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CAS No.: 1448584-12-0

S55746 Catalog No. CSN22926

Synonyms: BCL-201;Servier-1

S55746 is a potent and selective inhibitor of the anti-apoptotic protein B-cell lymphoma 2 (Bcl-2), with potential pro-apoptotic and antineoplastic activities.

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纯度 & 质量文件 批次:

靶点选择性

生物活性

  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT02603445Follicular Lymphoma, Mantle Ce... more >>ll Lymphoma Collapse <<Phase 1Completed-United States, New York ... more >> Novartis Investigative Site New York, New York, United States, 10017 United States, Texas Novartis Investigative Site Houston, Texas, United States, 77030 Austria Novartis Investigative Site Salzburg, Austria, 5020 France Novartis Investigative Site Pierre-Benite Cedex, France, 69495 Novartis Investigative Site Toulouse Cedex 9, France, 31059 Germany Novartis Investigative Site Freiburg, Germany, 79106 Novartis Investigative Site Mainz, Germany, 55131 Collapse <<
    NCT02920697Chronic Lymphocytic Leukaemia ... more >>(CLL) B-Cell Non-Hodgkin Lymphoma (NHL) Multiple Myeloma (MM) Collapse <<Phase 1Completed-Australia ... more >> The Alfred Hospital Malignant Haematology & Stem Cell Transplantation Services Melbourne, Australia, 3004 France Hopital Claude Huriez Lille, France CHU de Nantes Nantes, France Centre hospitalier Lyon Sud Pierre-Bénite, France Gustave Roussy Villejuif, France Germany Universitätsklinikum Carl Gustav Carus Dresden, Germany Städtisches Klinikum Schwabing Munich, Germany Universitätsklinikum Ulm Ulm, Germany Hungary National Oncology Institute Budapest, Hungary CRU Hungary Kft Miskolc, Hungary Korea, Republic of Severance Hospital Seoul, Korea, Republic of St. Mary's Hospital Seoul, Korea, Republic of Poland Warsaw Institute of Oncology Warsaw, Poland Warsaw Medical University Warsaw, Poland Singapore National Cancer Center (NCC) Singapore, Singapore National University Cancer Institute Singapore Singapore, Singapore United Kingdom University College London Hospitals London, United Kingdom Freeman Hospital Newcastle, United Kingdom Collapse <<

实验方案

技术信息

CAS号 1448584-12-0 储存条件
分子式 C43H42N4O6 运输 蓝冰
分子量 710.82 别名 BCL-201;Servier-1
溶解度
DMSO30.0 mg/mL (42.2 mM)
Waterinsoluble
动物实验配方

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