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5-HT Receptor

5-HT Receptor

货号 产品名 CAS号 信息
CSN23195 WAY 208466 2HCl 1207064-61-6 WAY-208466 2HCl is a selective serotonin 5-HT6 receptor agonist.
CSN23171 Tropanserin 85181-40-4 Tropanserin is a selective 5-HT3 receptor antagonist.
CSN11037 Sevoflurane 28523-86-6 Sevoflurane is a sweet-smelling, nonflammable, highly fluorinated methyl isopropyl ether used as an inhalational anaesthetic for induction and maintenance of general anesthesia.
CSN23100 SB 258719 HCl 1217674-10-6 Selective 5-HT7 antagonist
CSN23114 SGS 518 Oxalate 445441-27-0 Selective 5-HT6 antagonist
CSN23197 WAY 629 HCl 57756-44-2 Selective 5-HT2C agonist
CSN23112 SDZ SER 082 Fumarate 1417343-80-6 Selective 5-HT2B/2C antagonist
CSN23140 Tandospirone HCl 99095-10-0 Selective 5-HT1A partial agonist
CSN23208 Zimelidine 2HCl 60525-15-7 Selective 5-HT uptake inhibitor
CSN23095 SB 215505 162100-15-4 SB215505 is a potent 5-HT2B/2C receptor antagonist (pKi values are 8.3, 7.66 and 6.77 for 5-HT2B, 5-HT2C and 5-HT2A respectively). It Increases wakefulness and motor activity in rats.
CSN23104 SB 399885 HCl 402713-81-9 SB-399885 hydrochloride is a 5-HT6 receptor antagonist.
CSN23105 SB 699551 864741-95-7 SB 699551 is a selective 5-ht5a receptor antagonist (pKi values are 8.3, < 6.0, < 6.0, < 6.0, < 5.5 and < 5.5 for 5-ht5a, 5-HT1B/D, 5-HT2A, 5-HT2C, 5-HT1A and 5-HT7 receptors respectively).
CSN23098 SB 243213 HCl 200940-23-4 SB 243213 hydrochloride is a selective and high-affinity 5-hydroxytryptamine (5-HT)2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. SB 243213 hydrochloride has improved anxiolytic profile[1].
CSN23096 SB 221284 196965-14-7 SB 221284 is potent, selective 5-HT2C/2B receptor antagonist. SB 221284 are pKi values are 6.4, 7.9 and 8.6 for 5-HT2A, 2B and 2C receptors respectively.
CSN23094 SB 206553 HCl 1197334-04-5 SB 206553 HCl is a potent and selective 5-HT2B/5-HT2C receptor antagonist (rat 5-HT2B pA2 = 8.89, human 5-HT2C pKi = 7.92). It displays > 80-fold selectivity over all other 5-HT receptor subtypes and a variety of other receptors (pKi < 6).
CSN23093 SB 204741 152239-46-8 SB 204741 is potent and selective 5-HT2B receptor antagonist (pA2 = 7.95). It displays ≥ 135-fold selectivity over 5-HT2C (pKi = 5.82), 5-HT2A (pKi < 5.2), 5-HT1A, 1D, 1E, 5-HT3 and 5-HT4 receptors.
CSN23092 SB 204070 148688-01-1 SB 204070A is a highly selective 5-HT4 receptor antagonist.
CSN23091 SB 203186 HCl 207572-69-8 SB 203186 HCl is potent 5-HT4 receptor antagonist with high affinity for human atrial 5-HT4 receptors.
CSN23073 RS 102221 HCl 187397-18-8 RS-102221 HCl is a highly potent, selective 5-HT2C receptor antagonist.
CSN23066 Ro 04-6790 202466-68-0 Ro 04-6790 is a potent and selective 5-HT6 receptor antagonist (pKi values are 7.26 and 7.35 at rat and human 5-HT6 receptors respectively). Ro 04-6790 displays no affinity at a range of other receptors (IC50 > 10 μM).
CSN11813 Quetiapine 111974-69-7 Quetiapine is an atypical antipsychotic used in the treatment of schizophrenia, bipolar I mania, bipolar II depression, bipolar I depression.
