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Androgen Receptor

Androgen Receptor

货号 产品名 CAS号 信息
CSN21357 YK11 1370003-76-1 YK11 is a partial agonist of androgen receptor, with osteogenic activity.
CSN12743 RU 58841 154992-24-2 RU 58841 is a nonsteroidal antiandrogen for potential use as a topical treatment for androgen-dependent conditions including acne, pattern hair loss, and excessive hair growth.
CSN19838 RD 162 915087-27-3 RD 162 is an orally active and very potent antagonist of androgen receptor (AR) and is a second-generation of antiandrogen for the treatment of advanced prostate cancer and highly recommended tool in AR research.
CSN17523 RAD140 1182367-47-0 RAD140 is a potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM).
CSN17663 ORM-15341 1297537-33-7 ORM-15341 is a potent and full antagonist for human AR (hAR) with IC50 values of 38 nM as shown by transactivation assays in AR-HEK293 cells stably expressing full-length hAR and an androgen-responsive luciferase reporter gene construct.
CSN17664 ODM-201 1297538-32-9 ODM-201 is a competitive inhibitor of androgen receptor with IC50 value of 26 nM and inhibits AR nuclear translocation with Ki value of 11 nM.
CSN13442 Nomegestrol 58691-88-6 Nomegestrol is a steroidal progestin.
CSN16774 Nilutamide 63612-50-0 Nilutamide is a non-steroidal androgen receptor antagonist and also inhibits androgen biosynthesis in vitro.
CSN17614 N-desmethyl Enzalutamide 1242137-16-1 N-Desmethyl enzalutamide is a major metabolite of Enzalutamide, Enzalutamide (MDV3100) is an androgen-receptor (AR) antagonist with IC50 of 36 nM.
CSN18357 MK-0773 606101-58-0 MK-0773, one of selective androgen receptor modulators (SARMs), is a 4-aza-steroid that exhibited tissue selectivity in humans (IC50= 6.6 nM).
CSN11374 Megestryl Acetate 595-33-5 Megestryl Acetate is a synthetic progesterone analog.
CSN13670 LGD-4033 1165910-22-4 LGD-4033 is a nonsteroidal, oral SARM that binds to androgen receptor with high affinity (Ki of 1 nM) and selectivity.
CSN10977 Hydroxyflutamide 52806-53-8 Hydroxyflutamide is a derivative of the synthetic steroid ethisterone, that suppresses the production of gonadotrophins, and has some weak androgenic effects.
CSN11169 Hydromadinone 16469-74-2 Hydromadinone, is a steroidal progestin of the 17α-hydroxyprogesterone group.
CSN18667 GSK2881078 1539314-06-1 GSK 2881078 is a selective androgen receptor modulator potentially for the treatment of cachexia.
CSN17573 GLPG0492 R-Enantiomer 1215085-93-0 GLPG0492 R-enantiomer is the R-Enantiomer of GLPG-0492, which is a selective androgen receptor modulator.
CSN17572 GLPG0492 1215085-92-9 GLPG0492 is a selective androgen receptor modulator and exhibits anabolic activity on muscle, strongly dissociated from the androgenic activity on prostate after oral dosing.
CSN11095 Gestonorone 2137-18-0 Gestronol is a steroidal progestin of the 19-norprogesterone and 17α-hydroxyprogesterone groups.
CSN16707 Flutamide 13311-84-7 Flutamide is a competitive non-steroidal antagonist of androgen receptor.
CSN10468 EPI-001 227947-06-0 EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ∼6 μM and a selective PPAR-gamma modulator.
CSN12389 Enzalutamide 915087-33-1 Enzalutamide is an androgen-receptor (AR) antagonist with IC50 of 36 nM in LNCaP cells.
CSN10728 Cyproterone Acetate 427-51-0 Cyproterone Acetate is an antagonist and partial agonist of androgen receptor with IC50 value of 7.1 nM and EC50 value of 4μM.
CSN18075 Cortexolone 17 alpha-Propionate 19608-29-8 Cortexolone 17 alpha-propionate is a topical and peripherally selective androgen antagonist, which is used in treatment of acne and androgenic alopecia.
CSN16582 BMS-564929 627530-84-1 BMS-564929 is an androgen receptor (AR) agonist, binds to androgen receptor (AR) with a Ki of 2.11±0.16 nM.
CSN12437 Bicalutamide 90357-06-5 Bicalutamide is non-steroidal androgen receptor antagonist with IC50 value of 190 nM.
CSN17150 AZD3514 1240299-33-5 AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression.
CSN17338 Dimethylcurcumin 52328-98-0 ASC-J9, an antitumor agent, suppresses castration-resistant prostate cancer growth via degradation of full-length and splice variant androgen receptors.
CSN13830 Apalutamide 956104-40-8 ARN-509 can compeitively and selectively inhibit androgen receptor with IC50 value of 16 nM.
CSN20433 Androgen Receptor Modulator C7 2109805-69-6 Androgen receptor modulator C7 is a potent AR (ARE EC50 = 0.34 nM) and tissue-selective (N/C interaction EC50 = 1206 nM) modulator.
CSN22336 ACP-105 899821-23-9 ACP-105 is a potent nonsteroidal selective androgen receptor modulator (SARM) with partial agonist activity relative to the natural androgen testosterone.
CSN19392 3,3'-Diindolylmethane 1968-05-4 3,3'-Diindolylmethane is an AR structurally similar androgen receptor antagonist.
CSN23255 1-Phenylpentan-1-ol 583-03-9 1-Phenylpentan-1-ol is an intermediate for synthesis of β-amino-carbonyl-based androgen receptor antagonist.
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