400-920-2911 sales@csnpharm.cn
您的位置 : 首页 / Cell Cycle / HSP / XL888
CAS No.: 1149705-71-4
Synonyms: XL888
XL888 is a specific and ATP-competitive Hsp90 inhibitor with IC50 of 24 nM.
生物活性
靶点 | HSP90 IC50:24nM |
动物研究 | |
剂量 | Mice: 100 mg/kg[2] (p.o.) |
给药途径 | p.o. |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01657591 | Melanoma | Phase 1 | Active, not recruiting | June 2019 | United States, Florida ... more >> H. Lee Moffitt Cancer Center and Research Institute Tampa, Florida, United States, 33612 Collapse << |
NCT00796484 | Cancer | Phase 1 | Terminated(Sponsor decision) | - | United States, Pennsylvania ... more >> Hospital of the University of Pennsylvania Abramson Cancer Center Philadelphia, Pennsylvania, United States, 19104 United States, Texas South Texas Accelerated Research Therapeutics San Antonio, Texas, United States, 78229 Collapse << |
NCT02721459 | Melanoma Skin... more >> Cancer Collapse << | Phase 1 | Active, not recruiting | December 2021 | United States, Florida ... more >> H. Lee Moffitt Cancer Center and Research Institute Tampa, Florida, United States, 33612 Collapse << |
实验方案
技术信息
CAS号 | 1149705-71-4 | 储存条件 |
|
|||||||||
分子式 | C29H37N5O3 | 运输 | 蓝冰 | |||||||||
分子量 | 503.64 | 别名 | XL888 | |||||||||
溶解度 |
|
动物实验配方 |
|
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01657591 | Melanoma | Phase 1 | Active, not recruiting | June 2019 | United States, Florida ... more >> H. Lee Moffitt Cancer Center and Research Institute Tampa, Florida, United States, 33612 Collapse << |
NCT00796484 | Cancer | Phase 1 | Terminated(Sponsor decision) | - | United States, Pennsylvania ... more >> Hospital of the University of Pennsylvania Abramson Cancer Center Philadelphia, Pennsylvania, United States, 19104 United States, Texas South Texas Accelerated Research Therapeutics San Antonio, Texas, United States, 78229 Collapse << |
NCT02721459 | Melanoma Skin... more >> Cancer Collapse << | Phase 1 | Active, not recruiting | December 2021 | United States, Florida ... more >> H. Lee Moffitt Cancer Center and Research Institute Tampa, Florida, United States, 33612 Collapse << |
NCT03095781 | Adenocarcinoma of the Gastroes... more >>ophageal Junction Colorectal Adenocarcinoma Metastatic Pancreatic Adenocarcinoma Non-Resectable Cholangiocarcinoma Non-Resectable Hepatocellular Carcinoma Recurrent Cholangiocarcinoma Recurrent Colorectal Carcinoma Recurrent Gastric Carcinoma Recurrent Hepatocellular Carcinoma Recurrent Pancreatic Carcinoma Recurrent Small Intestinal Carcinoma Small Intestinal Adenocarcinoma Stage III Colorectal Cancer Stage III Gastric Cancer Stage III Hepatocellular Carcinoma Stage III Pancreatic Cancer Stage III Small Intestinal Cancer Stage IIIA Colorectal Cancer Stage IIIA Gastric Cancer Stage IIIA Hepatocellular Carcinoma Stage IIIA Small Intestinal Cancer Stage IIIB Colorectal Cancer Stage IIIB Gastric Cancer Stage IIIB Hepatocellular Carcinoma Stage IIIB Small Intestinal Cancer Stage IIIC Gastric Cancer Stage IV Colorectal Cancer Stage IV Gastric Cancer Stage IV Hepatocellular Carcinoma Stage IV Pancreatic Cancer Stage IV Small Intestinal Cancer Stage IVA Colorectal Cancer Stage IVA Hepatocellular Carcinoma Stage IVA Pancreatic Cancer Stage IVB Colorectal Cancer Stage IVB Hepatocellular Carcinoma Stage IVB Pancreatic Cancer Unresectable Pancreatic Carcinoma Unresectable Small Intestinal Carcinoma Collapse << | Phase 1 | Recruiting | June 2023 | United States, Georgia ... more >> Emory University Hospital Midtown Recruiting Atlanta, Georgia, United States, 30308 Contact: Shabnam Montazeri 404-686-0242 shabnam.montazeri@emory.edu Contact: Swathi Chinaranagari 404-686-0239 swathi.chinaranagari@emory.edu Emory University/Winship Cancer Institute Recruiting Atlanta, Georgia, United States, 30322 Contact: Audrey Atkins 404-778-4389 audrey.m.adkins@emory.edu Contact: Meredith Renfroe 404-778-2670 marenfr@emory.edu Emory Saint Joseph's Hospital Recruiting Atlanta, Georgia, United States, 30342 Contact: Alicia Escobar 678-843-7029 alicia.m.escobar@emory.edu Contact: Krystal Reese 678-843-5911 krystal.reese@emory.edu Collapse << |
靶点 | Description | IC50 |
---|---|---|
HSP90 | IC50:24nM |
联系我们
官方电话:400-920-2911
二维码
微信公众号 CSN官网