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GABA Receptor

GABA Receptor

货号 产品名 CAS号 信息
CSN13133 Thymol 89-83-8 Thymol, a natural product isolated and purified from the herbs of Thymus serpyllum L., is a positive allosteric modulator of human GABAA receptors and a homo-oligomeric GABA receptor from Drosophila melanogaster.
CSN11911 Securinine 5610-40-2 Securinine, a natural product isolated and purified from the leaves and twigs of Securinega suffruticosa with antifungal activity, induces apoptosis in human leukemia HL-60 cells, is a promising monocytic differentiation inducing agent for Acute Myeloid Leukemia (AML).
CSN20452 Ro 15-3890 84378-44-9 Ro 15-3890 is an antagonist of benzodiazepine receptor. It is a main metabolite of Ro 15-1788 (flumazenil).
CSN19514 Oxiracetam(Random Configuration) 62613-82-5 Oxiracetam is a derivative of gamma-aminobutyric acid (GABA) and used as a nootropic drug to improve memory and learning.
CSN23642 MRX-1024 348-67-4 MRX-1024 can inhibit the activation of GABAA receptor and exhibit relieving effect on hearing loss. It can used as a chemoprotective agent.
CSN25408 Isonipecotic acid 498-94-2 Isonipecotic acid is a specific GABAA receptor agonist.
CSN25409 Ganaxolone 38398-32-2 Ganaxolone, also known as CCD 1042 and C1042, is a CNS-selective GABAA modulator that acts on well-characterized targets in the brain known to have anxiolytic and anticonvulsant effects. Ganaxolone protects against seizures in diverse animal models, including the pentylenetetrazol, 6 Hz and amygdala kindling models. Ganaxolone is a positive allosteric modulator of the action of the GABAA receptor and, unlike benzodiazepines, there does not appear to be tolerance to the anticonvulsant effects of ganaxolone.
CSN27585 N-Methyl-9H-pyrido[3,4-b]indole-3-carboxamide 78538-74-6 FG 7142 (ZK 39106; LSU-65), a non-selectively benzodiazepine inverse agonist, has high affinity for the α1 subunit-containing GABAA receptor (Ki=91 nM). FG 7142 (ZK 39106; LSU-65) also modulates GABA-induced chloride flux at GABAA receptors expressing the α1 subunit (EC50= 137 nM). FG 7142 (ZK 39106; LSU-65) can increase tyrosine hydroxylation and cause upregulation of β-adrenoceptors in mouse cerebral cortex .
CSN21178 CGP52432 139667-74-6 CGP52432 is an antagonist of GABAB receptor with an IC50 of 85 nM.
CSN17089 Bemegride 64-65-3 Bemegride can stimulate central nervous system and release barbiturate poisoning.
CSN23429 L-Glutamic Acid 56-86-0 (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system.
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