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5-HT Receptor

5-HT Receptor

货号 产品名 CAS号 信息
CSN12245 Zolmitriptan 139264-17-8 Zolmitriptan is an agonist of 5-HT1B/5-HT1D receptors with anti-migraine properties.
CSN12174 Urapidil 34661-75-1 Urapidil is a sympatholytic antihypertensive drug.
CSN12150 Trimipramine Maleate 521-78-8 Trimipramine maleate is a serotonin transport and norepinephrine uptake blocker, is a tricyclic antidepressant (TCA) with antipsychotic and sedative properties.
CSN12032 Tandospirone 87760-53-0 Tandospirone is a potent and selective 5-HT1A receptor partial agonist (Ki = 27 nM) that displays selectivity over SR-2, SR-1C, α1-adrenergic, α2-adrenergic, D1 and D2 receptors (Ki values ranging from 1300-41000 nM).
CSN12475 Sumatriptan Succinate 103628-48-4 Sumatriptan Succinate can selectively bind to and activate 5-HT1 receptors.
CSN11037 Sevoflurane 28523-86-6 Sevoflurane is a sweet-smelling, nonflammable, highly fluorinated methyl isopropyl ether used as an inhalational anaesthetic for induction and maintenance of general anesthesia.
CSN11920 Setiptiline 57262-94-9 Setiptiline is a serotonin receptor antagonist.
CSN10540 Serotonin HCl 153-98-0 Serotonin HCl is an endogenous 5-HT receptor agonist.
CSN11875 Rupatadine 158876-82-5 Rupatadine is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 μM (rabbit platelet membranes/guinea pig cerebellum membranes).
CSN11853 Rizatriptan 144034-80-0 Rizatriptan a selective 5-HT1 receptor agonist used for the treatment of migraine headaches.
CSN11849 Ritanserin 87051-43-2 Ritanserin is a serotonin receptor antagonist which was never marketed for clinical use but has been used in scientific research.
CSN10944 Quetiapine Sulfoxide 2HCl 329218-11-3 Quetiapine sulfoxide is a metabolite of quetiapine, an atypical antipsychotic approved for the treatment of schizophrenia, bipolar disorder, and along with an antidepressant to treat major depressive disorder.
CSN11813 Quetiapine 111974-69-7 Quetiapine is an atypical antipsychotic used in the treatment of schizophrenia, bipolar I mania, bipolar II depression, bipolar I depression.
CSN11812 Quetiapine Fumarate 111974-72-2 Quetiapine Fumarate is a second-generation antipsychotic with affinity for D2, 5-HT2A, H1, alpha 1 and 5-HT1A receptors, used as an atypical antipsychotic for the treatment of schizophrenia, bipolar disorder, and major depressive disorder.
CSN11795 Prucalopride 179474-81-8 Prucalopride is a high-affinity 5-HT4 receptor agonist。
CSN10104 Pizotifen Malate 5189-11-7 Pizotifen Malate is a benzocycloheptene-based drug used to reduce the frequency of recurrent migraine headacheswith, with high affinity for 5-HT and dopamine receptors (Kis = 7.94 and 2.4 nM for 5-HT2C and D2, respectively).
CSN10126 Pizotifen 15574-96-6 Pizotifen is a highly selective 5-HT receptor blocking agent, which is a benzocycloheptane based drug.
CSN11724 Pindolol 13523-86-9 Pindolol is a nonselective β-blocker with partial beta-adrenergic receptor agonist activity, also functions as a 5-HT1A receptor weak partial agonist / antagonist (Ki=33nM).
CSN11590 Nuciferine 475-83-2 Nuciferine is naturally occuring alkaloid found in the plants Nymphaea caerulea and Nelumbo nucifera as a potent inverse agonist at human 5-HT7 receptor.
CSN10097 Naftidrofuryl Oxalate 3200-06-4 Naftidrofuryl oxalate is a drug used in the management of peripheral and cerebral vascular disorders as a vasodilator, enhance cellular oxidative capacity, and may also be a 5-HT2 receptor antagonist.
CSN11510 Nafronyl 31329-57-4 Naftidrofuryl is a vasodilator used in the management of peripheral and cerebral vascular disorders.
CSN11473 Mosapride Citrate 112885-42-4 Mosapride Citrate is both a selective 5HT4 agonist and a 5HT3 antagonist, use as a gastroprokinetic agent.
CSN11451 Mirtazapine 85650-52-8 Mirtazapine is a potent tetracyclic antidepressant.
CSN12364 Lurasidone HCl 367514-88-3 Lurasidone HCl is a multiple-target antagonist of dopamine D2 receptor, 5-HT2 receptor, 5-HT7 receptor, adrenergic α2A and α2C receptors, also works as a partial 5-HT1A receptor agonist. It used as an atypical antipsychotic medication for the treatment of several mental disorders.
