欢迎来到CSNpharm!产品仅用于科研!

400-920-2911 sales@csnpharm.cn

0

CRTH2

CRTH2

货号 产品名 CAS号 信息
CSN24302 MK-7246 1218918-62-7 MK-7246 is a potent and selective CRTH2 antagonist with Ki value of 2.5nM.
CSN20221 MK-2305 2101206-49-7 MK-2305 is a GPR40 partial agonist lower fasting glucose in the Goto Kakizaki rat via suppression of endogenous glucose production.
CSN18830 Fevipiprant 872365-14-5 Fevipiprant is a selective, potent, reversible competitive CRTh2 antagonist with an in vitro dissociation constant KD value of 1.1nM at the CRTh2 receptor and an IC50 value of 0.44 nM for inhibition of PGD2-induced eosinophil shape change in human whole blood.
CSN22382 CRTh2 antagonist 1 1379445-54-1 CRTh2 antagonist 1是 CRTh2 的拮抗剂,IC50 值为89 nM。
CSN26623 CAY10471 Racemate 844639-57-2 CAY 10471 is a potent, highly selective CRTH2/DP 2 receptor antagonist. CAY10471 binds to the human CRTH2/DP2, DP1, and TP receptors with Ki values of 0.6, 1200, and >10,000 nM. Cat#531655 is a racemic mixture of CAY10471.
CSN16482 AZD1981 802904-66-1 AZD1981 is a potent and selective CRTh2 antagonist and displaces radio-labelled PGD2 from human recombinant DP2 with high potency (pIC50 = 8.4).
CSN22681 Vidupiprant 1169483-24-2 AMG 853 is a potent dual CRTH2 and prostaglandin D2 (PGD2) receptor antagonist (IC50 values are 8 and 35 nM, respectively in plasma).
CSN25231 AM211 1175526-27-8 AM211 is a potent and selective prostaglandin D2 receptor type 2 antagonist with IC50 value of 4.9nM.
<< PREV 1 NEXT >>
联系
我们