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CAS No.: 1033805-22-9
Synonyms: LX1032;LX1606;Telotristat Ethyl
LX1606 is an orally-delivered inhibitor of tryptophan hydroxylase that reduces serotonin production.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT03453489 | Carcinoid Syndrome ... more >> Metastatic Nonfunctional Well Differentiated Neuroendocrine Neoplasm Collapse << | Phase 2 | Not yet recruiting | January 1, 2019 | United States, Michigan ... more >> Wayne State University/Karmanos Cancer Institute Not yet recruiting Detroit, Michigan, United States, 48201 Contact: Anthony F. Shields 313-576-8735 shieldsa@karmanos.org Principal Investigator: Anthony F. Shields, M.D. PhD. Sub-Investigator: Csaba Juhasz Sub-Investigator: Philip A. Philip, M.D. Sub-Investigator: Anteneh Tesfaye, M.D. Collapse << |
NCT00853047 | Carcinoid Syndrome | Phase 2 | Completed | - | United States, Arkansas ... more >> Hematology Oncology Services of Arkansas Little Rock, Arkansas, United States, 72205 United States, California UCSF Helen Diller Family Comprehensive Cancer Center San Francisco, California, United States, 94115 United States, Indiana St. Francis Medical Group Oncology and Hematology Specialists Indianapolis, Indiana, United States, 46237 United States, Iowa University of Iowa Iowa City, Iowa, United States, 52242 United States, Massachusetts Dana Farber Cancer Institute Boston, Massachusetts, United States, 02115 United States, Nebraska Nebraska Methodist Hospital Omaha, Nebraska, United States, 68114 United States, Texas UT M.D. Anderson Cancer Center Houston, Texas, United States, 77030 Texas Oncology - McAllen McAllen, Texas, United States, 78503 Texas Oncology - Weslaco Weslaco, Texas, United States, 78596 Collapse << |
NCT02683577 | - | - | Completed | - | - |
实验方案
技术信息
CAS号 | 1033805-22-9 | 储存条件 |
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分子式 | C27H26ClF3N6O3 | 运输 | 蓝冰 | |||
分子量 | 574.98 | 别名 | LX1032;LX1606;Telotristat Ethyl;Xermelo | |||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03453489 | Carcinoid Syndrome ... more >> Metastatic Nonfunctional Well Differentiated Neuroendocrine Neoplasm Collapse << | Phase 2 | Not yet recruiting | January 1, 2019 | United States, Michigan ... more >> Wayne State University/Karmanos Cancer Institute Not yet recruiting Detroit, Michigan, United States, 48201 Contact: Anthony F. Shields 313-576-8735 shieldsa@karmanos.org Principal Investigator: Anthony F. Shields, M.D. PhD. Sub-Investigator: Csaba Juhasz Sub-Investigator: Philip A. Philip, M.D. Sub-Investigator: Anteneh Tesfaye, M.D. Collapse << |
NCT00853047 | Carcinoid Syndrome | Phase 2 | Completed | - | United States, Arkansas ... more >> Hematology Oncology Services of Arkansas Little Rock, Arkansas, United States, 72205 United States, California UCSF Helen Diller Family Comprehensive Cancer Center San Francisco, California, United States, 94115 United States, Indiana St. Francis Medical Group Oncology and Hematology Specialists Indianapolis, Indiana, United States, 46237 United States, Iowa University of Iowa Iowa City, Iowa, United States, 52242 United States, Massachusetts Dana Farber Cancer Institute Boston, Massachusetts, United States, 02115 United States, Nebraska Nebraska Methodist Hospital Omaha, Nebraska, United States, 68114 United States, Texas UT M.D. Anderson Cancer Center Houston, Texas, United States, 77030 Texas Oncology - McAllen McAllen, Texas, United States, 78503 Texas Oncology - Weslaco Weslaco, Texas, United States, 78596 Collapse << |
NCT02683577 | - | - | Completed | - | - |
NCT03302845 | Drug-drug Interaction | Phase 1 | Completed | - | United States, Texas ... more >> Covance Clinical Research Unit Dallas, Texas, United States, 75247 Collapse << |
NCT02195635 | Drug Interactions | Phase 1 | Completed | - | United States, Florida ... more >> Lexicon Investigational Site Daytona Beach, Florida, United States, 32117 Collapse << |
NCT02683577 | Hepatic Impairment | Phase 1 | Completed | - | Moldova, Republic of ... more >> ARENSIA Exploratory Medicine Chisinau, Moldova, Republic of, MD-2025 Romania ARENSIA Exploratory Medicine Bucharest, Romania, 050159 Distr Collapse << |
NCT02155205 | QT Interval | Phase 1 | Completed | - | United States, Indiana ... more >> Lexicon Investigational Site Evansville, Indiana, United States, 47710 Collapse << |
