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CAS No.: 1086062-66-9
Synonyms: GSK458;GSK 212;GSK2126458
GSK2126458 is a highly selective and potent inhibitor of PI3K with Ki of 0.019 nM/0.13 nM/0.024 nM/0.06 nM and 0.18 nM/0.3 nM for p110α/β/δ/γ, mTORC1/2 , respectively.
规格 | 价格 | 促销价格 | 库存 | 数量 |
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生物活性
靶点 | mTORC1 Ki:0.18nM | mTORC2 Ki:0.3nM | p110α Ki:0.019nM | p110β Ki:0.13nM | p110γ Ki:0.06nM | 更多 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01725139 | Idiopathic Pulmonary Fibrosis | Phase 1 | Completed | - | United Kingdom ... more >> GSK Investigational Site London, United Kingdom, SW3 6NP Collapse << |
NCT00972686 | Solid Tumours | Phase 1 | Completed | - | United States, California ... more >> GSK Investigational Site San Francisco, California, United States, 94115 United States, New Jersey GSK Investigational Site New Brunswick, New Jersey, United States, 08901 United States, North Carolina GSK Investigational Site Chapel Hill, North Carolina, United States, 27599-7600 United States, Texas GSK Investigational Site Dallas, Texas, United States, 75246 GSK Investigational Site Houston, Texas, United States, 77030 United States, Utah GSK Investigational Site Salt Lake City, Utah, United States, 84112-5550 United States, Washington GSK Investigational Site Seattle, Washington, United States, 98109 Netherlands GSK Investigational Site Amsterdam, Netherlands, 1066 CX GSK Investigational Site Utrecht, Netherlands, 3584 CX Collapse << |
NCT01248858 | Cancer | Phase 1 | Terminated(The reason for term... more >>ination was lack of tolerability and efficacy of the combination treatment) Collapse << | - | United States, North Carolina ... more >> GSK Investigational Site Chapel Hill, North Carolina, United States, 27599-7305 United States, Tennessee GSK Investigational Site Nashville, Tennessee, United States, 37203 Canada, Ontario GSK Investigational Site Toronto, Ontario, Canada, M5G 2M9 Italy GSK Investigational Site Milano, Lombardia, Italy, 20132 Collapse << |
实验方案
技术信息
CAS号 | 1086062-66-9 | 储存条件 |
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分子式 | C25H17F2N5O3S | 运输 | 蓝冰 | |||||||||||||
分子量 | 505.50 | 别名 | GSK458;GSK 212;GSK2126458 | |||||||||||||
溶解度 |
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动物实验配方 |
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