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CAS No.: 599179-03-0
Synonyms: SCH-417690 maleate;SCH-D maleate;Vicriviroc (maleate)
Vicriviroc maleate is a CCR5 antagonist with IC50 of 0.91 nM in clinical development for the treatment of HIV-1.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00551330 | HIV Infections ... more >> Acquired Immunodeficiency Syndrome Collapse << | Phase 2 | Completed | - | - |
NCT00705419 | - | - | Completed | - | - |
NCT00243230 | HIV Infections | Phase 2 | Completed | - | - |
实验方案
技术信息
CAS号 | 599179-03-0 | 储存条件 |
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分子式 | C32H42F3N5O6 | 运输 | 蓝冰 | |
分子量 | 649.70 | 别名 | SCH-417690 maleate;SCH-D maleate;Vicriviroc (maleate);MK-7690;SCH-417690;SCH-D |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00551330 | HIV Infections ... more >> Acquired Immunodeficiency Syndrome Collapse << | Phase 2 | Completed | - | - |
NCT00705419 | - | - | Completed | - | - |
NCT00243230 | HIV Infections | Phase 2 | Completed | - | - |
NCT00686829 | HIV Infections | Phase 2 | Completed | - | - |
NCT00632073 | HIV Infections | Phase 1 | Completed | - | - |
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