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CAS No.: 934343-74-5
Synonyms: HSP-990
NVP-HSP990 is a potent and selective HSP90 inhibitor for HSP90α/β with IC50 of 0.6 nM/0.8 nM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00879905 | Advanced Solid Malignancies | Phase 1 | Completed | - | Canada, Ontario ... more >> Novartis Investigative Site Toronto, Ontario, Canada, M5G 2M9 France Novartis Investigative Site Toulouse Cedex 3, France, 31052 Spain Novartis Investigative Site Barcelona, Cataluña, Spain, 08035 Collapse << |
NCT01064089 | Advanced Solid Tumors | Phase 1 | Terminated | - | Japan ... more >> Novartis Investigative Site Nagoya, Aichi, Japan, 466-8560 Novartis Investigative Site Kashiwa, Chiba, Japan, 277-8577 Collapse << |
实验方案
技术信息
CAS号 | 934343-74-5 | 储存条件 |
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分子式 | C20H18FN5O2 | 运输 | 蓝冰 | |||||
分子量 | 379.39 | 别名 | HSP-990 | |||||
溶解度 |
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动物实验配方 |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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human A2058 cells | - | Cytotoxicity assay | - | Cytotoxicity against human A2058 cells in presence of HSF1 knock down treatment, IC50=0.0052 μM | 26164188 |
human A375 cells | - | Cytotoxicity assay | - | Cytotoxicity against human A375 cells in presence of HSF1 knock down treatment, IC50=0.006 μM | 26164188 |
human GTL16 cells | - | Cytotoxicity assay | 72 h | Cytotoxicity against human GTL16 cells after 72 hrs by CellTitre-Glo assay, IC50=0.014 μM | 25368984 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00879905 | Advanced Solid Malignancies | Phase 1 | Completed | - | Canada, Ontario ... more >> Novartis Investigative Site Toronto, Ontario, Canada, M5G 2M9 France Novartis Investigative Site Toulouse Cedex 3, France, 31052 Spain Novartis Investigative Site Barcelona, Cataluña, Spain, 08035 Collapse << |
NCT01064089 | Advanced Solid Tumors | Phase 1 | Terminated | - | Japan ... more >> Novartis Investigative Site Nagoya, Aichi, Japan, 466-8560 Novartis Investigative Site Kashiwa, Chiba, Japan, 277-8577 Collapse << |
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