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Adenosine Receptor

Adenosine Receptor

货号 产品名 CAS号 信息
CSN12242 ZM241385 139180-30-6 ZM241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor.
CSN19381 Xanthine 69-89-6 Xanthine is a natural occuring purine-base adenosine receptor antagonist, from which a number of stimulants such as caffeine and theobromine are derived.
CSN18277 Vipadenant   442908-10-3 Vipadenant is an adenosine antagonist with Ki of 1.3 nM and 68 nM for A2A and A1, respectively. Vipadenant is a selective A2A receptor antagonist with Ki values of 1.3, 68, 63, and 1,005 nM for A2A, A1, A2B, and A3 receptors, respectively, used in development for for Parkinson's disease.
CSN19829 Trabodenoson 871108-05-3 Trabodenoson is a potent and highly selective adenosine A1 receptor agonist.
CSN16416 Theophylline 58-55-9 Theophylline is a natural product present in tea and cocoa, working as a phosphodiesterase inhibitor, adenosine receptor blocker, and histone deacetylase activator.
CSN21258 Tecadenoson 204512-90-3 Tecadenoson is a selective A1 adenosine receptor agonist.
CSN23108 SCH 442416 316173-57-6 SCH-442416 is a selective adenosine A2A receptor antagonist. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). It displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM).
CSN11901 SCH-58261 160098-96-4 SCH 58261 is a potent and selective A2a adenosine receptor antagonist with Ki of 2.3 nM and 2 nM for rat A2a and bovine A2a, respectively.
CSN21946 Proxyphylline 603-00-9 Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles.
CSN11787 Propentofylline 55242-55-2 Propentofylline, a xanthine derivative with purported neuroprotective effects, acts as a c-AMP phosphodiesterase inhibitor, a nerve growth factor stimulator, an adenosine transport inhibitor and a non-selective adenosine receptor antagonist.
CSN12717 Preladenant 377727-87-2 Preladenant is a highly selective and competitive A2A receptor antagonist with Ki value of 1.1nM, used in trials studying the treatment of brain diseases, such as parkinson disease, movement disorders, antipsychotic agents and parkinsonian disorders.
CSN23050 PQ 69 910045-32-8 PQ 69 is a potent and selective A1 receptor inverse agonist taht exhibits high binding affinity at A1 receptor with Kis of 0.07 and 0.96 nM for rat and human receptors respectively.
CSN23113 SDZ WAG 994 130714-47-5 Potent, selective A1 agonist
CSN23153 TC-G 1004 1061747-72-5 Potent and selective A2A antagonist
CSN16615 Norisoboldine 23599-69-1 Norisoboldine is an isoquinoline alkaloid isolated and purfied from the roots of Lindera aggregata, which acts as an AhR agonist, and enhances the function of the adenosine A1 receptor.
CSN20000 Neladenoson Dalanate 1239309-58-0 Neladenoson dalanate is a potent and selective adenosine A1 receptor agonist, and potentially useful for treatment of cardiovascular diseases.
CSN18541 N6-[2-(4-Aminophenyl)ethyl]adenosine 89705-21-5 N6-[2-(4-Aminophenyl)ethyl]adenosine is a potent, non-selective A3 adenosine receptor agonist.
CSN22994 N6-Cyclopentyladenosine 41552-82-3 N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 2.3 nM for human A1 receptor.
CSN11502 N6-Cyclohexyladenosine 36396-99-3 N6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM).
CSN18631 N-[(4-Aminophenyl)methyl]adenosine 95523-13-0 N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor, with Ki of 29 nM for rat ecto-5′-nucleotidase.
CSN25517 N-(2-Hydroxyethyl)adenosine 4338-48-1 N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action.
CSN22989 MRS 3777 Hemioxalate 1186195-57-2 MRS 3777 Hemioxalate is a high affinity adenosine A3 receptor antagonist with Ki of 47 nM.
CSN22988 MRS 1754 264622-58-4 MRS 1754 is a selective adenosine A2B receptor antagonist with Ki of 1.97 nM for hA2B.
CSN22987 MRS 1706 264622-53-9 MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist with Ki of 1.39 nM.
CSN18529 LUF6000 890087-21-5 LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).