CSN12407 Loxapine 1977-10-2 Loxapine succinate is a D2DR and D4DR inhibitor, serotonergic receptor antagonist and also a dibenzoxazepine anti-psychotic agent.
CSN11251 Ketanserin Tartrate 83846-83-7 Ketanserin Tartrate is a water soluble selective 5-HT2A and 5-HT1D antagonist.
CSN11471 Indeloxazine HCl 65043-22-3 Indeloxazine hydrochloride is an antidepressant and cerebral activator.
CSN11195 Imipramine HCl 113-52-0 Imipramine HCl is a tricyclic inhibitor of both serotonin and norepinephrine transporters with Ki values of 7.7 nM and 67 nM, respectively.
CSN11019 Flibanserin 167933-07-5 Flibanserin is a serotonergic antidepressant used to treat hypoactive sexual desire disorder. It is also a P-Glycoprotein Inhibitor.
CSN10898 Eletriptan Hydrobromide 177834-92-3 Eletriptan Hydrobromide is a high-affinity agonist of 5-HT1B and 5-HT1D receptor with Ki values of 0.92 nM and 3.14 nM, respectively.
CSN10816 Dihydroergotamine Mesylate 6190-39-2 Dihydroergotamine mesylate is an ergot alkaloid used to treat migraines.
CSN10727 Cyproheptadine Hydrochloride Sesquihydrate 41354-29-4 Cyproheptadine Hydrochloride Sesquihydrate is a serotonin antagonist and a histamine H1 blocker used as antipruritic, appetite stimulant, antiallergic, and for the post-gastrectomy dumping syndrome, etc.
CSN10716 Cyclobenzaprine HCl 6202-23-9 Cyclobenzaprine HCl is a 5-HT2 receptor antagonist as a skeletal muscle relaxant and a central nervous system (CNS) depressant with elimination half-life of ‎32 hours.
CSN10686 Clozapine N-oxide 34233-69-7 Clozapine N-oxide is a major metabolite of clozapine noted to decrease SR-2A(5-HT2 serotonin receptor) density in vitro.
CSN10658 Citalopram Hydrobromide 59729-32-7 Citalopram Hydrobromide is a highly selective and potent 5-HT uptake inhibitor with no effect on noradrenalin or dopamine uptake.
CSN10655 Cisapride 81098-60-4 Cisapride is a 5-HT4 agonist which can stimulate intestinal ACh release.
CSN10625 Chlorpromazine HCl 69-09-0 Chlorpromazine HCl is a multiple-target antagonist for dopamine D2, 5HT2A, potassium channel and sodium channel with Ki values of 363 nM and 8.3 nM for D2 and 5HT2A, respectively.
CSN10511 Buspirone HCl 33386-08-2 Buspirone hydrochloride is an anxiolytic psychotropic drug, is used to treat generalized anxiety disorder (GAD).
CSN10491 Bromperidol 10457-90-6 Bromperidol is a butyrophenone derivative, is a potent and long-acting neuroleptic, used as an antipsychotic in the treatment of schizophrenia.
CSN10484 BRL-15572 2HCl 193611-72-2 BRL-15572 2HCl is a selective h5-HT1D antagonist, displaying 60-fold selectivity over h5-HT1B and exhibiting little or no affinity for a range of other receptor types.
CSN10719 Blonanserin 132810-10-7 Blonanserin is a D2/5-HT2 receptor antagonist, atypical antipsychotic.
CSN12124 Asenapine 65576-45-6 Asenapine inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor(1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM.
CSN12463 Aripiprazole 129722-12-9 Aripiprazole is a multiple-target agent used to treat schizophrenia and bipolar disorder, working as both a silent antagonist and a high-efficacy partial agonist of D2 receptor, as well as works as a partial agonist of 5-HT1A/5-HT2A, 5-HT2 receptor,a potent inverse agonist of 5-HT2B receptor, a functional antagonist of 5-HT7 receptor.
CSN10289 Amitriptyline HCl 549-18-8 Amitriptyline HCl is a multiple-target molecular as an inhibitor of both 5-HT and NA reuptake (SNRI), and also a TrkA/B agonist.
CSN10268 Alprenolol HCl 13707-88-5 Alprenolol HCl is an antagonist of both 5-HT1A receptor and β-adrenoceptor.
CSN10249 Almotriptan Malate 181183-52-8 Almotriptan Malate a serotonin 5HT-1B/1D-receptor agonist with high affinity for the 5-HT(1B) and 5-HT(1D) receptors, used to treat migraine.
CSN10250 Almotriptan 154323-57-6 Almotriptan is a 5-HT1B/1D-receptor agonist used to treat migraine.
CSN23783 AVN492 1220646-23-0
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