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PDK-1

PDK-1

货号 产品名 CAS号 信息
CSN17521 PS48 1180676-32-7 PS48 is a phosphoinositide-dependent protein kinase-1 (PDK1) activator with Kd value of 10.3 μM and binds exclusively to the PIF-binding pocket of PDK1, distinct from the ATP binding site.
CSN17379 PDK1 Inhibitor 1001409-50-2 PDK1 inhibitor is a potent and selective inhibitor of PDK1 with potential as anticancer agent.
CSN12988 OSU-03012 742112-33-0 OSU-03012 is a potent inhibitor of recombinant PDK-1 with IC50 of 5 μM and 2-fold increase in potency over OSU-02067.
CSN17589 GSK2334470 1227911-45-6 GSK2334470 is a PDK1 inhibitor with IC50 of ~10 nM, with no activity at other close related AGC-kinases.
CSN12711 BX795 702675-74-9 BX795 is a potent and selective dual inhibitor of TBK1/PDK1 with IC50s of 2 nM/6 nM respectively, also inhibit Aurora B and IκB kinase ε (IKKε).
CSN19146 BX517 850717-64-5 BX517 is a potent and selective inhibitor of PDK1 with IC50 of 6 nM.
CSN17175 BX-912 702674-56-4 BX-912 is a selective inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1) with IC50 of 12 nM, showing > 10 fold selectivity over PKA, PKC, C-Kit, EGFR etc.
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