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Neurotensin Receptor

Neurotensin Receptor

货号 产品名 CAS号 信息
CSN20523 SR48692 146362-70-1 SR48692 is an orally available neurotensin antagonist; selective for NTS1 over NTS2 (apparent affinity, Ke, is 36 nM for NTS1), and competitively inhibits binding of [125I]-neurotensin to HT29 and N1E115 cell membranes (IC50 values are 15.3 and 20.4 nM respectively).
CSN20424 PD149163 169528-11-4 PD149163, a neurotensin receptor 1 agonist, decreases methamphetamine self-administration in DBA/2J mice without causing excessive sedation.
CSN17874 ML314 1448895-09-7 ML314 is a potent molecule agonist of NTR1 (EC50 = 1.9 μM) and shows good selectivity against NTR2 and GPR35, but did not stimulate Ca2+ mobilization.
CSN22867 JMV 449 139026-66-7
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