欢迎来到 CSNpharm! 产品仅用于科研!
首页 400-920-2911

P2Y Receptor

P2Y Receptor

货号 产品名 CAS号 信息
CSN23371 UDP disodium salt 27821-45-0 UDP disodium salt is an endogenous agonist of P2Y receptor which preferentially activates P2Y6. It exhibis antagonistic effect on the P2Y14 receptor.
CSN12090 Ticlopidine 55142-85-3 Ticlopidine is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (ADP) receptor inhibitor.
CSN13719 Ticlopidine HCl 53885-35-1 Ticlopidine HCl is an adenosine diphosphate (ADP) receptor inhibitor that against platelet aggregation with IC50 of ~2 μM.
CSN12826 Ticagrelor 274693-27-5 Ticagrelor is a reversibly and oral active P2Y12 receptor antagonist with Ki of 2 nM, also inhibits CYP2C9 and midazolam 4-hydroxylation with IC50 of 10.5 μM and 8.2 μM respectively.
CSN12020 Suramin Sodium 129-46-4 Suramin sodium salt is a polysulfonated naphthylurea that inhibits the binding of calmodulin to recognition sites on the ryanodine receptor-1 (IC50 = 4.9 μM), blocks G protein coupling to GPCRs, and non-selectively antagonizes P2 purinergic receptors(10-100 μM).
CSN17880 Suramin 145-63-1 Suramin is a polysulfonated naphthylurea that inhibits the binding of calmodulin to recognition sites on the ryanodine receptor-1 (IC50 = 4.9 μM), blocks G protein coupling to GPCRs, and non-selectively antagonizes P2 purinergic receptors(10-100 μM).
CSN20191 PSB-0739 Sodium 1052087-90-7 PSB-0739 is an extremely potent and selective competitive P2Y12 receptor antagonist (pA2 of 9.8).
CSN18256 Prasugrel Maleic Acid 389574-20-3 Prasugrel maleic acid is a platelet inhibitor with IC50 value of 1.8 μM.
CSN16171 Prasugrel 150322-43-3 Prasugrel is a platelet inhibitor with IC50 value of 1.8 μM.
CSN12325 Prasugren HCl 389574-19-0 Prasugrel hydrochloride is a platelet inhibitor with IC50 value of 1.8 μM.
CSN13178 N6-(4-Hydroxybenzyl)-adenosine 110505-75-4 N6-(4-Hydroxybenzyl)adenosine is an inhibitor of platelet aggregation induced in vitro by collagen and their activity range was demonstrated (IC50: 6.77-141 μM).
CSN11479 MRS 2578 711019-86-2 MRS2578 is a potent and selective P2Y6 nucleotide receptor antagonist with IC50 of 37 nM, exhibits insignificant activity at P2Y1, P2Y2, P2Y4,and P2Y11 receptors.
CSN20190 MRS2395 491611-55-3 MRS2395 is an antagonist for the P2Y12 purinoceptor, which causes platelet aggregation in rats via ADP induction.
CSN13637 Clopidogrel Thiolactone 1147350-75-1 Clopidogrel thiolactone is a P2Y12 receptor inhibitor, is a potent antiplatelet agent.
CSN10679 Clopidogrel Bisulfate 135046-48-9 Clopidogrel is an inhibitor of platelet aggregation that is used to decrease the risk of myocardial infarction and stroke in patients known to have atherosclerosis. Clopidogrel has been linked to rare instances of idiosyncratic, clinically apparent acute liver injury.
CSN15727 Clopidogrel 113665-84-2 Clopidogrel is a P2Y12 receptor blocker (IC50 = 100 nM).
CSN15854 Clopidogrel Hydrogen Sulfate 120202-66-6 Clopidogrel Hydrogen Sulfate is the functional enantiomer of clopidogrel and a potent P2Y12 receptor antagonist.
CSN22574 AR-C 69931 Tetrasodium 163706-36-3 Cangrelor is a potent and competitive P2Y12 receptor inhibitor that inhibits of ADP-induced platelet aggregation.
CSN21162 BPTU 870544-59-5 BPTU allosteric antagonist of P2Y1 wtih IC50 of 0.06-0.3 μM with antithrombotic effect and reduces platelet aggregation.
CSN18578 AZD1283 919351-41-0 AZD1283 is a potent antagonist of the P2Y12 receptor with EC50 of 3.0 ug/kg/min, TI > 10 and with binding IC50 of 11 nM.
CSN20192 AR-C 66096 Tetrasodium 145782-74-7 AR-C 66096 tetrasodium is a potent and selective P2Y12 receptor antagonist which blocks ADP-induced inhibition of adenylyl cyclase in vitro (pKB =7.6) and inhibits ADP-induced aggregation of washed human platelets (pIC50 = 8.16).
CSN23813 Diquafosol Tetrasodium 211427-08-6
<< PREV 1 NEXT >>