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Transforming Growth Factor beta (TGFβ) Receptor

TGF-beta Receptor

货号 产品名 CAS号 信息
CSN13732 SB-505124 HCl 356559-13-2 SB-505124 HCl is a selective inhibitor of TGFβR for ALK4, ALK5 with IC50 of 129 nM and 47 nM, respectively, also inhibits ALK7, but does not inhibit ALK1, 2, 3, or 6.
CSN18520 R268712 879487-87-3 R268712 is a potent and selective inhibitor of ALK5 with an IC50 of 2.5 nM.
CSN15840 ML347 1062368-49-3 ML347 is a highly selective ALK1/ALK2 inhibitor with IC50s of 46/32 nM and shows > 300-fold selectivity for ALK2 vs. ALK3.
CSN13478 LY2109761 700874-71-1 LY2109761 is a selective TGF-β receptor type I/II (TβRI/II) dual inhibitor with Ki of 38 nM and 300 nM, respectively and is shown to negatively affect the phosphorylation of Smad2.
CSN13876 LDN-214117 1627503-67-6 LDN-214117 is a potent and selective ALK2 inhibitor with IC50 of 22 nM with > 100 fold selectivity for ALK5, and also inhibits BMP6 (IC50=100 nM).
CSN22554 LDN-193189 2HCl 1435934-00-1 LDN-193189 2HCl is a potent and selective ALK2 and ALK3 inhibitor.
CSN13159 GW788388 452342-67-5 GW788388 is a selective ALK5 inhibitor with IC50 of 18 nM and also inhibits TGF-β type II receptor and activin type II receptor.
CSN22227 EW-7197 HCl 1352610-25-3 EW-7197 HCl is a small-molecule ATP-competitive inhibitor of TGFβRI (ALK5) with an IC50 of 12.9 nM.
CSN19475 A 77-01 607737-87-1 A77-01 is a potent inhibitor of TGF-β type I receptor superfamily activin-like kinase ALK5 with IC50 of 25 nM.
CSN13090 A 83-01 909910-43-6 A 83-01 is a selective inhibitor of TGF-β type I receptor ALK5 kinase, type I activin/nodal receptor ALK4 and type I nodal receptor ALK7, with IC50 values of 12, 45 and 7.5 nM, respectively.
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