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CGRP Receptor

CGRP Receptor

货号 产品名 CAS号 信息
CSN21471 HCGRP-(8-37) 119911-68-1 α-CGRP(8-37), huma is a human calcitonin gene-related peptide (hCGRP) fragment and also an antagonist of CGRP receptor.
CSN32914 Vazegepant 1337918-83-8 Zavegepant is a highly potent, selective and structurally unique small molecule CGRP receptor antagonist.
CSN22530 Ubrogepant 1374248-77-7 Ubrogepant is an oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine.
CSN26144 CGRP antagonist 4 217438-17-0 SB-268262 is a selective non-peptide CGRP antagonist with IC50 value of 0.83nM for inhibition of CGRP-activated adenylyl cyclase stimulation in SK-N-MC cell membranes.
CSN24283 Rat CGRP-(8-37) TFA salt N/A Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonist.
CSN18095 Olcegepant 204697-65-4 Olcegepant is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor (IC50= 0.03 nM).
CSN13170 MK-3207 957118-49-9 MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC50= 0.12 nM; Ki value= 0.024 nM), showing highly selective versus human AM1, AM2, CTR, and AMY3.
CSN13169 MK-3207 HCl 957116-20-0 MK-3207 HCl is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, and AMY3
CSN13778 Telcagepant 781649-09-0 MK-0974 is a highly potent, selective, and orally bioavailable CGRP receptor antagonist with Ki values of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors respectively, displaying > 1500-fold lower affinity for the canine and rat receptors.
CSN24284 HCGRP-(8-37) TFA salt N/A HCGRP-(8-37)
CSN22373 CGRP antagonist 1 1123757-49-2 CGRP antagonist 1 is a highly potent CGRP receptor antagonist with a Ki and IC50 of 35 and 57 nM, respectively.
CSN17659 (5S,6S,9R)-5-Amino-6-(2,3-difluorophenyl)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-9-yl 4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxylate 1289023-67-1 BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.
CSN51428 Atogepant 1374248-81-3
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