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| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN18928 | COH29 | 1190932-38-7 | COH29 is a potent ribonucleotide reductase (RNR) inhibitor with anticancer activity with IC50 value of 8 μM in KB cell. |
| CSN18942 | KRIBB11 | 342639-96-7 | KRIBB11 is an inhibitor of heat shock factor (HSF) inhibitor, with IC50 of 1.2 μM. |
| CSN18997 | 6,7-Dimethoxy-N-(2-methyl-4-phenoxyphenyl)quinazolin-4-amine hydrochloride | 2002381-31-7 | APS-2-79 HCl is a KSR (Kinase suppressor of Ras)-dependent MAPK modulator which can stabilize KSR inactive state with an IC50 value of 120 nM, resulting in inhibition of oncogenic Ras signaling, antagonizing the Ras–MAPK pathway. |
| CSN18952 | BI-9564 | 1883429-22-8 | BI-9564 is an inhibitor of BRD9 (IC50 = 75 nM) and BRD7 (IC50 = 3.4 µM). |
| CSN18941 | Apoptozole | 1054543-47-3 | Apoptozole is an inhibitor of heat shock protein 70 (HSP70) and Hsc70. It induces caspase-dependent apoptosis. |
| CSN18947 | SF1670 | 345630-40-2 | SF1670 is a selective PTEN inhibitor with IC50 value of 2 μM. |
| CSN18937 | N-(3-(((2-Hydroxynaphthalen-1-yl)methylene)amino)phenyl)-2-phenylpropanamide | 1105698-15-4 | Salermide, a reverse amide, can act as an inhibitor of sirt, especially of sirt2, with the property of inducing apoptosis of tumor cells. |
| CSN18940 | Sirtuin modulator 1 | 2070015-26-6 | SRT3025 HCl is an orally available sirtuin modulator. |
| CSN18956 | MM-102 TFA | 1883545-52-5 | MM-102 trifluoroacetate is a potent WDR5/mLL interaction inhibitor, achieves IC50 = 2.4 nM with an estimated Ki < 1 nM in WDR5 binding assay, which is > 200 times more potent than the ARA peptide. |
| CSN18970 | 6H05 trifluoroacetate | 2061344-88-3 | 6H05 trifluoroacetate is a selective, and allosteric inhibitor of oncogenic mutant K-Ras (G12C). |
| CSN18953 | GSK6853 | 1910124-24-1 | GSK6853 selectively inhibits the BRPF1 bromodomain with the pKd value of 9.5. |
| CSN18955 | SGC2085 | 1821908-48-8 | SGC2085 is a selectivel and potent CARM1 inhibitor with IC50 value of 50 nM. |
| CSN18935 | Tirbanibulin Mesylate | 1080645-95-9 | KX2-391 mesylate is an inhibitor of Src that targets the peptide substrate site of Src, with GI50 of 9-60 nM in cancer cell lines. |
| CSN19011 | Naquotinib mesylate | 1448237-05-5 | Naquotinib mesylate is a mutant-selective irreversible EGFR inhibitor with IC50 of 70 nM for NCI-H1650 cell growth,inhibits growth of non-small cell lung cancer (NSCLC) cells with EGFR activating and T790M resistance mutations. |
| CSN18950 | E7820 | 289483-69-8 | E7820 is an angiogenesis inhibitor by suppressing integrin a2, a cell adhesion molecule expressed on endothelial cells. |
| CSN18996 | Motixafortide | 664334-36-5 | BKT140 is a CXCR4 antagonist with an IC50 value of ~1 nM. |
| CSN18933 | Soblidotin | 149606-27-9 | Auristatin PE is a synthetic Dolastatin 10 derivative and inhibitor oftubulinpolymerization. |
| CSN18965 | DDP-38003 2HCl | 1831167-98-6 | DDP-38003 2HCl is an orally available inhibitor of histone lysine-specific demethylase 1A (KDM1A/LSD1) with an IC50 of 84 nM. |
| CSN18944 | Debio 0932 | 1061318-81-7 | Debio 0932 is a heat shock protein 90 (HSP90) inhibitor with strong affinity for HSP90 alpha/beta, high oral bioavailability and potent anti-proliferative activity against a broad range of cancer cell lines (with a mean IC50 of 220 nmol/L). |
| CSN18974 | CFMTI | 864864-17-5 | CFMTI is a potent and selective metabotropic glutamate receptor (mGluR)1 allosteric antagonist with IC50 of 2.6 nM. |
| CSN18986 | Amiselimod HCl | 942398-84-7 | Amiselimod HCl is a sphingosine 1-phosphate receptor-1 (S1P1) modulator, designed to reduce the bradycardia effects associated with fingolimod and other S1P receptor modulators. |
| CSN18924 | Ellipticine HCl | 5081-48-1 | Ellipticine HCl is a potent antineoplastic agent and inhibits DNA topoisomerase II activities. |
