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CAS No.: 1240299-33-5
AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01162395 | Prostate Cancer | Phase 1 | Completed | - | United States, Oregon ... more >> Research Site Portland, Oregon, United States Netherlands Research Site Amsterdam, Netherlands United Kingdom Research Site Glasgow, United Kingdom Research Site Manchester, United Kingdom Research Site Surrey, United Kingdom Collapse << |
NCT01351688 | Prostate Cancer | Phase 1 | Completed | - | Japan ... more >> Research Site Sagamihara, Kanagawa, Japan Research Site Sunto-gun, Shizuoka, Japan Collapse << |
实验方案
技术信息
CAS号 | 1240299-33-5 | 储存条件 |
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分子式 | C25H32F3N7O2 | 运输 | 蓝冰 | |
分子量 | 519.56 | 别名 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01162395 | Prostate Cancer | Phase 1 | Completed | - | United States, Oregon ... more >> Research Site Portland, Oregon, United States Netherlands Research Site Amsterdam, Netherlands United Kingdom Research Site Glasgow, United Kingdom Research Site Manchester, United Kingdom Research Site Surrey, United Kingdom Collapse << |
NCT01351688 | Prostate Cancer | Phase 1 | Completed | - | Japan ... more >> Research Site Sagamihara, Kanagawa, Japan Research Site Sunto-gun, Shizuoka, Japan Collapse << |
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