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CAS No.: 851723-84-7
Synonyms: OC000459
OC000459 is a potent and selective D prostanoid receptor 2 (DP2) antagonist with IC50 of 13 nM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00290381 | Allergic Rhinitis | Phase 1 | Completed | - | United Kingdom ... more >> National Heart & Lung Institute Clinical Studies Unit London, United Kingdom, SW3 6HP Collapse << |
NCT02660489 | Asthma Rhinov... more >>irus Picornaviridae Infections Common Cold Collapse << | Phase 2 | Unknown | February 2018 | United Kingdom ... more >> St Mary's Hospital Recruiting London, Greater London, United Kingdom, W2 1PG Contact: Hugo Farne, BMBCh MA 07590 250487 asthma.trial@imperial.ac.uk Contact: Maria-Belén Trujillo-Torralbo, BSc 07590 250487 asthma.trial@imperial.ac.uk Collapse << |
NCT00697281 | Allergic Rhinitis | Phase 2 | Completed | - | Austria ... more >> Allergie Zentrum Wien West, Vienna Challenge Chamber Vienna, Austria, 1150 VIENNA Collapse << |
实验方案
技术信息
CAS号 | 851723-84-7 | 储存条件 |
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分子式 | C21H17FN2O2 | 运输 | 蓝冰 | |||||
分子量 | 348.37 | 别名 | OC000459 | |||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00290381 | Allergic Rhinitis | Phase 1 | Completed | - | United Kingdom ... more >> National Heart & Lung Institute Clinical Studies Unit London, United Kingdom, SW3 6HP Collapse << |
NCT02660489 | Asthma Rhinov... more >>irus Picornaviridae Infections Common Cold Collapse << | Phase 2 | Unknown | February 2018 | United Kingdom ... more >> St Mary's Hospital Recruiting London, Greater London, United Kingdom, W2 1PG Contact: Hugo Farne, BMBCh MA 07590 250487 asthma.trial@imperial.ac.uk Contact: Maria-Belén Trujillo-Torralbo, BSc 07590 250487 asthma.trial@imperial.ac.uk Collapse << |
NCT00697281 | Allergic Rhinitis | Phase 2 | Completed | - | Austria ... more >> Allergie Zentrum Wien West, Vienna Challenge Chamber Vienna, Austria, 1150 VIENNA Collapse << |
NCT00890877 | Mild to Moderate Persistent As... more >>thma Collapse << | Phase 2 | Completed | - | Bulgaria ... more >> Research site Sofia, Bulgaria Hungary Research site Gyor, Hungary Poland Research site Warsaw, Poland Romania Research site Bucharest, Romania Russian Federation Research site Moscow, Russian Federation Ukraine Research site Kiev, Ukraine Collapse << |
NCT01056692 | Bronchial Asthma | Phase 2 | Completed | - | United Kingdom ... more >> King's College London School of Medicine London, United Kingdom, SE5 9PJ Medicines Evaluation Unit Manchester, United Kingdom, M23 9LT Collapse << |
NCT01057927 | Asthma | Phase 2 | Completed | - | Russian Federation ... more >> Sverdlovsk Regional Hospital #1 Ekaterinburg, Russian Federation, 620102 Research Institute of Pulmonology Moscow, Russian Federation, 105077 Burdenko Main Military Hospital Moscow, Russian Federation, 105229 City Hospital #23 Moscow, Russian Federation, 109240 City Hospital #7 Moscow, Russian Federation, 115446 Vishnevsky Central Military Hospital #3 Moscow, Russian Federation, 194354 Leningrad Regional Hospital St Petersbrug, Russian Federation, 194291 St George City Hospital St Petersbrug, Russian Federation, 194354 St Petersburg Medical Academy of Postgraduate Education St Petersburg, Russian Federation, 190068 St Petersburg Medical Academy St Petersburg, Russian Federation, 190068 Outpatient Clinic #94 St Petersburg, Russian Federation, 193231 St Petersbrug Hospital of the Russian Academy of Science St Petersburg, Russian Federation, 194017 Russian Center of Emergency and Radiology Medicine St Petersburg, Russian Federation, 194044 St Petersburg State Pediatrics Academy St Petersburg, Russian Federation, 194100 Central Medical Unit #122 St Petersburg, Russian Federation, 194291 St George City Hospital St Petersburg, Russian Federation, 194354 Collapse << |
NCT02002208 | Atopic Dermatitis | Phase 2 | Completed | - | United Kingdom ... more >> University of Sheffield Sheffield, United Kingdom Collapse << |
NCT01056783 | Eosinophilic Esophagitis | Phase 2 | Completed | - | Switzerland ... more >> Swiss EoE Research Group Olten, Switzerland, CH-4600 Collapse << |
NCT02002208 | - | - | Completed | - | - |
NCT01448902 | Allergic Rhinitis | Phase 2 | Completed | - | Austria ... more >> Vienna Challenge Chamber Vienna, Austria Collapse << |
NCT02341521 | Asthma | Phase 1 | Completed | - | United Kingdom ... more >> Simbec Research Merthyr Tydfil, Wales, United Kingdom, CF48 4DR Collapse << |
NCT01056575 | Healthy Volunteers | Phase 1 | Completed | - | United Kingdom ... more >> Simbec Research Ltd Merthyr Tydfil, United Kingdom, CF48 4DR Collapse << |
NCT02560610 | Severe Eosinophilic Asthma | Phase 2 | Recruiting | June 2018 | United Kingdom ... more >> University of Oxford Recruiting Oxford, Oxfordshire, United Kingdom Contact: Ian Pavord, Professor 01865 612893 ian.pavord@ndm.ox.ac.uk Collapse << |
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