NCT02147808 | Drug Interactions | Phase 1 | Completed | - | United States, Wisconsin ... more >> Lexicon Investigational Site Madison, Wisconsin, United States, 53704 Collapse << |
NCT03442725 | Renal Impairment | Phase 1 | Completed | - | Belgium ... more >> A.T.C. s.a., Clinical Pharmacology Unit, CHU Sart-Tilman Liège, Belgium, B-4000 Germany CRS Clinical Research Services Kiel GmbH Kiel, Germany, D-24105 Moldova, Republic of ARENSIA Exploratory Medicine Phase I Unit, Republican Clinical Hospital Chisinau, Moldova, Republic of, MD-2025 Romania ARENSIA Unit in Spitalul de Nefrologie Bucharest, Romania Collapse << |
NCT03423446 | Hepatic Impairment | Phase 1 | Completed | - | United States, Florida ... more >> Lexicon Investigational Site Miami, Florida, United States, 33014 Lexicon Investigational Site Orlando, Florida, United States, 32809 United States, Texas Lexicon Investigational Site San Antonio, Texas, United States, 78215 Collapse << |
NCT02157584 | Healthy | Phase 1 | Completed | - | United States, Wisconsin ... more >> Lexicon Investigational Site Madison, Wisconsin, United States, 53704 Collapse << |
NCT02157558 | Drug Interactions | Phase 1 | Completed | - | United States, Texas ... more >> Lexicon Investigational Site Dallas, Texas, United States, 75247 Collapse << |
NCT03223428 | - | - | Recruiting | December 2021 | United States, North Carolina ... more >> RTI-HS Recruiting Research Triangle Park, North Carolina, United States, 27709 Collapse << |
NCT01104415 | Symptoms of Carcinoid Syndrome | Phase 2 | Completed | - | Germany ... more >> Lexicon Investigational Site Bad Berka, Germany Lexicon Investigational Site Berlin, Germany Lexicon Investigational Site Halle, Germany Lexicon Investigational Site Lubeck, Germany Lexicon Investigational Site Marburg, Germany Lexicon Investigational Site Munich, Germany United Kingdom Lexicon Investigational Site Basingstoke, United Kingdom Lexicon Investigational Site Cambridge, United Kingdom Lexicon Investigational Site London, United Kingdom Lexicon Investigational Site Manchester, United Kingdom Collapse << |
NCT01104415 | - | - | Completed | - | - |
NCT01677910 | Carcinoid Syndrome | Phase 3 | Completed | - | - |
NCT01456052 | - | - | Completed | - | - |
NCT02026063 | Carcinoid Syndrome | Phase 3 | Active, not recruiting | - | - |
NCT01456052 | Ulcerative Colitis | Phase 2 | Completed | - | United States, Arkansas ... more >> Lexicon Investigational Site Little Rock, Arkansas, United States, 72205 United States, California Lexicon Investigational Site Anaheim, California, United States, 92801 Lexicon Investigational Site Santa Monica, California, United States, 90404 United States, New York Lexicon Investigational Site Great Neck, New York, United States, 11021 Lexicon Investigational Site New York, New York, United States, 10017 United States, Oklahoma Lexicon Investigational Site Tulsa, Oklahoma, United States, 74135 United States, Texas Lexicon Investigational Site Houston, Texas, United States, 77030 Lexicon Investigational Site San Antonio, Texas, United States, 78229 United States, Utah Lexicon Investigational Site Ogden, Utah, United States, 84405 Lexicon Investigational Site Sandy City, Utah, United States, 84094 United States, Washington Lexicon Investigational Site Seattle, Washington, United States, 98195 Lithuania Lexicon Investigational Site Kaunas, Lithuania, LT-50009 Lexicon Investigational Site Klaipeda, Lithuania, LT-92288 Lexicon Investigational Site Siauliai, Lithuania, LT-76231 Lexicon Investigational Site Vilnius, Lithuania, LT-03215 Lexicon Investigational Site Vilnius, Lithuania, LT-08661 Poland Lexicon Investigational Site Krakow, Poland, 31531 Lexicon Investigational Site Lodz, Poland, 90302 Lexicon Investigational Site Sopot, Poland, 81756 Lexicon Investigational Site Warszawa, Poland, 03580 Lexicon Investigational Site Wroclaw, Poland, 53025 Lexicon Investigational Site Wroclaw, Poland, 54144 Slovakia Lexicon Investigational Site Nitra, Slovakia, 94901 Lexicon Investigational Site Nove Mesto nad Vahom, Slovakia, 91501 Collapse << |
NCT02063659 | - | - | Completed | - | - |
NCT01932528 | Carcinoid Syndrome | Phase 1 | Completed | - | United Kingdom ... more >> Lexicon Investigational Site Nottingham, United Kingdom, NG11 6JS Collapse << |
NCT01677910 | - | - | Completed | - | - |
NCT02063659 | Carcinoid Syndrome | Phase 3 | Completed | - | - |
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