400-920-2911 sales@csnpharm.cn
您的位置 : 首页 / Natural Product / Miscellaneous / Plitidepsin
CAS No.: 137219-37-5
Synonyms: Aplidine;Aplidin;dehydrodemnin B. US brand name: Aplidin
Aplidine is a cyclic depsipeptide isolated from the marine tunicate Aplidium albicans. Plitidepsin displays a broad spectrum of antitumor activities, inducing apoptosis by triggering mitochondrial cytochrome c release, initiating the Fas/DC95, JNK pathway and activating caspase 3 activation.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00229203 | Multiple Myeloma | Phase 2 | Completed | - | United States, Massachusetts ... more >> Jerome Lipper Multiple Myeloma Center - Dept of Medical Oncology - Dana Farber Cancer Institute Boston, Massachusetts, United States, 02115 Collapse << |
NCT00229203 | - | - | Completed | - | - |
NCT00884286 | Leukemia Lymp... more >>homa Collapse << | Phase 2 | Completed | - | France ... more >> Centre Hospitalier Lyon Sud Lyon, France, 69495 Hôpital Saint- Louis Paris, France, 75475 Institut Gustave Roussy Villejuif, France, 94805 Italy Istituto di ematologia e oncologia medica "L. e. A. Seragnoli" Bologna, Italy, 40138 Fondazione IRCCS Istituto Nazionale dei Tumori Milano, Italy, 20133 Ospedaliero Universitaria de Modena Modena, Italy, 41100 Peru Instituto Nacional de Enfermedades Neoplásicas (INEN) Surquillo, Lima, Peru, 34 Puerto Rico Hospital Español Auxilio Mutuo de Puerto Rico Inc. San Juan, Puerto Rico, 00919 Spain Hospital Clinico de Barcelona Barcelona, Spain, 08036 Hospital Morales Meseguer Murcia, Spain, 3008 Hospital Universitario de Salamanca Salamanca, Spain, 37707 Switzerland Istituto Oncologico della Svizzera Italiana - Ospedale San Giovanni Bellinzona, Switzerland, CH-6500 Collapse << |
实验方案
技术信息
CAS号 | 137219-37-5 | 储存条件 |
|
|
分子式 | C57H87N7O15 | 运输 | 蓝冰 | |
分子量 | 1110.34 | 别名 | Aplidine;Aplidin;dehydrodemnin B. US brand name: Aplidin;PM90001 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00229203 | Multiple Myeloma | Phase 2 | Completed | - | United States, Massachusetts ... more >> Jerome Lipper Multiple Myeloma Center - Dept of Medical Oncology - Dana Farber Cancer Institute Boston, Massachusetts, United States, 02115 Collapse << |
NCT00229203 | - | - | Completed | - | - |
NCT00884286 | Leukemia Lymp... more >>homa Collapse << | Phase 2 | Completed | - | France ... more >> Centre Hospitalier Lyon Sud Lyon, France, 69495 Hôpital Saint- Louis Paris, France, 75475 Institut Gustave Roussy Villejuif, France, 94805 Italy Istituto di ematologia e oncologia medica "L. e. A. Seragnoli" Bologna, Italy, 40138 Fondazione IRCCS Istituto Nazionale dei Tumori Milano, Italy, 20133 Ospedaliero Universitaria de Modena Modena, Italy, 41100 Peru Instituto Nacional de Enfermedades Neoplásicas (INEN) Surquillo, Lima, Peru, 34 Puerto Rico Hospital Español Auxilio Mutuo de Puerto Rico Inc. San Juan, Puerto Rico, 00919 Spain Hospital Clinico de Barcelona Barcelona, Spain, 08036 Hospital Morales Meseguer Murcia, Spain, 3008 Hospital Universitario de Salamanca Salamanca, Spain, 37707 Switzerland Istituto Oncologico della Svizzera Italiana - Ospedale San Giovanni Bellinzona, Switzerland, CH-6500 Collapse << |
NCT00780143 | Relapsed/Refractory Leukemia | Phase 1 Phase 2 | Terminated(Poor recruitment) | - | United States, New Jersey ... more >> The Cancer Institute of New Jersey New Brunswick, New Jersey, United States, 08901 Collapse << |
NCT01149681 | Myelofibrosis | Phase 2 | Completed | - | United States, Minnesota ... more >> Mayo Clinic Rochester, Minnesota, United States, 55905 Italy Azienda Ospedaliero Universitaria Careggi di Firenze Firenze, Italy, 50134 Collapse << |
NCT00780975 | Prostate Cancer | Phase 2 | Terminated(Poor recruitment) | - | United States, Michigan ... more >> University of Michigan Comprehensive Cancer Center Ann Arbor, Michigan, United States, 48109-0473 United States, Washington Seattle Cancer Care Alliance Seattle, Washington, United States, 98109 Collapse << |
