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CAS No.: 870653-45-5
Synonyms: 5-(4-Phenoxybutoxy)psoralen;SPS-4251;AS-77
PAP-1 is a selective inhibitor of Kv1.3, voltage-gated K+ channel, it potently inhibits human T effector memory cell proliferation with EC50 of 2 nM and delayed hypersensitivity.
生物活性
靶点 | Potassium Channel KV1.3 EC50:2nM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01349920 | - | - | Completed | - | - |
NCT00564109 | - | - | Unknown | - | Switzerland ... more >> Recruiting Zurich, Switzerland Collapse << |
NCT01258179 | - | - | Terminated(low recruitment) | - | Switzerland ... more >> Department of Visceral and Transplantation Surgery Zurich, CH/Zürich, Switzerland, 8091 Collapse << |
实验方案
技术信息
CAS号 | 870653-45-5 | 储存条件 |
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分子式 | C21H18O5 | 运输 | 蓝冰 | |||||
分子量 | 350.36 | 别名 | 5-(4-Phenoxybutoxy)psoralen;SPS-4251;AS-77 | |||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01349920 | - | - | Completed | - | - |
NCT00564109 | - | - | Unknown | - | Switzerland ... more >> Recruiting Zurich, Switzerland Collapse << |
NCT01258179 | - | - | Terminated(low recruitment) | - | Switzerland ... more >> Department of Visceral and Transplantation Surgery Zurich, CH/Zürich, Switzerland, 8091 Collapse << |
NCT01349920 | - | - | Completed | - | - |
NCT02329171 | Cervical Intraepithelial Neopl... more >>asia Collapse << | Phase 3 | Terminated(Insufficient number... more >> of participants.) Collapse << | - | Netherlands ... more >> Maastricht University Medical Centre Maastricht, Netherlands, 6202AZ Collapse << |
NCT01638611 | Healthy | Phase 1 | Completed | - | United States, Nebraska ... more >> Celerion Lincoln, Nebraska, United States, 68502 Collapse << |
靶点 | Description | IC50 |
---|---|---|
Potassium Channel KV1.3 | EC50:2nM |
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