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CAS No.: 1260533-36-5

Pimitespib Catalog No. CSN22232

Synonyms: TAS-116

TAS-116 is a potent and selective HSP90α/β inhibitor with Kis of 34.7 nM, 21.3 nM, respectively.

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靶点选择性

生物活性

  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT02965885Advanced Solid TumorsPhase 1RecruitingMarch 2020United States, Ohio ... more >> Gabrail Cancer Center Recruiting Canton, Ohio, United States, 44718 University Hospitals Case Medical Center Recruiting Cleveland, Ohio, United States, 44106 United States, South Carolina Greenville Health System, Institute for Translational Oncology Research Recruiting Greenville, South Carolina, United States, 29605 United States, Virginia US Oncology - Virginia Cancer Specialists, P.C. Recruiting Fairfax, Virginia, United States, 86885 Italy Policlinico S.Orsola-Malpighi, U.O. Oncologia Medica Recruiting Bologna, Italy, 40138 Contact: Stefania Salvagni    0039 0512142204    stefania.salvagni@aosp.bo.it    Azienda Ospedaliero-Universitaria Policlinico-Vittorio Emanuele Oncologia Medica Recruiting Catania, Italy, 95123 Contact: Soto Parra    0039 0953782426    hsotoparra@policlinico.unict.it    Contact       hsotoparra@yahoo.it    Istituto Europeo di Oncologia , Sviluppo di Nuovi Farmaci per Terapie Innovative Recruiting Milano, Italy, 20141 Contact: Giuseppe Curigliano    0039 0257489439    giuseppe.curigliano@ieo.it    Regina Elena National Cancer Institute Not yet recruiting Roma, Italy, 00144 Contact: Francesco Cognetti    0039 0652666919    francesco.cognetti@ifo.gov.it    United Kingdom Northern Centre for Cancer Care Recruiting Newcastle Upon Tyne, England, United Kingdom Contact: Ruth Plummer    +44 (0) 191 208 4414    Ruth.Plummer@newcastle.ac.uk    Division of Cancer Studies, Kings College London Recruiting London, United Kingdom, SE19 9RT Sarah Cannon Research Institute UK Recruiting London, United Kingdom, W1G 6AD The Christie NHS Foundation Trust Institute of Cancer Sciences, University of Manchester Recruiting Manchester, United Kingdom, M20 4BX Royal Marsden Recruiting Sutton, United Kingdom, SM2 5PTT Collapse <<

实验方案

技术信息

CAS号 1260533-36-5 储存条件
分子式 C25H26N8O 运输 蓝冰
分子量 454.53 别名 TAS-116

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