CSN23099 SB 258585 HCl 1216468-02-8 Potent, selective 5-HT6 antagonist
CSN23130 SR 57227 HCl 77145-61-0 Potent and selective 5-HT3 agonist
CSN23193 WAY 161503 HCl 276695-22-8 Potent and selective 5-HT2C agonist
CSN10104 Pizotifen Malate 5189-11-7 Pizotifen Malate is a benzocycloheptene-based drug used to reduce the frequency of recurrent migraine headacheswith, with high affinity for 5-HT and dopamine receptors (Kis = 7.94 and 2.4 nM for 5-HT2C and D2, respectively).
CSN10097 Naftidrofuryl Oxalate 3200-06-4 Naftidrofuryl oxalate is a drug used in the management of peripheral and cerebral vascular disorders as a vasodilator, enhance cellular oxidative capacity, and may also be a 5-HT2 receptor antagonist.
CSN11473 Mosapride Citrate 112885-42-4 Mosapride Citrate is both a selective 5HT4 agonist and a 5HT3 antagonist, use as a gastroprokinetic agent.
CSN12407 Loxapine 1977-10-2 Loxapine succinate is a D2DR and D4DR inhibitor, serotonergic receptor antagonist and also a dibenzoxazepine anti-psychotic agent.
CSN11251 Ketanserin Tartrate 83846-83-7 Ketanserin Tartrate is a water soluble selective 5-HT2A and 5-HT1D antagonist.
CSN11471 Indeloxazine HCl 65043-22-3 Indeloxazine HCl is an antidepressant and cerebral activator.
CSN21789 Perospirone HCl 3H2O 129273-38-7 In CHO cells expressing human 5-HT1A receptors, perospirone shows a high affinity (Ki = 0.72 nM), and exhibits partial agonistic efficacy.
CSN11188 Iloperidone 133454-47-4 Iloperidone is a D2/5-HT2 receptor antagonist, which is an atypical antipsychotic for the treatment of schizophrenia symptoms.
CSN23084 S 14506 HCl 286369-38-8 Highly potent 5-HT1A agonist; displays unique binding mechanism
CSN23194 WAY 181187 Oxalate 1883548-85-3 High affinity and selective 5-HT6 agonist
CSN14586 Galanolactone 115753-79-2 Galanolactone, a natural product isolated and purified from the rhizomes of Zingiber officinale Roscoe with cytotoxic activity, has anti-5-HT effect, a diterpenoid isolated from ginger, is related to antagonism of 5-HT3 receptors, exerts anti-obesity effect through down regulation of adipogenic transcription factors and adipogenic marker genes, and inhibits nitric oxide production with IC(50) values ranging from 5.5 to 28.5 μM.
CSN11019 Flibanserin 167933-07-5 Flibanserin is a serotonergic antidepressant used to treat hypoactive sexual desire disorder. It is also a P-Glycoprotein Inhibitor.
CSN24769 F-15599   635323-95-4 F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist with Ki value of 3.4nM.
CSN23783 AVN492 1220646-23-0 AVN492 is a selective antagonist of 5-HT6R with Ki of 91 pM.
CSN12463 Aripiprazole 129722-12-9 Aripiprazole is a multiple-target agent used to treat schizophrenia and bipolar disorder, working as both a silent antagonist and a high-efficacy partial agonist of D2 receptor, as well as works as a partial agonist of 5-HT1A/5-HT2A, 5-HT2 receptor,a potent inverse agonist of 5-HT2B receptor, a functional antagonist of 5-HT7 receptor.
CSN24980 5-Methoxytryptamine 608-07-1 5-Methoxytryptamine is a tryptamine derivative that acts as a full agonist at the 5-HT1, 5-HT2, 5-HT4, 5-HT6, and 5-HT7 receptors.
CSN23078 RS 67506 HCl 168986-61-6 5-HT4 partial agonist
CSN23074 RS 23597-190 HCl 149719-06-2 5-HT4 antagonist
CSN23076 RS 39604 HCl 167710-87-4 5-HT4 antagonist
CSN23077 RS 56812 HCl 143339-12-2 5-HT3 partial agonist
CSN23090 SB 200646 HCl 143797-62-0 5-HT2C/2B antagonist
CSN23085 S 32212 HCl 847871-78-7 5-HT2C inverse agonist; α2-adrenoceptor antagonist
CSN23215 α-Methyl-5-hydroxytryptamine Maleate 97469-12-0 5-HT2B agonist
CSN23080 RU 24969 Hemisuccinate 66611-27-6 5-HT1A and 5-HT1B agonist
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