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CAS No.: 1702967-37-0
Synonyms: PSMA-617;WHO-11010
PSMA-617, also know as vipivotide tetraxetan. It is a ligand used to make 177Lu-PSMA-617, which is a radioactive molecule to fight cancer. PSMA617 possesses a small peptide, which was designed to target prostate-specific membrane antigen (PSMA). PSMA617 demonstrates high radiolytic stability for at least 72 h. PSMA617 has high inhibition potency (equilibrium dissociation constant Ki=2.34±2.94 nM on LNCaP; Ki=0.37±0.21 nM enzymatically determined). 177 Lu-PSMA-617 offers a potential additional life-prolonging treatment option for men with mCRPC.
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实验方案
技术信息
CAS号 | 1702967-37-0 | 储存条件 |
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分子式 | C49H71N9O16 | 运输 | 蓝冰 | |
分子量 | 1042.14 | 别名 | PSMA-617;WHO-11010 |
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