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CAS No.: 136647-02-4
Synonyms: UK-78282 Hydrochloride;UK-78282 HCl
UK-78282 is a blocker of the KV1.3 and KV1.4 voltage-gated potassium channels in T lymphocytes (IC50 values are 0.28 and 0.17 μM respectively) which suppresses T lymphocyte mitogenesis and leads to membrane depolarization and also blocks KV1.4 expressed in heart and brain.
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CAS号 | 136647-02-4 | 储存条件 |
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分子式 | C29H36ClNO2 | 运输 | 蓝冰 | |
分子量 | 466.05 | 别名 | UK-78282 Hydrochloride;UK-78282 HCl |
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