CSN19808 LAS38096 851371-22-7 LAS38096 is a potent, selective, and efficacious A2B adenosine receptor antagonist.
CSN22873 KW 3902 136199-02-5 KW 3902 is a Selective adenosine A1 receptor antagonist with Ki of 0.19 nM.
CSN12709 Istradefylline 155270-99-8 Istradefylline is a very potent, selective and orally active adenosine A2A receptor antagonist (Ki=2.2 nM) in experimental models of Parkinson's disease.
CSN22860 ISAM 140 932191-62-3 ISAM 140 is a high affinity A2B receptor antagonist with Ki of 3.49 nM.
CSN23107 SCH 202676 Hydrobromide 265980-25-4 Inhibitor of ligand binding to G-protein-coupled receptors
CSN16958 IB-MECA 152918-18-8 IB-MECA is an agonist of the adenosine A3 receptor with EC50 values of 0.11 μM. IB-MECA is a potent and selective A3 adenosine receptor agonist with Ki value of 1.1, 54 and 56 nM for A3, A1 and A2A receptors, respectively, which possessing cardioprotective effect and reduces infarct size upon reperfusion in rats.
CSN22848 HEMADO 403842-38-6 HEMADO is a high affinity and selective adenosine A3 receptor agonist with Ki of 1.1 nM for human A3.
CSN17618 GR79236 124555-18-6 GR79236 is a highly potent and selective adenosine A1 receptor agonist (Ki = 3.1 nM) that has analgesic and anti-inflammatory actions in humans and animals.
CSN10909 Enprofylline 41078-02-8 Enprofylline is a xanthine derivative used in the treatment of asthma, which acts as a bronchodilator.
CSN23120 SLV 320 251945-92-3 Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1].
CSN21199 CPI444 1202402-40-1 CPI-444 is an orally administered antagonist of the adenosine A2A receptor. Upon oral administration, CPI-444 binds to adenosine A2A receptors expressed on the surface of immune cells, including T-lymphocytes, natural killer (NK) cells, macrophages and dendritic cells (DCs).
CSN10605 CGS 21680 120225-54-9 CGS 21680 is an adenosine A2 receptor agonist with IC50 of 22 nM, exhibits 140-fold over A1 receptor.
CSN18682 CGS 21680 HCl 124431-80-7 CGS 21680 HCl is A2A adenosine receptor agonist with Ki value of 27 nM, which can be used to distinguish A2A- and A2B-mediated effect and shows affinity for both A1 and A3 adenosine receptors.
CSN10537 Capadenoson 544417-40-5 Capadenoson is an oral active, potent and selective adenosine A1 receptor agonist.
CSN23897 BAY-545 1699717-32-2 BAY-545 is a structure-optimizd adenosine receptor A2B antagonist with IC50 value of of 59 nM.
CSN24164 BAY-218 2162982-11-6 BAY-218 is an AHR antagonist.
CSN22708 BAY 60-6583 910487-58-0 BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor.
CSN21468 Alloxazine 490-59-5 Alloxazine is a selective antagonist of A2B adenosine receptor.
CSN21333 Adenosine Antagonist-1 431040-19-6 Adenosine antagonist-1 is an adenosine A3 receptor (AA3R) antagonist.
CSN25244 Adenosine amine congener   96760-69-9 Adenosine amine congener hydrate is a potent aqueous-soluble A1 adenosine receptor agonist with Ki value of 0.85nM for binding against [3H]N6-cyclohexyladenosine in rat cerebral cortex membranes.
CSN12871 Acefylline 652-37-9 Acefylline is an adenosine receptor antagonist, a stimulant drug of the xanthine chemical class.
CSN17909 AB-MECA 152918-26-8 AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors.
CSN17107 2-Cl-IB-MECA 163042-96-4 2-Cl-IB-MECA is a highly selective A3 adenosine receptor agonist with Ki value of 0.33nM, displaying 2500- and 1400-fold selectivity over A1 and A2A receptors, respectively.
CSN22617 (±)-5'-Chloro-5'-deoxy-ENBA 103626-26-2 (±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist with Ki of 0.51 nM.
CSN25359 2-Chloroadenosine 146-77-0
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