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CAS No.: 911295-24-4

MPP 2HCl Catalog No. CSN21407

Synonyms: N/A

Selective, high affinity silent antagonist at ERα receptors. Displays > 200-fold selectivity for ERα over ERβ. Ki values are 2.7 and 1800 nM at ERα and ERβ receptors respectively.

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靶点选择性

生物活性

  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT03411525Health Services Misuse ... more >> Physician's Practice Patterns Guideline Adherence Unnecessary Procedures Health Care Costs Collapse <<Not ApplicableRecruitingMarch 1, 2019United States, Michigan ... more >> IHA Family & Internal Medicine - West Arbor Not yet recruiting Ann Arbor, Michigan, United States, 48103 Contact: Martha Hammond    734-887-4396    martha_hammond@ihacares.com    IHA Internal Medicine - Domino's Farms Not yet recruiting Ann Arbor, Michigan, United States, 48105 Contact: Brett Lamphier    734-995-0303    brett_lamphier@ihacares.com    Michigan Medicine Briarwood Medical Group Not yet recruiting Ann Arbor, Michigan, United States, 48108 Contact: Meghan Moore    734-998-5729    megkatmo@umich.edu    Michigan Medicine East Ann Arbor Health and Geriatrics Center Recruiting Ann Arbor, Michigan, United States, 48109 Contact: Kathie Antieau    734-647-6563    kantieau@umich.edu    University of Michigan Medical School Not yet recruiting Ann Arbor, Michigan, United States, 48109 Contact: Jeffrey T Kullgren, MS, MD, MPH    734-845-3613    jkullgre@umich.edu    Contact: Eve Kerr, MD, MPH    734-845-3504    ekerr@umich.edu    Principal Investigator: Jeffrey T Kullgren, MD, MS, MPH          Sub-Investigator: Jane Forman, ScD, MHS          Principal Investigator: Eve Kerr, MD,MPH          Sub-Investigator: Hyungjin Kim, ScD          Sub-Investigator: Erin Krupka, PhD, MS, MPP          Sub-Investigator: Barbara Soyster, MD          Michigan Medicine Brighton Health Center Not yet recruiting Brighton, Michigan, United States, 48116 Contact: Kristin Lemerand    810-494-2560    kmuzer@umich.edu    IHA Family & Internal Medicine - Cherry Hill Recruiting Canton, Michigan, United States, 48187 Contact: Jody Haney    734-747-6766 ext 18054    martha_hammond@ihacares.com    Michigan Medicine Canton Health Center Not yet recruiting Canton, Michigan, United States, 48187 Contact: Michell Conner    734-844-5391    blancham@med.umich.edu    IHA Internal Medicine - Towsley Not yet recruiting Ypsilanti, Michigan, United States, 48197 Contact: Greg Robinson    734-712-1300    greg_robinson@ihacares.com Collapse <<
    NCT02738450Down SyndromePhase 1RecruitingMarch 2021United States, Arizona ... more >> St. Joseph's Hospital and Medical Center - Barrow Neurology Clinics Recruiting Phoenix, Arizona, United States, 85013 Contact: Sandy Quintanilla    602-406-7054    Sandy.Quintanilla@DignityHealth.org    Principal Investigator: Anna Burke, MD          United States, California UCSD Adult Down Syndrome Program Recruiting La Jolla, California, United States, 92037-1712 Contact: Asmaa Al-hamdani, M.B.Ch.B, MAS    +1(858) 249 2526    aalhamda@ucsd.edu    Principal Investigator: William Mobley, MD          United States, Maryland Johns Hopkins University Active, not recruiting Baltimore, Maryland, United States, 21224 United States, Massachusetts Massachusetts General Hospital Recruiting Boston, Massachusetts, United States, 02114 Contact: Amy Torres, BS    617-726-7927    aetorres@partners.org    Principal Investigator: Brian Skotko, MD, MPP Collapse <<
    NCT02812225Brain Concussion ... more >> Mild Traumatic Brain Injury Collapse <<Not ApplicableRecruitingMarch 2019United States, Massachusetts ... more >> Beth Israel Deconess Medical Center Emergency Medicine Recruiting Boston, Massachusetts, United States, 02215 Contact: Elinita Rosseto    617-754-2334    erosseto@bidmc.harvard.edu    Contact: Ted Raddell    (617) 754-2334       Principal Investigator: Stephen Epstein, MD, MPP          United States, Ohio University of Cincinnati, Department of Emergency Medicine Recruiting Cincinnati, Ohio, United States, 45267-0769 Contact: Christopher Barczak, MT, CCRP    513-558-8091    christopher.barczak@uc.edu    Contact: Cristina Spinner, CCRP    (513) 558-0698    cristina.spinner@uc.edu    Principal Investigator: Natalie Kreitzer, MD          United States, Tennessee Mountain States Health Alliance Recruiting Johnson City, Tennessee, United States, 37604 Contact: Christy Adkins    423-431-5647    adkinsCE2@msha.com    Contact: Nonna Stepanov, MD    (423) 431-5647    StepanovNV@msha.com    Principal Investigator: Tanzid Shams, MD Collapse <<
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实验方案

技术信息

CAS号 911295-24-4 储存条件
分子式 C29H33Cl2N3O3 运输 蓝冰
分子量 542.50 别名 N/A

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