欢迎来到 CSNpharm! 产品仅用于科研!
首页 Compound Arrays 促销产品
400-920-2911 sales@csnpharm.cn    

GABA Receptor

GABA Receptor

货号 产品名 CAS号 信息
CSN19031 U93631 152273-12-6 U93631 is a ligand of GABAA receptor ligand (IC50 = 100 nM) which can induce a rapid decay of GABA-induced chloride currents.
CSN12084 Tiagabine 115103-54-3 Tiagabine is an anti-convulsive medication and a selective gamma-aminobutyric acid (GABA) reuptake inhibitor.
CSN12085 Tiagabine HCl 145821-59-6 Tiagabine HCl is an inhibitor of gamma-aminobutyric acid (GABA) reuptake (IC50 = 67 nM in vivo) with anticonvulsant effect.
CSN13133 Thymol 89-83-8 Thymol, a natural product isolated and purified from the herbs of Thymus serpyllum L., is a positive allosteric modulator of human GABAA receptors and a homo-oligomeric GABA receptor from Drosophila melanogaster.
CSN12077 Thiocolchicoside 602-41-5 Thiocolchicoside is a small molecule muscle relaxant and anti-inflammatory agent, shown to function as a competitive GABAA (gamma-aminobutyric acid type A) receptor antagonist.
CSN11911 Securinine 5610-40-2 Securinine, a natural product isolated and purified from the leaves and twigs of Securinega suffruticosa with antifungal activity, induces apoptosis in human leukemia HL-60 cells, is a promising monocytic differentiation inducing agent for Acute Myeloid Leukemia (AML).
CSN19979 Sanggenon D 81422-93-7 Sanggenon D, a natural product isolated and purified from the root bark of Morus alba L.
CSN19798 Ro 48-6791 172407-17-9 Ro 48-6791 is a GABA receptor agonist potentially for the use of anesthesia.
CSN11846 Rilmazafone 99593-25-6 Rilmazafone is a water-soluble benzodiazepine prodrug developed in Japan. It has sedative and hypnotic effects.
CSN17380 Remimazolam Benzenesulfonate 1001415-66-2 Remimazolam benzenesulfonate is a GABA agonist that acts on GABA receptor, specifically GABA-alpha.
CSN10515 Progabide 62666-20-0 Progabide is an analog and prodrug of gamma-aminobutyric acid. It is commonly used in the treatment of epilepsy with agonistic activity for both the GABAA and GABAB receptors. Progabide has been investigated for many diseases besides epilepsy, including Parkinson's disease, schizophrenia, clinical depression and anxiety disorder with varying success.
CSN11770 Primidone 125-33-7 Primidone is a pyrimidinedione derivative with anticonvulsant activity.
CSN11714 Phytol 150-86-7 Phytol can activite PPARα and attenuate the inflammatory response by inhibiting neutrophil migration and oxidative stress. Phytol is isolated from the leaves of black tea and acts as an aromatic ingredient.
CSN23337 Phenibut 1078-21-3 Phenibut, a GABA analogue, is a central nervous system depressant with anxiolytic and sedative effects.
CSN11659 Pazinaclone 103255-66-9 Pazinaclone is a sedative and anxiolytic drug in the cyclopyrrolone family of drugs.
CSN19514 Oxiracetam(Random Configuration) 62613-82-5 Oxiracetam is a derivative of gamma-aminobutyric acid (GABA) and used as a nootropic drug to improve memory and learning.
CSN18575 Lorediplon 917393-39-6 Lorediplon, non-benzodiazepine hypnotic drug, acts as a modulator of GABAA receptor with the effect of promoting sleep.
CSN19849 Loreclezole HCl 2227372-56-5 Loreclezole HCl is a subtype-selective GABAA receptor modulator. Acts as a positive allosteric modulator of β2 or β3-subunit containing receptors.
CSN16300 L-Cycloserine 339-72-0 L-cycloserine is an inhibitor of serine palmitoyltransferase and block sphingosine biosynthesis. It has antibiotic effective against mycobacterium tuberculosis.
CSN15698 L-838,417 286456-42-6 L-838417 is a subtype-selective GABAA receptor partial agonist. L-838417 selectively binds to α1, α2, α3 and α5 subunits (Ki values are 0.79, 0.67, 0.67 and 2.25 nM respectively) but displays no efficacy at α1 (α1-sparing). L-838417 exhibits non-sedative anxiolytic, antinociceptive and anti-inflammatory activity.
CSN17671 L-655,708 130477-52-0 L-655708 is a potent α5 subunit-selective GABAA receptor inverse agonist (Ki = 0.45 nM).