| CSN18964 | EPZ031686 | 2095161-11-6 | EPZ031686 is a noncompetitive inhibitor for SMYD3 and MEKK2 with a Ki=1.2 nM and 1.1 nM respectively. |
| CSN18987 | ARS-853 | 1629268-00-3 | ARS-853 is an inhibitor of KRAS G12C with IC50 of 2.5 μM. |
| CSN18967 | Ilginatinib maleate | 1354799-87-3 | NS-018 maleate is an ATP-competitive small-molecule inhibitor of JAK2 with IC50 of 470?nM in Ba/F3-JAK2V617F cells . |
| CSN18925 | CCT244747 | 1404095-34-6 | CCT244747 is potent, highly selective, orally active, ATP competitive CHK1 inhibitor with IC50 of 29-170nM. |
| CSN18995 | MK-0812 Succinate | 851916-42-2 | MK-0812 succinate is a potent and selective CCR2 antagonist with low nM affinity for CCR2 on human monocytes. |
| CSN18976 | DFMTI | 864864-86-8 | DFMTI can completely block the rmGlu1 L757V glutamate response. |
| CSN18966 | NVP-BSK805 2HCl | 1942919-79-0 | NVP-BSK805 2HCl is a potent and selective ATP-competitive JAK2 inhibitor with IC50 of 0.5 nM and > 20-fold selectivity towards JAK1, JAK3 and TYK2. |
| CSN18978 | TCS-OX2-29 | 372523-75-6 | TCS-OX2-29 is a potent and selective orexin 2 (OX2) receptor antagonist with IC50 of 40 nM. |
| CSN18934 | PF-2771 | 2070009-55-9 | PF-2771 is a potent, selective CENP-E inhibitor, PF-2771 inhibits CENP-E motor activity with an IC50 of 16.1 ± 1.2 nM. |
| CSN18926 | NU6300 | 2070015-09-5 | NU6300 is the first covalent ATP-competitive CDK2 inhibitor. |
| CSN18927 | ML241 HCl | 2070015-13-1 | ML241 HCl is a potent and selective inhibitors of p97 ATPase with IC50 values of 100 nM. |
| CSN18921 | Pyridostatin HCl | 1781882-65-2 | Pyridostatin HCl is a G-quadruplex-interacting drug which can promote growth arrest in human cancer cells by inducing replication- and transcription-dependent DNA damage. |
| CSN18929 | SJB3-019A | 2070015-29-9 | SJB3-019A is a potent USP1 inhibitor, 5 times more potent than SJB2-043 in promoting ID1 degradation and cytoxicity in K562 cells with IC50 of 0.0781 μM. |
| CSN18930 | THZ1 Hydrochloride | 2070018-35-6 | THZ1 HCl is a selective and potent covalent CDK7 inhibitor with IC50 of 3.2 nM. |
| CSN18932 | BAY1217389 | 1554458-53-5 | BAY1217389 is a potent, and selective inhibitor of the monopolar spindle 1 (MPS1) kinase with an IC50 value less than 10 nM. |
| CSN18943 | PU-H71 HCl | 2095432-24-7 | PU-H71 HCl is a potent Hsp90 inhibitor with IC50 of 50 nM. |
| CSN18954 | MS049 | 1502816-23-0 | MS 049 is a potent, selective, and cell-active dual inhibitor of PRMT4 and PRMT6 with IC 50 of 34 nM and 43 nM respectively. |
| CSN18963 | CBB1003 hydrochloride | 2070015-02-8 | CBB1003 HCl is a histone demethylase LSD1 inhibitor with IC50 of 10.54 μM. |
| CSN18957 | BET-BAY 002 (S enantiomer) | 2070009-49-1 | BET-BAY 002 S-enantiomer is the S-enantiomer of BET-BAY 002. |
| CSN18951 | OSU-T315 | 2070015-22-2 | ILK-IN-2 is a ILK inhibitor. |
| CSN18958 | CARM1-IN-1 HCl | 2070018-31-2 | CARM1-IN-1 HCl is a potent and specific CARM1 (Coactivator-associated arginine methyltransferase 1) inhibitor with IC50 of 8.6 μM and shows very low activity against PRMT1 and SET7 (IC50 > 600 μM). |
| CSN18959 | CBB1007 hydrochloride | 2070014-96-7 | CBB1007 HCl is a cell-permeable amidino-guanidinium compound that acts as a potent, reversible and substrate competitive LSD1 selective inhibitor (IC50 = 5.27 μM for hLSD1). |
| CSN18960 | CBB1007 3HCl | 2070015-03-9 | CBB1007 3HCl is a cell-permeable amidino-guanidinium compound that acts as a potent, reversible and substrate competitive LSD1 selective inhibitor (IC50 = 5.27 μM for hLSD1). |
| CSN19008 | (1S,3R,5R)-PIM447 dihydrochloride | 2096989-57-8 | (1S,3R,5R)-PIM447 2HCl an PIM inhibitor with IC50 values of 0.095 μM for Pim1, 0.522 μM for Pim2 and 0.369 μM for Pim3. |
| CSN19010 | Naquotinib | 1448232-80-1 | Naquotinib is an irreversible mutant EGFR inhibitor with potential antineoplastic activity. |
| CSN18931 | Monastrol | 329689-23-8 | Monastrol is a specific and allosteric inhibitor of mitotic molecular motor kinesin Eg5 with IC50 value of 14 μM. |
