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CAS No.: 1061353-68-1
Synonyms: VS-4718;SR-2516
PND-1186 is a potent FAK inhibitor with IC50 of 1.5 nM.
生物活性
靶点 | FAK IC50:1.5nM |
动物研究 | |
剂量 | Mice: 30 mg/kg, 100 mg/kg[2] (s.c.) |
给药途径 | s.c. |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01849744 | Non Hematologic Cancers ... more >> Metastatic Cancer Collapse << | Phase 1 | Terminated(Sponsor's decision ... more >>to deprioritize the program.) Collapse << | - | United States, Arizona ... more >> HonorHealth Research Institute Scottsdale, Arizona, United States, 85258 United States, California Samuel Oschin Comprehensive Cancer Institute, Cedars-Sinai Medical Center Los Angeles, California, United States, 90048 United States, Florida Florida Cancer Specialists Sarasota, Florida, United States, 34232 United States, Missouri Washington University School of Medicine, Division of Oncology Saint Louis, Missouri, United States, 63110 United States, Tennessee Sarah Cannon Research Institute Nashville, Tennessee, United States, 37203 Collapse << |
NCT02651727 | Pancreatic Cancer | Phase 1 | Terminated(the company's decis... more >>ion to de-prioritize 4718 development) Collapse << | - | United States, Missouri ... more >> Washington University School of Medicine Saint Louis, Missouri, United States, 63110 United States, Pennsylvania Gettysburg Cancer Center Gettysburg, Pennsylvania, United States, 17325 Collapse << |
NCT02215629 | Relapsed or Refractory Acute M... more >>yeloid Leukemia Relapsed or Refractory B-Cell Acute Lymphoblastic Leukemia Collapse << | Phase 1 | Withdrawn | November 2016 | - |
实验方案
技术信息
CAS号 | 1061353-68-1 | 储存条件 |
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分子式 | C25H26F3N5O3 | 运输 | 蓝冰 | |||||||||||||
分子量 | 501.50 | 别名 | VS-4718;SR-2516 | |||||||||||||
溶解度 |
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动物实验配方 |
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NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01849744 | Non Hematologic Cancers ... more >> Metastatic Cancer Collapse << | Phase 1 | Terminated(Sponsor's decision ... more >>to deprioritize the program.) Collapse << | - | United States, Arizona ... more >> HonorHealth Research Institute Scottsdale, Arizona, United States, 85258 United States, California Samuel Oschin Comprehensive Cancer Institute, Cedars-Sinai Medical Center Los Angeles, California, United States, 90048 United States, Florida Florida Cancer Specialists Sarasota, Florida, United States, 34232 United States, Missouri Washington University School of Medicine, Division of Oncology Saint Louis, Missouri, United States, 63110 United States, Tennessee Sarah Cannon Research Institute Nashville, Tennessee, United States, 37203 Collapse << |
NCT02651727 | Pancreatic Cancer | Phase 1 | Terminated(the company's decis... more >>ion to de-prioritize 4718 development) Collapse << | - | United States, Missouri ... more >> Washington University School of Medicine Saint Louis, Missouri, United States, 63110 United States, Pennsylvania Gettysburg Cancer Center Gettysburg, Pennsylvania, United States, 17325 Collapse << |
NCT02215629 | Relapsed or Refractory Acute M... more >>yeloid Leukemia Relapsed or Refractory B-Cell Acute Lymphoblastic Leukemia Collapse << | Phase 1 | Withdrawn | November 2016 | - |
靶点 | Description | IC50 |
---|---|---|
FAK | IC50:1.5nM |
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