CSN12568 Ginkgolide A 15291-75-5 Ginkgolide A is an antagonist of g-aminobutyric acid (GABA) with Ki of 14.5 μM and also can activate PAF. It is purified from the leaves of ginkgo biloba tree.
CSN16036 Gaboxadol HCl 85118-33-8 Gaboxadol HCl is a systemically active GABAA receptor agonist and GABAA-ρ receptor antagonist. Displays antinociceptive, anticonvulsant and sedative effects. Hypnotic agent that enhances delta activity within non-REM sleep in rats.
CSN15872 Gabazine Hydrobromide 104104-50-9 Gabazine hydrobromide is a drug that acts as an antagonist at GABAA receptors. It is used in scientific research and has no role in medicine, as it would be expected to produce convulsions if used in humans.
CSN12825 Gabapentin 60142-96-3 Gabapentin is an analogue of GABA that used to treat seizures and neuropathic pain.
CSN16669 Gabapentin HCl 60142-95-2 Gabapentin is a GABA analogue, used to treat seizures and neuropathic pain.
CSN20431 EVT-201 308239-86-3 EVT-201 is a benzodiazepine derivative drug and partial positive allosteric modulator of the benzodiazepine site of the GABA receptor.
CSN10962 Etifoxine 21715-46-8 Etifoxine is potentiator of GABAA receptor function in cultured neurons.
CSN18338 Etifoxine HCl 56776-32-0 Etifoxine HCl is a potentiator of β2 or β3 subunit-containing GABAA receptor that promotes axonal regeneration. It shows anxiolytic activity with no effects.
CSN16005 Cloxacillin Sodium 642-78-4 Cloxacillin is a semisynthetic antibiotic that belongs to the group of the isoxazolylpenicillins and is used to treat infections caused by species of staphylococci that produce beta-lactamase due to its inhibitory effects on beta-lactamase binding.
CSN10673 Clomethiazole 533-45-9 Clomethiazole can act as an agonist of GABAA and modulator of glycine receptor. It is a sedative used in the treatment of alcohol withdrawal.
CSN18672 CGS-9896 77779-36-3 CGS-9896 is an anxiolytic drug used in scientific research.
CSN17089 Bemegride 64-65-3 Bemegride can stimulate central nervous system and release barbiturate poisoning.
CSN10524 Baclofen 1134-47-0 Baclofen, a gamma-amino-butyric acid derivative, is a selective GABAB agonist with IC50 of 200 nM which used as a skeletal muscle relaxant.
CSN25262 AZD7325 942437-37-8 AZD-7325 is a GABA-Aα2,3 selective receptor modulator.
CSN16275 AWD 131-138 188116-07-6 AWD 131-138 is a partial agonist of benzodiazepine receptor with effective anticonvulsant and anxiolytic properties.
CSN10227 Afloqualone 56287-74-2 Afloqualone is an agonist of GABA receptor and has muscle-relaxant effects.
CSN10198 Acamprosate Calcium 77337-73-6 Acamprosate calcium is an agonist of GABA receptor. It can act as a modulator of glutamatergic systems and reduce alcohol consumption in animal models of alcohol addiction.
CSN23521 6-Methyl-2-phenyl-4H-chromen-4-one 29976-75-8 6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.
CSN23331 6-Hydroxyflavone 6665-83-4 6-Hydroxyflavone is a naturally occurring flavone, with anti-inflammatory activity. 6-Hydroxyflavone exhibits inhibitory effect towards bovine hemoglobin (BHb) glycation. 6-Hydroxyflavone can activate AKT, ERK 1/2, and JNK signaling pathways to effectively promote osteoblastic differentiation. 6-Hydroxyflavone inhibits the LPS-induced NO production[1] [2].
CSN23335 5-methoxyflavone 42079-78-7 5-Methoxyflavone, belonged to Flavonoid family, is a DNA polymerase-beta inhibitor and neuroprotective agent against beta-amyloid toxicity. possess central nervous system (CNS) depressant effect mediated through the ionotropic GABAA receptors.
CSN12782 4-Aminobutyric Acid 56-12-2 4-Aminobutyric acid exhibits inhibitory activity on central nervous system (CNS). It is a natural neurotransmitter.
CSN23429 L-Glutamic Acid 56-86-0 (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system.
CSN10435 (+)-Bicuculline 485-49-4 (+)-Bicuculline is an antagonist of GABAA receptor with IC50 of 2 μM and also shows inhibition of Ca(2+)-activated potassium channels.
CSN25408 Isonipecotic acid 498-94-2
CSN25410 Saclofen 125464-42-8
CSN25409 Ganaxolone 38398-32-2
<< PREV 1 2 3 NEXT >>