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CAS No.: 875320-29-9
Synonyms: JNJ-26481585
Quisinostat is an orally available, potent HDAC inhibitor with IC50 values of 0.11 nM for HDAC1.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00677105 | Lymphoma Neop... more >>lasms Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Glasgow, United Kingdom Leeds, United Kingdom London, United Kingdom Manchester, United Kingdom Newcastel Upon Tyne, United Kingdom Sutton, United Kingdom Collapse << |
NCT02728492 | Non-small Cell Lung Cancer ... more >> Epithelial Ovarian Cancer Collapse << | Phase 1 | Completed | - | Russian Federation ... more >> Russian Oncological Research Center n.a. N. N. Blokhin RAMS Moscow, Russian Federation, 115478 State Budgetary Healthcare Institution of Stavropol Territory "Pyatigorsk oncology dispensary" Pyatigorsk, Russian Federation, 357502 Saint-Peterburg State Budgetary healthcare Institution "City Clinical Oncology Dispensary" Saint-Petersburg, Russian Federation, 197022 BioEq LLC Saint-Petersburg, Russian Federation, 197342 State Budget Institution of healthcare "Saint-Petersburg clinical research and practical centre of specialized medical aid (oncology)" Saint-Petersburg, Russian Federation, 197758 State Healthcare Institution of Yaroslavl region "Regional Clinical oncology hospital" Yaroslavl, Russian Federation, 150054 Collapse << |
NCT00676728 | Advanced or Refractory Leukemi... more >>a Myelodysplastic Syndromes Collapse << | Phase 1 | Terminated(Sponsor Decision) | - | United States, Maryland ... more >> Baltimore, Maryland, United States United States, Texas Houston, Texas, United States Collapse << |
实验方案
技术信息
CAS号 | 875320-29-9 | 储存条件 |
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分子式 | C21H26N6O2 | 运输 | 蓝冰 | |
分子量 | 394.47 | 别名 | JNJ-26481585 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00677105 | Lymphoma Neop... more >>lasms Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Glasgow, United Kingdom Leeds, United Kingdom London, United Kingdom Manchester, United Kingdom Newcastel Upon Tyne, United Kingdom Sutton, United Kingdom Collapse << |
NCT02728492 | Non-small Cell Lung Cancer ... more >> Epithelial Ovarian Cancer Collapse << | Phase 1 | Completed | - | Russian Federation ... more >> Russian Oncological Research Center n.a. N. N. Blokhin RAMS Moscow, Russian Federation, 115478 State Budgetary Healthcare Institution of Stavropol Territory "Pyatigorsk oncology dispensary" Pyatigorsk, Russian Federation, 357502 Saint-Peterburg State Budgetary healthcare Institution "City Clinical Oncology Dispensary" Saint-Petersburg, Russian Federation, 197022 BioEq LLC Saint-Petersburg, Russian Federation, 197342 State Budget Institution of healthcare "Saint-Petersburg clinical research and practical centre of specialized medical aid (oncology)" Saint-Petersburg, Russian Federation, 197758 State Healthcare Institution of Yaroslavl region "Regional Clinical oncology hospital" Yaroslavl, Russian Federation, 150054 Collapse << |
NCT00676728 | Advanced or Refractory Leukemi... more >>a Myelodysplastic Syndromes Collapse << | Phase 1 | Terminated(Sponsor Decision) | - | United States, Maryland ... more >> Baltimore, Maryland, United States United States, Texas Houston, Texas, United States Collapse << |
NCT02948075 | Ovarian Cancer | Phase 2 | Completed | - | Russian Federation ... more >> Federal State budget Scientific Agency "Russian Oncological Research Center n.a. N.N. Blokhin" Moscow, Russian Federation, 115478 Medical Radiological Scientific Center n.a. A.F. Tsyb - branch of Federal State Budget Agency "Public Medical Scientific Radiology Center" of Ministry of Health of Russian Federation Obninsk, Russian Federation, 249036 State Budget Agency of Stavropol Territory Healthcare Pyatigorsk Oncologic Dispensary Pyatigorsk, Russian Federation, 357502 State Budget Agency of Healthcare "Leningradsky Regional Oncologic Dispensary" St. Petersburg, Russian Federation, 191014 State Budget Healthcare Agency "St-Petersburg clinical scientific-practical center of specialized types of medical care (oncology)" St. Petersburg, Russian Federation, 197758 St-Petersburg State Budget Agency of Healthcare "Municipal Clinical Oncological Dispensary" St. Petersburg, Russian Federation Collapse << |
NCT01486277 | Lymphoma, T-Cell, Cutaneous | Phase 2 | Completed | - | United States, Pennsylvania ... more >> Pittsburgh, Pennsylvania, United States France Nantes Cedex 1, France Paris, France Pessac, France Germany Kiel, Germany Minden, Germany Portugal Lisboa, Portugal Porto, Portugal Spain Madrid N/A, Spain Málaga, Spain Valencia, Spain United Kingdom London, United Kingdom Manchester, United Kingdom Collapse << |
NCT01464112 | Multiple Myeloma | Phase 1 | Completed | - | France ... more >> Lille Cedex, France Nantes, France Tours, France Collapse << |
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