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CAS No.: 1114544-31-8

Ponatinib HCl Catalog No. CSN21067

Synonyms: AP24534 hydrochloride;Ponatinib HCl;Ponatinib (hydrochloride)

Ponatinib is a multi-targeted kinase inhibitor with IC50 of 0.37 nM, 1.1 nM, 1.5 nM, 2.2 nM, and 5.4 nM for Abl, PDGFRα, VEGFR2, FGFR1, and Src respectively.

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生物活性

  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT02551718Acute Leukemia of Ambiguous Li... more >>neage Recurrent Adult Acute Lymphoblastic Leukemia Recurrent Adult Acute Myeloid Leukemia Recurrent Childhood Acute Lymphoblastic Leukemia Recurrent Childhood Acute Myeloid Leukemia Refractory Acute Myeloid Leukemia Refractory Adult Acute Lymphoblastic Leukemia Refractory Childhood Acute Lymphoblastic Leukemia Collapse <<Not ApplicableRecruiting-United States, Washington ... more >> Fred Hutch/University of Washington Cancer Consortium Recruiting Seattle, Washington, United States, 98109 Contact: Pamela S. Becker    206-616-1589    pbecker@u.washington.edu    Principal Investigator: Pamela S. Becker Collapse <<
    NCT01883219Philadelphia Chromosome Positi... more >>ve Acute Lymphocytic Leukemia Stem Cell Transplantation Minimal Residual Disease Collapse <<Phase 2UnknownNovember 2017China, Guangdong ... more >> Department of Hematology,Nanfang Hospital, Southern Medical University Recruiting Guangzhou, Guangdong, China, 510515 Contact: Ren Lin, MD    +86-020-61641613    lansinglinren@hotmail.com Collapse <<
    NCT03624530Philadelphia Chromosome Positi... more >>ve Acute Lymphocytic Leukemia Tyrosine Kinase Inhibitor Minimal Residual Disease Allogeneic Hematopoietic Stem Cell Transplantation Collapse <<Phase 2 Phase 3RecruitingJuly 2022China, Guangdong ... more >> Department of Hematology,Nanfang Hospital, Southern Medical University Recruiting Guangzhou, Guangdong, China, 510515 Contact: Li Xuan    +86-020-62787883    356135708@qq.com    Principal Investigator: Qifa Liu Collapse <<
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实验方案

技术信息

CAS号 1114544-31-8 储存条件
分子式 C29H28ClF3N6O 运输 蓝冰
分子量 569.02 别名 AP24534 hydrochloride;Ponatinib HCl;Ponatinib (hydrochloride);AP-24534

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