400-920-2911 sales@csnpharm.cn
CAS No.: 459868-92-9
Synonyms: AG-014699 phosphate;PF-01367338 phosphate;Rucaparib (phosphate)
Rucaparib phosphate is an inhibitor of PARP with Ki of 1.4 nM for PARP1, also showing binding affinity to eight other PARP domains.
规格 | 价格 | 促销价格 | 库存 | 数量 |
---|
生物活性
靶点 | PARP1 Ki:1.4nM |
动物研究 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
剂量 | Mice: 2 mg/kg - 150 mg/kg[5] (p.o.), 0.05 mg/kg - 10 mg/kg[1] (i.p.) Rat: 15 mg/kg[5] (i.v.) | ||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
给药途径 | p.o., i.p., i.v. | ||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
动物药代数据 |
|
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT03442556 | ATM Gene Mutation ... more >> BRCA1 Gene Mutation BRCA2 Gene Mutation Castration Levels of Testosterone Castration-Resistant Prostate Carcinoma Homologous Recombination Deficiency Prostate Carcinoma Metastatic in the Bone PSA Level Greater Than or Equal to Two PSA Progression Stage IV Prostate Adenocarcinoma AJCC v7 Collapse << | Phase 2 | Recruiting | May 15, 2024 | United States, Washington ... more >> Fred Hutch/University of Washington Cancer Consortium Recruiting Seattle, Washington, United States, 98109 Contact: Heather H. Cheng 206-606-1406 hhcheng@uw.edu Principal Investigator: Heather H. Cheng Collapse << |
NCT03552471 | BRCA1 Gene Mutation ... more >> BRCA2 Gene Mutation Folate Receptor Alpha Positive Recurrent Fallopian Tube Carcinoma Recurrent Ovarian Carcinoma Recurrent Primary Peritoneal Carcinoma Recurrent Uterine Corpus Carcinoma Recurrent Uterine Serous Carcinoma Recurrent Uterine Carcinosarcoma Platinum Resistant Ovarian Cancer Collapse << | Phase 1 | Recruiting | August 29, 2021 | United States, Ohio ... more >> Ohio State University Comprehensive Cancer Center Recruiting Columbus, Ohio, United States, 43210 Contact: Floor Backes, MD 614-293-3873 Principal Investigator: Floor Backes Collapse << |
实验方案
技术信息
CAS号 | 459868-92-9 | 储存条件 |
|
|||||||||||||
分子式 | C19H21FN3O5P | 运输 | 蓝冰 | |||||||||||||
分子量 | 421.36 | 别名 | AG-014699 phosphate;PF-01367338 phosphate;Rucaparib (phosphate);AG-014699;PF-01367338;AG14699 (as phosphate salt);AG-14699;AG014447 (as free base);AG-014447;Rucaparib;Rubraca;瑞卡帕布磷酸盐 | |||||||||||||
溶解度 |
|
动物实验配方 |
|