CAS No.: 204519-66-4
Talnetant HCl Catalog No. CSN18094
Synonyms: SB 223412 hydrochloride;SB 223412-A;SB-223412 HCl
Talnetant HCl is a potent and selective NK3 receptor antagonist (ki=1.4 nM, hNK-3-CHO), 100-fold selective for the hNK-3 versus hNK-2 receptor, with no affinity for the hNK-1 at concentrations up to 100 μM.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Houghton LA, Cremonini F, et al. Effect of the NK(3) receptor antagonist, talnetant, on rectal sensory function and compliance in healthy humans. Neurogastroenterol Motil. 2007 Sep;19(9):732-43.
- [2] Giardina GA, Raveglia LF, et al. Discovery of a novel class of selective non-peptide antagonists for the human neurokinin-3 receptor. 2. Identification of (S)-N-(1-phenylpropyl)-3-hydroxy-2-phenylquinoline-4-carboxamide (SB 223412).
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 204519-66-4 | 储存条件 |
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| 分子式 | C25H23ClN2O2 | 运输 | 蓝冰 | |
| 分子量 | 418.92 | 别名 | SB 223412 hydrochloride;SB 223412-A;SB-223412 HCl |
