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CAS No.: 1702967-37-0

Vipivotide tetraxetan Catalog No. CSN26878

Synonyms: PSMA-617;WHO-11010

PSMA-617, also know as vipivotide tetraxetan. It is a ligand used to make 177Lu-PSMA-617, which is a radioactive molecule to fight cancer. PSMA617 possesses a small peptide, which was designed to target prostate-specific membrane antigen (PSMA). PSMA617 demonstrates high radiolytic stability for at least 72 h. PSMA617 has high inhibition potency (equilibrium dissociation constant Ki=2.34±2.94 nM on LNCaP; Ki=0.37±0.21 nM enzymatically determined). 177 Lu-PSMA-617 offers a potential additional life-prolonging treatment option for men with mCRPC.

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CAS号 1702967-37-0 储存条件
分子式 C49H71N9O16 运输 蓝冰
分子量 1042.14 别名 PSMA-617;WHO-11010

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