NCT00884286 | - | - | Completed | - | - |
NCT00780143 | - | - | Terminated(Poor recruitment) | - | - |
NCT00788099 | Advanced Solid Tumors ... more >> Lymphomas Collapse << | Phase 1 | Completed | - | United States, New Jersey ... more >> The Cancer Institute of New Jersey (CINJ) New Brunswick, New Jersey, United States, 08901 France Institut Gustave Roussy Villejuif, France, 94800 Collapse << |
NCT03117361 | Multiple Myeloma | Phase 2 | Terminated(PharmaMar has decid... more >>ed to end this study due to the slow recruitment rate of the trial) Collapse << | - | France ... more >> CHRU de Lille - Hôpital Claude Huriez Lille, France, 59037 Institut Gustave Roussy Villejuif, France, 94800 Italy Policlinico Vittorio Emanuele Hospital Catania, Italy, 95123 Istituto Scientifico Romagnolo per lo Studio e la Cura dei Tumori Meldola, Italy, 47014 Azienda Ospedaliera Città della Salute e della Scienza di Torino Torino, Italy, 00126 Spain Hospital Universitario Germans Trias i Pujol Badalona, Barcelona, Spain, 08916 Clinica Universidad de Navarra Pamplona, Navarra, Spain, 31008 Institut Català d´Oncologia Girona Girona, Spain, 17007 Institut Català d´Oncologia L´Hospitalet Hospitalet de Llobregat, Spain, 08908 Hospital General Universitario J.M. Morales Meseguer Murcia, Spain, 30008 Hospital Universitario de Salamanca Salamanca, Spain, 37007 Complexo Hospitalario Universitario de Santiago Santiago De Compostela, Spain, 15706 Complejo Hospitalario Regional Virgen Del Rocio Sevilla, Spain, 41013 Collapse << |
NCT01102426 | Relapsed/Refractory Multiple M... more >>yeloma Collapse << | Phase 3 | Completed | - | - |
NCT02100657 | Multiple Myeloma | Phase 1 | Completed | - | France ... more >> Institut Gustave Roussy Villejuif, France, 94805 Spain Hospital Universitario Germans Trias I Pujol Badalona, Barcelona, Spain, 08916 Clínica Universidad de Navarra Pamplona, Navarra, Spain, 31008 MD Anderson Cancer Center Madrid Madrid, Spain, 28033 Hospital Universitario Salamanca Salamanca, Spain, 37007 Hospital Universitario Virgen del Rocío Sevilla, Spain, 41013 Hospital Universitari i Politècnic la Fe Valencia, Spain, 46026 Collapse << |
NCT01876043 | Adult Patients With Unresectab... more >>le Locally Advanced or Metastatic, Relapsed/Refractory Dedifferentiated Liposarcoma Collapse << | Phase 2 | Terminated | December 2015 | France ... more >> Centre Oscar Lambret Lille, France, 59020 Centre Léon Bérard Lyon, France, 69373 Hôpital de la Timone Marseille, France, 13385 Institut Curie Paris, France, 75005 Institut Claudius Regaud Toulouse, France, 31052 Institut Gustave Roussy Villejuif, France, 94800 Collapse << |
NCT03070964 | Lymphoma | Phase 2 | Terminated(The main reason tha... more >>t motivated the study termination was the slow recruitment of the trial.) Collapse << | - | United States, Illinois ... more >> Northwestern University Medical School Chicago, Illinois, United States, 60611 United States, Washington Fred Hutchinson Cancer Research Center Seattle, Washington, United States, 98109 Czechia Faculty Hospital Ostrava Ostrava, Czechia, 708 52 Fakultni Nemocnice Praha Praha, Czechia, 100 34 Italy Ospedale Clinico Aviano Aviano, Pordenone, Italy, 33081 Instituto di Ematologia "Seragnoli" Bologna, Italy, 40138 Spedali Civili di Brescia Brescia, Italy, 25123 Azienda Ospedaliera Universitaria Careggi Firenze, Italy, 50134 Spain Hospital Clínic i Provincial de Barcelona Barcelona, Spain, 08036 Hospital Universitari Vall d'Hebron Barcelona, Spain, 119 - 129 Centro Oncológico MD Anderson International España Madrid, Spain, 28033 Hospital Universitario 12 de Octubre Madrid, Spain, 28041 Hospital Universitario La Paz Madrid, Spain, 28046 Hospital Universitari Son Espases Palma de Mallorca, Spain, 07010 Hospital Universitario de Salamanca Salamanca, Spain, 37007 Hospital Universitario Marqués de Valdecilla Santander, Spain, 39008 Hospital Virgen del Rocío Sevilla, Spain, 41013 Collapse << |
联系我们
官方电话:400-920-2911
二维码
微信公众号 CSN官网