CAS No.: 606101-58-0
MK-0773 Catalog No. CSN18357
Synonyms: PF-05314882
MK-0773, one of selective androgen receptor modulators (SARMs), is a 4-aza-steroid that exhibited tissue selectivity in humans (IC50= 6.6 nM).
| 规格 | 价格 | 促销价格 | 库存 | 数量 |
|---|
400-920-2911
sales@csnpharm.cn
tech@csnpharm.cn
纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 临床研究
NCT号 适应症或疾病 临床期 招募状态 预计完成时间 地点 NCT01017458 Healthy Phase 1 Completed - - NCT00529659 Sarcopenia Phase 2 Completed - - NCT01011725 Osteoporosis Phase 1 Completed - - - 更多
- 参考文献
- [1] Lagojda A, Kuehne D, et al. Identification of selected in vitro generated phase-I metabolites of the steroidal selective androgen receptor modulator MK-0773 for doping control purposes. Eur J Mass Spectrom (Chichester). 2016;22(2):49-59.
- [2] Schmidt A, Kimmel DB, et al. Discovery of the selective androgen receptor modulator MK-0773 using a rational development strategy based on differential transcriptional requirements for androgenic anabolism versus reproductive physiology. J Biol Chem. 2010 May 28;285(22):17054-64.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 606101-58-0 | 储存条件 |
|
|
| 分子式 | C27H34FN5O2 | 运输 | 蓝冰 | |
| 分子量 | 479.59 | 别名 | PF-05314882 |
