinel 117928-94-6 Rapastinel is a putative NMDAR functional glycine-site partial agonist.
CSN23523 Quinolinic acid 89-00-9 Quinolinic acid is both a selective agonist at NMDA receptors and also a precursor for the formation of NAD+.
CSN16857 QNZ46 1237744-13-6 QNZ46 is a noncompetitive and voltage-independent GluN2C/GluN2D-selective NMDA antagonist with IC50 values of 3, 6, 229 μM for GluN2D, GluN2C, GluN2A, respectively.
CSN11780 Procyclidine HCl 1508-76-5 Procyclidine hydrochloride is an potent anti-cholinergic agent, and is also known to have NMDA antagonist properties.
CSN17346 PEAQX 459836-30-7 PEAQX is a potent and orally active NMDA antagonist with a 15-fold preference for human NMDA receptors with the 1A/2A (IC50=270 nM), rather than 1A/2B(29,600 nM).
CSN19272 PEAQX Tetrasodium Hydrate N/A PEAQX is a potent and orally active NMDA antagonist with a 15-fold preference for human NMDA receptors with the 1A/2A (IC50=270 nM), rather than 1A/2B(29,600 nM).
CSN11619 Orphenadrine HCl 341-69-5 Orphenadrine hydrochloride is an uncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 6.0 ±0.7 μM.
CSN11618 Orphenadrine Citrate 4682-36-4 Orphenadrine Citrate is both an uncompetitive NMDA receptor antagonist IC50 value of 16.2 µM and a mAChR antagonist with IC50 value of 0.37 µM.
CSN17347 NMDA-IN-1 700878-19-9 NMDA-IN-1 is a potent and NR2B-selective NMDA antagonist with Ki of 0.85 nM. Its NR2B Ca2+ influx IC50 is 9.7 nM without activities on NR2A, NR2C, NR2D, hERG-channel and α1-adrenergic receptor.
CSN13790 NMDA   6384-92-5 NMDA is an amino acid derived specific agonist at the NMDA receptor.
CSN11379 Mephenesin 59-47-2 Mephenesin is a centrally acting muscle relaxant which may work as an NMDA receptor antagonist.
CSN11501 Memantine 19982-08-2 Memantine is the first in a class of Alzheimer's disease medications acting on the glutamatergic system by blocking NMDA receptors.
CSN13695 MDL-29951 130798-51-5 MDL-29951 is a glycine antagonist of NMDA receptor activation (Ki=0.14 mM, [3H]glycine binding) in vitro and in vivo.
CSN13916 MDL 105519 161230-88-2 MDL 105519 is a potent and selective inhibitor of [3H]glycine binding to the NMDA receptor with Kd of 3.89 nM.
CSN20030 Lanicemine 153322-05-5 Lanicemine is a low-trapping NMDA receptor antagonist. Lanicemine is used the management of severe and treatment-resistant depression. Lanicemine was originally developed as a neuroprotective agent, but was redeveloped as an antidepressant.
CSN17128 L-701,324 142326-59-8 L-701324 is an orally active and long acting anticonvulsant with high affinity and selectivity for the glycine site on the NMDA receptor.
CSN21303 Kynurenic Acid Sodium 2439-02-3 Kynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid is also a selective ligand of the GPR35 receptor.
CSN11186 Ifenprodil Tartrate 23210-58-4 Ifenprodil Tartrate is a high affinity and atypical noncompetitive NMDA receptor antagonist with IC50 of 0.3 μM.
CSN21125 Ibotenic Acid 2552-55-8 Ibotenic acid has agonist activity at both the N-methyl-D-aspartate (NMDA) and trans-ACPD or metabolotropic quisqualate (Qm) receptor sites.
CSN22199 GNE 5729 2026635-66-3 GNE 5729 is a brain permeable positive allosteric modulator of NMDAR, with an EC50 of 37 nM for GluN2A, 4.7 and 9.5 μM for GluN2C and GluN2D, respectively.
CSN22417 GNE 0723 1883518-31-7 GNE 0723 is a brain permeable positive allosteric modulator of NMDAR, with an EC50 of 21 nM for GluN2A, 7.4 and 6.2 μM for GluN2C and GluN2D, respectively.
CSN10988 Felbamate 25451-15-4 Felbamate is a potent nonsedative anticonvulsant whose clinical effect may be related to the inhibition of N-methyl-D-aspartate (NMDA) .
CSN17519 Felbamate Hydrate 1177501-39-1 Felbamate is a potent nonsedative anticonvulsant whose clinical effect may be related to the inhibition of N-methyl-D-aspartate (NMDA) .
CSN10256 Eliprodil 119431-25-3 Eliprodil can antogonize GluN2B-selective NMDA in a non-competitive manner with IC50 value of 1 μM. It is also a σ1 ligand with Ki value of 0.013 μM.
CSN18296 CIQ 486427-17-2 CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit.
CSN19842 CGP 37849 127910-31-0 CGP 37849 is a potent, selective and competitive NMDA receptor antagonist (Ki = 35 nM).
CSN10502 Budipine 57982-78-2 Budipine is an uncompetitive NMDAR antagonist used as an antiparkinson agent.
CSN22349 Apimostinel 1421866-48-9 Apimostinel is an oral NMDA receptor partial agonist.
CSN17580 (-)-MK 801 Maleate 121917-57-5 (-)-MK 801 maleate is the enantiomer of (+)-MK-801, which is a highly potent and selective non-competitive NMDA glutamate receptor antagonist .
CSN13883 (+)-MK 801 Maleate 77086-22-7 (+)-MK 801 Maleate is a highly potent, selective and non-competitive NMDA receptor antagonist with Ki of 30.5 nM.
CSN23784 Radiprodil 496054-87-6
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